Jacobson KA - Search Results

1

P2Y1 antagonists: combining receptor-based modeling and QSAR for a quantitative prediction of the biological activity based on consensus scoring.

Costanzi S, Tikhonova IG, Ohno M, Roh EJ, Joshi BV, Colson AO, Houston D, Maddileti S, Harden TK, Jacobson KA. Costanzi S, et al. Among authors: jacobson ka. J Med Chem. 2007 Jul 12;50(14):3229-41. doi: 10.1021/jm0700971. Epub 2007 Jun 12. J Med Chem. 2007. PMID: 17564423

2

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

3

Adenosine A1 and A2 receptors: structure--function relationships.

van Galen PJ, Stiles GL, Michaels G, Jacobson KA. van Galen PJ, et al. Among authors: jacobson ka. Med Res Rev. 1992 Sep;12(5):423-71. doi: 10.1002/med.2610120502. Med Res Rev. 1992. PMID: 1513184 Free PMC article. Review. No abstract available.

4

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.

Jacobson KA, van Galen PJ, Williams M. Jacobson KA, et al. J Med Chem. 1992 Feb 7;35(3):407-22. doi: 10.1021/jm00081a001. J Med Chem. 1992. PMID: 1738138 Free PMC article. Review. No abstract available.

5

Functionalized congener approach to muscarinic antagonists: analogues of pirenzepine.

Karton Y, Bradbury BJ, Baumgold J, Paek R, Jacobson KA. Karton Y, et al. Among authors: jacobson ka. J Med Chem. 1991 Jul;34(7):2133-45. doi: 10.1021/jm00111a032. J Med Chem. 1991. PMID: 2066986 Free PMC article.

6

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Jacobson KA, Barone S, Kammula U, Stiles GL. Jacobson KA, et al. J Med Chem. 1989 May;32(5):1043-51. doi: 10.1021/jm00125a019. J Med Chem. 1989. PMID: 2709373 Free PMC article.

7

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

8

Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors.

Siddiqi SM, Jacobson KA, Esker JL, Olah ME, Ji XD, Melman N, Tiwari KN, Secrist JA 3rd, Schneller SW, Cristalli G, et al. Siddiqi SM, et al. Among authors: jacobson ka. J Med Chem. 1995 Mar 31;38(7):1174-88. doi: 10.1021/jm00007a014. J Med Chem. 1995. PMID: 7707320 Free PMC article.

9

Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors.

Jacobson KA, Siddiqi SM, Olah ME, Ji XD, Melman N, Bellamkonda K, Meshulam Y, Stiles GL, Kim HO. Jacobson KA, et al. J Med Chem. 1995 May 12;38(10):1720-35. doi: 10.1021/jm00010a017. J Med Chem. 1995. PMID: 7752196 Free PMC article.

10

Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor.

Kim J, Wess J, van Rhee AM, Schöneberg T, Jacobson KA. Kim J, et al. Among authors: jacobson ka. J Biol Chem. 1995 Jun 9;270(23):13987-97. doi: 10.1074/jbc.270.23.13987. J Biol Chem. 1995. PMID: 7775460 Free PMC article.

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