DeHaven RN - Search Results

1

Biaryl cannabinoid mimetics--synthesis and structure-activity relationship.

Worm K, Zhou QJ, Stabley GJ, DeHaven RN, Dolle RE. Worm K, et al. Among authors: dehaven rn. Bioorg Med Chem Lett. 2007 Jul 1;17(13):3652-6. doi: 10.1016/j.bmcl.2007.04.059. Epub 2007 Apr 25. Bioorg Med Chem Lett. 2007. PMID: 17507224

2

trans-3,4-dimethyl-4-(3-carboxamidophenyl)piperidines: a novel class of micro-selective opioid antagonists.

Le Bourdonnec B, Belanger S, Cassel JA, Stabley GJ, DeHaven RN, Dolle RE. Le Bourdonnec B, et al. Among authors: dehaven rn. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4459-62. doi: 10.1016/j.bmcl.2003.09.012. Bioorg Med Chem Lett. 2003. PMID: 14643346

3

(4-Carboxamido)phenylalanine is a surrogate for tyrosine in opioid receptor peptide ligands.

Dolle RE, Machaut M, Martinez-Teipel B, Belanger S, Cassel JA, Stabley GJ, Graczyk TM, DeHaven RN. Dolle RE, et al. Among authors: dehaven rn. Bioorg Med Chem Lett. 2004 Jul 5;14(13):3545-8. doi: 10.1016/j.bmcl.2004.04.039. Bioorg Med Chem Lett. 2004. PMID: 15177470

4

Azepinone as a conformational constraint in the design of kappa-opioid receptor agonists.

Tuthill PA, Seida PR, Barker W, Cassel JA, Belanger S, DeHaven RN, Koblish M, Gottshall SL, Little PJ, DeHaven-Hudkins DL, Dolle RE. Tuthill PA, et al. Among authors: dehaven rn, dehaven hudkins dl. Bioorg Med Chem Lett. 2004 Nov 15;14(22):5693-7. doi: 10.1016/j.bmcl.2004.08.041. Bioorg Med Chem Lett. 2004. PMID: 15482950

5

Arylacetamide kappa opioid receptor agonists with reduced cytochrome P450 2D6 inhibitory activity.

Le Bourdonnec B, Ajello CW, Seida PR, Susnow RG, Cassel JA, Belanger S, Stabley GJ, DeHaven RN, DeHaven-Hudkins DL, Dolle RE. Le Bourdonnec B, et al. Among authors: dehaven rn, dehaven hudkins dl. Bioorg Med Chem Lett. 2005 May 16;15(10):2647-52. doi: 10.1016/j.bmcl.2005.03.020. Bioorg Med Chem Lett. 2005. PMID: 15863335

6

Potent and highly selective kappa opioid receptor agonists incorporating chroman- and 2,3-dihydrobenzofuran-based constraints.

Chu GH, Gu M, Cassel JA, Belanger S, Graczyk TM, DeHaven RN, Conway-James N, Koblish M, Little PJ, DeHaven-Hudkins DL, Dolle RE. Chu GH, et al. Among authors: dehaven rn, dehaven hudkins dl. Bioorg Med Chem Lett. 2005 Dec 1;15(23):5114-9. doi: 10.1016/j.bmcl.2005.08.094. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16203140

7

Novel phenylamino acetamide derivatives as potent and selective kappa opioid receptor agonists.

Chu GH, Gu M, Cassel JA, Belanger S, Stabley GJ, DeHaven RN, Conway-James N, Koblish M, Little PJ, DeHaven-Hudkins DL, Dolle RE. Chu GH, et al. Among authors: dehaven rn, dehaven hudkins dl. Bioorg Med Chem Lett. 2006 Feb;16(3):645-8. doi: 10.1016/j.bmcl.2005.10.034. Epub 2005 Nov 2. Bioorg Med Chem Lett. 2006. PMID: 16263278

8

Synthesis and structure-activity relationships of a new series of 2alpha-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as mu-selective opioid antagonists.

Le Bourdonnec B, Goodman AJ, Michaut M, Ye HF, Graczyk TM, Belanger S, DeHaven RN, Dolle RE. Le Bourdonnec B, et al. Among authors: dehaven rn. Bioorg Med Chem Lett. 2006 Feb 15;16(4):864-8. doi: 10.1016/j.bmcl.2005.11.010. Epub 2005 Nov 18. Bioorg Med Chem Lett. 2006. PMID: 16298525

9

Elucidation of the bioactive conformation of the N-substituted trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidine class of mu-opioid receptor antagonists.

Le Bourdonnec B, Goodman AJ, Michaut M, Ye HF, Graczyk TM, Belanger S, Herbertz T, Yap GP, DeHaven RN, Dolle RE. Le Bourdonnec B, et al. Among authors: dehaven rn. J Med Chem. 2006 Dec 14;49(25):7278-89. doi: 10.1021/jm060486f. J Med Chem. 2006. PMID: 17149858

10

Novel malonamide derivatives as potent kappa opioid receptor agonists.

Chu GH, Gu M, Cassel JA, Belanger S, Graczyk TM, DeHaven RN, Conway-James N, Koblish M, Little PJ, DeHaven-Hudkins DL, Dolle RE. Chu GH, et al. Among authors: dehaven rn, dehaven hudkins dl. Bioorg Med Chem Lett. 2007 Apr 1;17(7):1951-5. doi: 10.1016/j.bmcl.2007.01.053. Epub 2007 Jan 25. Bioorg Med Chem Lett. 2007. PMID: 17307360

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