Marquez VE - Search Results

1

Human P2Y(6) receptor: molecular modeling leads to the rational design of a novel agonist based on a unique conformational preference.

Costanzi S, Joshi BV, Maddileti S, Mamedova L, Gonzalez-Moa MJ, Marquez VE, Harden TK, Jacobson KA. Costanzi S, et al. Among authors: marquez ve. J Med Chem. 2005 Dec 29;48(26):8108-11. doi: 10.1021/jm050911p. J Med Chem. 2005. PMID: 16366591 Free PMC article.

2

2-Substitution of adenine nucleotide analogues containing a bicyclo[3.1.0]hexane ring system locked in a northern conformation: enhanced potency as P2Y1 receptor antagonists.

Kim HS, Ohno M, Xu B, Kim HO, Choi Y, Ji XD, Maddileti S, Marquez VE, Harden TK, Jacobson KA. Kim HS, et al. Among authors: marquez ve. J Med Chem. 2003 Nov 6;46(23):4974-87. doi: 10.1021/jm030127+. J Med Chem. 2003. PMID: 14584948 Free PMC article.

3

Methanocarba modification of uracil and adenine nucleotides: high potency of Northern ring conformation at P2Y1, P2Y2, P2Y4, and P2Y11 but not P2Y6 receptors.

Kim HS, Ravi RG, Marquez VE, Maddileti S, Wihlborg AK, Erlinge D, Malmsjö M, Boyer JL, Harden TK, Jacobson KA. Kim HS, et al. Among authors: marquez ve. J Med Chem. 2002 Jan 3;45(1):208-18. doi: 10.1021/jm010369e. J Med Chem. 2002. PMID: 11754592 Free PMC article.

4

Synthesis, biological activity, and molecular modeling of ribose-modified deoxyadenosine bisphosphate analogues as P2Y(1) receptor ligands.

Nandanan E, Jang SY, Moro S, Kim HO, Siddiqui MA, Russ P, Marquez VE, Busson R, Herdewijn P, Harden TK, Boyer JL, Jacobson KA. Nandanan E, et al. Among authors: marquez ve. J Med Chem. 2000 Mar 9;43(5):829-42. doi: 10.1021/jm990249v. J Med Chem. 2000. PMID: 10715151 Free PMC article.

5

Ring-Constrained (N)-methanocarba nucleosides as adenosine receptor agonists: independent 5'-uronamide and 2'-deoxy modifications.

Lee K, Ravi G, Ji XD, Marquez VE, Jacobson KA. Lee K, et al. Among authors: marquez ve. Bioorg Med Chem Lett. 2001 May 21;11(10):1333-7. doi: 10.1016/s0960-894x(01)00213-x. Bioorg Med Chem Lett. 2001. PMID: 11392549 Free PMC article.

6

A conformationally locked analogue of the anti-HIV agent stavudine. An important correlation between pseudorotation and maximum amplitude.

Choi Y, George C, Comin MJ, Barchi JJ Jr, Kim HS, Jacobson KA, Balzarini J, Mitsuya H, Boyer PL, Hughes SH, Marquez VE. Choi Y, et al. Among authors: marquez ve. J Med Chem. 2003 Jul 17;46(15):3292-9. doi: 10.1021/jm030116g. J Med Chem. 2003. PMID: 12852759

7

A new synthetic route to (North)-methanocarba nucleosides designed as A3 adenosine receptor agonists.

Joshi BV, Moon HR, Fettinger JC, Marquez VE, Jacobson KA. Joshi BV, et al. Among authors: marquez ve. J Org Chem. 2005 Jan 21;70(2):439-47. doi: 10.1021/jo0487606. J Org Chem. 2005. PMID: 15651784

8

Methanocarba analogues of purine nucleosides as potent and selective adenosine receptor agonists.

Jacobson KA, Ji X, Li AH, Melman N, Siddiqui MA, Shin KJ, Marquez VE, Ravi RG. Jacobson KA, et al. Among authors: marquez ve. J Med Chem. 2000 Jun 1;43(11):2196-203. doi: 10.1021/jm9905965. J Med Chem. 2000. PMID: 10841798 Free PMC article.

9

Synthesis and purine receptor affinity of 6-oxopurine nucleosides and nucleotides containing (N)-methanocarba-pseudoribose rings.

Ravi G, Lee K, Ji X, Kim HS, Soltysiak KA, Marquez VE, Jacobson KA. Ravi G, et al. Among authors: marquez ve. Bioorg Med Chem Lett. 2001 Sep 3;11(17):2295-300. doi: 10.1016/s0960-894x(01)00450-4. Bioorg Med Chem Lett. 2001. PMID: 11527718 Free PMC article.

10

Synthesis of enantiomerically pure (S)-methanocarbaribo uracil nucleoside derivatives for use as antiviral agents and P2Y receptor ligands.

Melman A, Zhong M, Marquez VE, Jacobson KA. Melman A, et al. Among authors: marquez ve. J Org Chem. 2008 Oct 17;73(20):8085-8. doi: 10.1021/jo801224j. Epub 2008 Sep 24. J Org Chem. 2008. PMID: 18811198 Free PMC article.

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