Giardinà D - Search Results

1

Recent advances in alpha1-adrenoreceptor antagonists as pharmacological tools and therapeutic agents.

Rosini M, Bolognesi ML, Giardinà D, Minarini A, Tumiatti V, Melchiorre C. Rosini M, et al. Among authors: giardina d. Curr Top Med Chem. 2007;7(2):147-62. doi: 10.2174/156802607779318244. Curr Top Med Chem. 2007. PMID: 17266603 Review.

2

Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety.

Melchiorre C, Angeli P, Bolognesi ML, Chiarini A, Giardinà D, Gulini U, Leonardi A, Marucci G, Minarini A, Pigini M, Quaglia W, Rosini M, Tumiatti V. Melchiorre C, et al. Among authors: giardina d. Pharm Acta Helv. 2000 Mar;74(2-3):181-90. doi: 10.1016/s0031-6865(99)00049-7. Pharm Acta Helv. 2000. PMID: 10812956 Review. No abstract available.

3

Structure--activity relationships among novel phenoxybenzamine-related beta-chloroethylamines.

Giardinà D, Crucianelli M, Angeli P, Buccioni M, Gulini U, Marucci G, Sagratini G, Melchiorre C. Giardinà D, et al. Bioorg Med Chem. 2002 May;10(5):1291-303. doi: 10.1016/s0968-0896(01)00395-9. Bioorg Med Chem. 2002. PMID: 11886792

4

(+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues.

Marucci G, Angeli P, Buccioni M, Gulini U, Melchiorre C, Sagratini G, Testa R, Giardinà D. Marucci G, et al. Among authors: giardina d. Eur J Pharmacol. 2005 Oct 17;522(1-3):100-7. doi: 10.1016/j.ejphar.2005.08.044. Epub 2005 Oct 6. Eur J Pharmacol. 2005. PMID: 16213480

5

Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.

Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D. Sagratini G, et al. Among authors: giardina d. Bioorg Med Chem. 2007 Mar 15;15(6):2334-45. doi: 10.1016/j.bmc.2007.01.028. Epub 2007 Jan 19. Bioorg Med Chem. 2007. PMID: 17276073

6

Doxazosin-related alpha1-adrenoceptor antagonists with prostate antitumor activity.

Giardinà D, Martarelli D, Sagratini G, Angeli P, Ballinari D, Gulini U, Melchiorre C, Poggesi E, Pompei P. Giardinà D, et al. J Med Chem. 2009 Aug 13;52(15):4951-4. doi: 10.1021/jm8016046. J Med Chem. 2009. PMID: 19719240

7

Synthesis and α1-adrenoceptor antagonist activity of tamsulosin analogues.

Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Poggesi E, Giardinà D. Sagratini G, et al. Among authors: giardina d. Eur J Med Chem. 2010 Dec;45(12):5800-7. doi: 10.1016/j.ejmech.2010.09.042. Epub 2010 Sep 25. Eur J Med Chem. 2010. PMID: 20934789

8

Structure-activity relationships in prazosin-related compounds. Effect of replacing a piperazine ring with an alkanediamine moiety on alpha 1-adrenoreceptor blocking activity.

Giardinà D, Brasili L, Gregori M, Massi M, Picchio MT, Quaglia W, Melchiorre C. Giardinà D, et al. J Med Chem. 1989 Jan;32(1):50-5. doi: 10.1021/jm00121a011. J Med Chem. 1989. PMID: 2562855

9

Structure-activity relationships for prazosin and WB 4101 analogues as alpha 1-adrenoreceptor antagonists.

Giardinà D, Bertini R, Brancia E, Brasili L, Melchiorre C. Giardinà D, et al. J Med Chem. 1985 Sep;28(9):1354-7. doi: 10.1021/jm00147a042. J Med Chem. 1985. PMID: 2863379

10

Structure-activity relationships among benextramine-related tetraamine disulfides. Chain length effect on alpha-adrenoreceptor blocking activity.

Quaglia W, Brasili L, Cristalli G, Giardinà D, Picchio MT, Melchiorre C. Quaglia W, et al. Among authors: giardina d. J Med Chem. 1988 Sep;31(9):1861-6. doi: 10.1021/jm00117a030. J Med Chem. 1988. PMID: 2900899

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