Qiang L - Search Results

1

Synthesis and structure-activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonists.

Wu WL, Burnett DA, Spring R, Qiang L, Sasikumar TK, Domalski MS, Greenlee WJ, O'Neill K, Hawes BE. Wu WL, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3668-73. doi: 10.1016/j.bmcl.2006.04.061. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16690312

2

Tetrahydroisoquinolines as MCH-R1 antagonists.

Sasikumar TK, Qiang L, Wu WL, Burnett DA, Greenlee WJ, O'Neill K, Hawes BE, van Heek M, Graziano M. Sasikumar TK, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4917-21. doi: 10.1016/j.bmcl.2006.06.055. Epub 2006 Jul 7. Bioorg Med Chem Lett. 2006. PMID: 16824753

3

Novel aminobenzimidazoles as selective MCH-R1 antagonists for the treatment of metabolic diseases.

Sasikumar TK, Qiang L, Burnett DA, Greenlee WJ, Hawes BE, Kowalski TJ, O'Neill K, Spar BD, Weig B. Sasikumar TK, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2006 Oct 15;16(20):5427-31. doi: 10.1016/j.bmcl.2006.07.058. Epub 2006 Aug 2. Bioorg Med Chem Lett. 2006. PMID: 16889961

4

Tricyclic thienopyridine-pyrimidones/thienopyrimidine-pyrimidones as orally efficacious mGluR1 antagonists for neuropathic pain.

Sasikumar TK, Qiang L, Burnett DA, Greenlee WJ, Li C, Heimark L, Pramanik B, Grilli M, Bertorelli R, Lozza G, Reggiani A. Sasikumar TK, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2009 Jun 15;19(12):3199-203. doi: 10.1016/j.bmcl.2009.04.104. Epub 2009 May 3. Bioorg Med Chem Lett. 2009. PMID: 19433355

5

Discovery of new SCH 39166 analogs as potent and selective dopamine D1 receptor antagonists.

Qiang L, Sasikumar TK, Burnett DA, Su J, Tang H, Ye Y, Mazzola RD Jr, Zhu Z, McKittrick BA, Greenlee WJ, Fawzi A, Smith M, Zhang H, Lachowicz JE. Qiang L, et al. Bioorg Med Chem Lett. 2010 Feb 1;20(3):836-40. doi: 10.1016/j.bmcl.2009.12.100. Epub 2010 Jan 4. Bioorg Med Chem Lett. 2010. PMID: 20061148

6

Design and synthesis of tricyclic sulfones as gamma-secretase inhibitors with greatly reduced Notch toxicity.

Xu R, Cole D, Asberom T, Bara T, Bennett C, Burnett DA, Clader J, Domalski M, Greenlee W, Hyde L, Josien H, Li H, McBriar M, McKittrick B, McPhail AT, Pissarnitski D, Qiang L, Rajagopalan M, Sasikumar T, Su J, Tang H, Wu WL, Zhang L, Zhao Z. Xu R, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2010 Apr 15;20(8):2591-6. doi: 10.1016/j.bmcl.2010.02.080. Epub 2010 Feb 23. Bioorg Med Chem Lett. 2010. PMID: 20236824

7

A-ring modifications on the triazafluorenone core structure and their mGluR1 antagonist properties.

Sasikumar TK, Qiang L, Burnett DA, Greenlee WJ, Li C, Grilli M, Bertorelli R, Lozza G, Reggiani A. Sasikumar TK, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2010 Apr 15;20(8):2474-7. doi: 10.1016/j.bmcl.2010.03.004. Epub 2010 Mar 10. Bioorg Med Chem Lett. 2010. PMID: 20346665

8

Tricyclic sulfones as orally active gamma-secretase inhibitors: synthesis and structure-activity relationship studies.

Sasikumar TK, Qiang L, Burnett DA, Cole D, Xu R, Li H, Greenlee WJ, Clader J, Zhang L, Hyde L. Sasikumar TK, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2010 Jun 15;20(12):3632-5. doi: 10.1016/j.bmcl.2010.04.104. Epub 2010 May 5. Bioorg Med Chem Lett. 2010. PMID: 20493690

9

Synthesis and SAR development of novel mGluR1 antagonists for the treatment of chronic pain.

Brumfield S, Korakas P, Silverman LS, Tulshian D, Matasi JJ, Qiang L, Bennett CE, Burnett DA, Greenlee WJ, Knutson CE, Wu WL, Sasikumar TK, Domalski M, Bertorelli R, Grilli M, Lozza G, Reggiani A, Li C. Brumfield S, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2012 Dec 1;22(23):7223-6. doi: 10.1016/j.bmcl.2012.09.048. Epub 2012 Oct 2. Bioorg Med Chem Lett. 2012. PMID: 23084894

10

A-ring modification of SCH 900229 and related chromene sulfone γ-secretase inhibitors.

Wu WL, Sasikumar TK, Domalski MS, Qiang L, Burnett DA, Clader J, Greenlee WJ, Chan TM, Lee J, Zhang L. Wu WL, et al. Among authors: qiang l. Bioorg Med Chem Lett. 2013 Feb 1;23(3):850-3. doi: 10.1016/j.bmcl.2012.11.054. Epub 2012 Nov 28. Bioorg Med Chem Lett. 2013. PMID: 23265902

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

518 results

Search Page

Filters