Synthesis, antimalarial activity, and preclinical pharmacology of a novel series of 4'-fluoro and 4'-chloro analogues of amodiaquine. Identification of a suitable "back-up" compound for N-tert-butyl isoquine.
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J Med Chem. 2009 Apr 9;52(7):1828-44. doi: 10.1021/jm8012757.
J Med Chem. 2009.
PMID: 19284751
Free article.