Werbovetz K - Search Results

1

A thalidomide analogue with in vitro antiproliferative, antimitotic, and microtubule-stabilizing activities.

Li PK, Pandit B, Sackett DL, Hu Z, Zink J, Zhi J, Freeman D, Robey RW, Werbovetz K, Lewis A, Li C. Li PK, et al. Among authors: werbovetz k. Mol Cancer Ther. 2006 Feb;5(2):450-6. doi: 10.1158/1535-7163.MCT-05-0254. Mol Cancer Ther. 2006. PMID: 16505120

2

Purification, characterization, and drug susceptibility of tubulin from Leishmania.

Werbovetz KA, Brendle JJ, Sackett DL. Werbovetz KA, et al. Mol Biochem Parasitol. 1999 Jan 5;98(1):53-65. doi: 10.1016/s0166-6851(98)00146-7. Mol Biochem Parasitol. 1999. PMID: 10029309

3

Selective antimicrotubule activity of N1-phenyl-3,5-dinitro-N4,N4-di-n-propylsulfanilamide (GB-II-5) against kinetoplastid parasites.

Werbovetz KA, Sackett DL, Delfín D, Bhattacharya G, Salem M, Obrzut T, Rattendi D, Bacchi C. Werbovetz KA, et al. Mol Pharmacol. 2003 Dec;64(6):1325-33. doi: 10.1124/mol.64.6.1325. Mol Pharmacol. 2003. PMID: 14645662

4

Synthesis and antitubulin activity of N1- and N4-substituted 3,5-dinitro sulfanilamides against African trypanosomes and Leishmania.

Bhattacharya G, Herman J, Delfín D, Salem MM, Barszcz T, Mollet M, Riccio G, Brun R, Werbovetz KA. Bhattacharya G, et al. J Med Chem. 2004 Mar 25;47(7):1823-32. doi: 10.1021/jm0304461. J Med Chem. 2004. PMID: 15027874

5

Conformationally restricted analogs of Combretastatin A-4 derived from SU5416.

Li PK, Xiao Z, Hu Z, Pandit B, Sun Y, Sackett DL, Werbovetz K, Lewis A, Johnsamuel J. Li PK, et al. Among authors: werbovetz k. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5382-5. doi: 10.1016/j.bmcl.2005.09.001. Epub 2005 Oct 6. Bioorg Med Chem Lett. 2005. PMID: 16213720

6

Antikinetoplastid antimitotic activity and metabolic stability of dinitroaniline sulfonamides and benzamides.

George TG, Johnsamuel J, Delfín DA, Yakovich A, Mukherjee M, Phelps MA, Dalton JT, Sackett DL, Kaiser M, Brun R, Werbovetz KA. George TG, et al. Bioorg Med Chem. 2006 Aug 15;14(16):5699-710. doi: 10.1016/j.bmc.2006.04.017. Epub 2006 May 3. Bioorg Med Chem. 2006. PMID: 16675220

7

Leishmania tarentolae: purification and characterization of tubulin and its suitability for antileishmanial drug screening.

Yakovich AJ, Ragone FL, Alfonzo JD, Sackett DL, Werbovetz KA. Yakovich AJ, et al. Exp Parasitol. 2006 Dec;114(4):289-96. doi: 10.1016/j.exppara.2006.04.008. Epub 2006 Jun 5. Exp Parasitol. 2006. PMID: 16753146 Free PMC article.

8

Synthesis, biological evaluation, and molecular modeling of 3,5-substituted-N1-phenyl-N4,N4-di-n-butylsulfanilamides as antikinetoplastid antimicrotubule agents.

George TG, Endeshaw MM, Morgan RE, Mahasenan KV, Delfín DA, Mukherjee MS, Yakovich AJ, Fotie J, Li C, Werbovetz KA. George TG, et al. Bioorg Med Chem. 2007 Sep 15;15(18):6071-9. doi: 10.1016/j.bmc.2007.06.042. Epub 2007 Jun 27. Bioorg Med Chem. 2007. PMID: 17618122 Free PMC article.

9

Inhibitors of tubulin assembly identified through screening a compound library.

Morgan RE, Ahn S, Nzimiro S, Fotie J, Phelps MA, Cotrill J, Yakovich AJ, Sackett DL, Dalton JT, Werbovetz KA. Morgan RE, et al. Chem Biol Drug Des. 2008 Dec;72(6):513-24. doi: 10.1111/j.1747-0285.2008.00729.x. Chem Biol Drug Des. 2008. PMID: 19090918 Free PMC article.

10

Antitrypanosomal activity of 1,2-dihydroquinolin-6-ols and their ester derivatives.

Fotie J, Kaiser M, Delfín DA, Manley J, Reid CS, Paris JM, Wenzler T, Maes L, Mahasenan KV, Li C, Werbovetz KA. Fotie J, et al. J Med Chem. 2010 Feb 11;53(3):966-82. doi: 10.1021/jm900723w. J Med Chem. 2010. PMID: 20047276

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