Conejo-Garcia A - Search Results

1

The inhibition of factor inhibiting hypoxia-inducible factor (FIH) by beta-oxocarboxylic acids.

Banerji B, Conejo-Garcia A, McNeill LA, McDonough MA, Buck MR, Hewitson KS, Oldham NJ, Schofield CJ. Banerji B, et al. Chem Commun (Camb). 2005 Nov 21;(43):5438-40. doi: 10.1039/b510707e. Epub 2005 Oct 4. Chem Commun (Camb). 2005. PMID: 16261239

2

A prodrug system for hydroxylamines based on esterase catalysis.

Conejo-Garcia A, Schofield CJ. Conejo-Garcia A, et al. Bioorg Med Chem Lett. 2005 Sep 15;15(18):4004-9. doi: 10.1016/j.bmcl.2005.06.026. Bioorg Med Chem Lett. 2005. PMID: 15990293

3

Evaluation of aspirin metabolites as inhibitors of hypoxia-inducible factor hydroxylases.

Lienard BM, Conejo-García A, Stolze I, Loenarz C, Oldham NJ, Ratcliffe PJ, Schofield CJ. Lienard BM, et al. Chem Commun (Camb). 2008 Dec 21;(47):6393-5. doi: 10.1039/b814440k. Epub 2008 Nov 5. Chem Commun (Camb). 2008. PMID: 19048166

4

Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor.

Conejo-Garcia A, McDonough MA, Loenarz C, McNeill LA, Hewitson KS, Ge W, Liénard BM, Schofield CJ, Clifton IJ. Conejo-Garcia A, et al. Bioorg Med Chem Lett. 2010 Oct 15;20(20):6125-8. doi: 10.1016/j.bmcl.2010.08.032. Epub 2010 Aug 10. Bioorg Med Chem Lett. 2010. PMID: 20822901

5

Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases.

Chowdhury R, Candela-Lena JI, Chan MC, Greenald DJ, Yeoh KK, Tian YM, McDonough MA, Tumber A, Rose NR, Conejo-Garcia A, Demetriades M, Mathavan S, Kawamura A, Lee MK, van Eeden F, Pugh CW, Ratcliffe PJ, Schofield CJ. Chowdhury R, et al. ACS Chem Biol. 2013 Jul 19;8(7):1488-96. doi: 10.1021/cb400088q. Epub 2013 Jun 12. ACS Chem Biol. 2013. PMID: 23683440

6

Plasmodium falciparum Choline Kinase Inhibition Leads to a Major Decrease in Phosphatidylethanolamine Causing Parasite Death.

Serrán-Aguilera L, Denton H, Rubio-Ruiz B, López-Gutiérrez B, Entrena A, Izquierdo L, Smith TK, Conejo-García A, Hurtado-Guerrero R. Serrán-Aguilera L, et al. Sci Rep. 2016 Sep 12;6:33189. doi: 10.1038/srep33189. Sci Rep. 2016. PMID: 27616047 Free PMC article.

7

Bispyridinium cyclophanes: novel templates for human choline kinase inhibitors.

Conejo-García A, Campos JM, Sánchez-Martín RM, Gallo MA, Espinosa A. Conejo-García A, et al. J Med Chem. 2003 Aug 14;46(17):3754-7. doi: 10.1021/jm030792i. J Med Chem. 2003. PMID: 12904080

8

Influence of the linker in bispyridium compounds on the inhibition of human choline kinase.

Conejo-García A, Báñez-Coronel M, Sánchez-Martín RM, Rodríguez-González A, Ramos A, Ramírez de Molina A, Espinosa A, Gallo MA, Campos JM, Lacal JC. Conejo-García A, et al. J Med Chem. 2004 Oct 21;47(22):5433-40. doi: 10.1021/jm0496537. J Med Chem. 2004. PMID: 15481981

9

Towards a model for the inhibition of choline kinase by a new type of inhibitor.

Conejo-García A, Entrena A, Campos JM, Sánchez-Martín RM, Gallo MA, Espinosa A. Conejo-García A, et al. Eur J Med Chem. 2005 Mar;40(3):315-9. doi: 10.1016/j.ejmech.2004.09.016. Epub 2004 Nov 11. Eur J Med Chem. 2005. PMID: 15725501

10

Symmetrical bis-quinolinium compounds: new human choline kinase inhibitors with antiproliferative activity against the HT-29 cell line.

Sánchez-Martín R, Campos JM, Conejo-García A, Cruz-López O, Báñez-Coronel M, Rodríguez-González A, Gallo MA, Lacal JC, Espinosa A. Sánchez-Martín R, et al. J Med Chem. 2005 May 5;48(9):3354-63. doi: 10.1021/jm049061o. J Med Chem. 2005. PMID: 15857141

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