Sauer D - Search Results

1

Discovery of a novel small molecule binding site of human survivin.

Wendt MD, Sun C, Kunzer A, Sauer D, Sarris K, Hoff E, Yu L, Nettesheim DG, Chen J, Jin S, Comess KM, Fan Y, Anderson SN, Isaac B, Olejniczak ET, Hajduk PJ, Rosenberg SH, Elmore SW. Wendt MD, et al. Among authors: sauer d. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3122-9. doi: 10.1016/j.bmcl.2007.03.042. Epub 2007 Mar 16. Bioorg Med Chem Lett. 2007. PMID: 17391963

2

Statistical analysis of the effects of common chemical substituents on ligand potency.

Hajduk PJ, Sauer DR. Hajduk PJ, et al. J Med Chem. 2008 Feb 14;51(3):553-64. doi: 10.1021/jm070838y. Epub 2008 Jan 4. J Med Chem. 2008. PMID: 18173228

3

Utilization of NMR-derived fragment leads in drug design.

Huth JR, Sun C, Sauer DR, Hajduk PJ. Huth JR, et al. Methods Enzymol. 2005;394:549-71. doi: 10.1016/S0076-6879(05)94023-8. Methods Enzymol. 2005. PMID: 15808237

4

Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties.

Bruncko M, McClellan WJ, Wendt MD, Sauer DR, Geyer A, Dalton CR, Kaminski MA, Weitzberg M, Gong J, Dellaria JF, Mantei R, Zhao X, Nienaber VL, Stewart K, Klinghofer V, Bouska J, Rockway TW, Giranda VL. Bruncko M, et al. Among authors: sauer dr. Bioorg Med Chem Lett. 2005 Jan 3;15(1):93-8. doi: 10.1016/j.bmcl.2004.10.026. Bioorg Med Chem Lett. 2005. PMID: 15582418

5

Elimination of antibacterial activities of non-peptide luteinizing hormone-releasing hormone (LHRH) antagonists derived from erythromycin A.

Randolph JT, Sauer DR, Haviv F, Nilius AM, Greer J. Randolph JT, et al. Bioorg Med Chem Lett. 2004 Mar 22;14(6):1599-602. doi: 10.1016/j.bmcl.2003.12.059. Bioorg Med Chem Lett. 2004. PMID: 15006412

6

Synthesis and SAR of highly potent and selective dopamine D3-receptor antagonists: variations on the 1H-pyrimidin-2-one theme.

Geneste H, Amberg W, Backfisch G, Beyerbach A, Braje WM, Delzer J, Haupt A, Hutchins CW, King LL, Sauer DR, Unger L, Wernet W. Geneste H, et al. Bioorg Med Chem Lett. 2006 Apr 1;16(7):1934-7. doi: 10.1016/j.bmcl.2005.12.079. Epub 2006 Jan 24. Bioorg Med Chem Lett. 2006. PMID: 16439127

7

Nonpeptide luteinizing hormone-releasing hormone antagonists derived from erythromycin A: design, synthesis, and biological activity of cladinose replacement analogues.

Randolph JT, Waid P, Nichols C, Sauer D, Haviv F, Diaz G, Bammert G, Besecke LM, Segreti JA, Mohning KM, Bush EN, Wegner CD, Greer J. Randolph JT, et al. Among authors: sauer d. J Med Chem. 2004 Feb 26;47(5):1085-97. doi: 10.1021/jm030418i. J Med Chem. 2004. PMID: 14971889

8

Microwave-assisted synthesis utilizing supported reagents: a rapid and efficient acylation procedure.

Sauer DR, Kalvin D, Phelan KM. Sauer DR, et al. Org Lett. 2003 Nov 27;5(24):4721-4. doi: 10.1021/ol0358915. Org Lett. 2003. PMID: 14627424

9

Rapid and efficient synthesis of 1,2,4-oxadiazoles utilizing polymer-supported reagents under microwave heating.

Wang Y, Miller RL, Sauer DR, Djuric SW. Wang Y, et al. Org Lett. 2005 Mar 3;7(5):925-8. doi: 10.1021/ol050007r. Org Lett. 2005. PMID: 15727476

10

Use of polymer-supported Pd reagents for rapid and efficient Suzuki reactions using microwave heating.

Wang Y, Sauer DR. Wang Y, et al. Org Lett. 2004 Aug 5;6(16):2793-6. doi: 10.1021/ol048972p. Org Lett. 2004. PMID: 15281771

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

254 results

Search Page

Filters