Grasso S - Search Results

1

Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors.

Ettari R, Nizi E, Di Francesco ME, Dude MA, Pradel G, Vicík R, Schirmeister T, Micale N, Grasso S, Zappalà M. Ettari R, et al. Among authors: grasso s. J Med Chem. 2008 Feb 28;51(4):988-96. doi: 10.1021/jm701141u. Epub 2008 Jan 31. J Med Chem. 2008. PMID: 18232656

2

Novel potent AMPA/kainate receptor antagonists: synthesis and anticonvulsant activity of a series of 2-[(4-alkylsemicarbazono)-(4-amino-phenyl)methyl]-4,5-methylenedioxyphenylacetic acid alkyl esters.

Micale N, Zappalà M, Grasso S, Puja G, De Sarro G, Ferreri G, De Sarro A, Toma L, De Micheli C. Micale N, et al. Among authors: grasso s. J Med Chem. 2002 Sep 26;45(20):4433-42. doi: 10.1021/jm020863y. J Med Chem. 2002. PMID: 12238923

3

1-aryl-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents.

Zappalà M, Grasso S, Micale N, Zuccalà G, Menniti FS, Ferreri G, De Sarro G, De Micheli C. Zappalà M, et al. Among authors: grasso s. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4427-30. doi: 10.1016/j.bmcl.2003.09.032. Bioorg Med Chem Lett. 2003. PMID: 14643339

4

Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents.

Micale N, Kozikowski AP, Ettari R, Grasso S, Zappalà M, Jeong JJ, Kumar A, Hanspal M, Chishti AH. Micale N, et al. Among authors: grasso s. J Med Chem. 2006 Jun 1;49(11):3064-7. doi: 10.1021/jm060405f. J Med Chem. 2006. PMID: 16722625

5

Structure-activity study of 2,3-benzodiazepin-4-ones noncompetitive AMPAR antagonists: identification of the 1-(4-amino-3-methylphenyl)-3,5-dihydro-7,8-ethylenedioxy-4H-2,3-benzodiazepin-4-one as neuroprotective agent.

Micale N, Colleoni S, Postorino G, Pellicanò A, Zappalà M, Lazzaro J, Diana V, Cagnotto A, Mennini T, Grasso S. Micale N, et al. Among authors: grasso s. Bioorg Med Chem. 2008 Mar 1;16(5):2200-11. doi: 10.1016/j.bmc.2007.11.080. Epub 2007 Dec 5. Bioorg Med Chem. 2008. PMID: 18083036

6

Nonpeptidic vinyl and allyl phosphonates as falcipain-2 inhibitors.

Ettari R, Nizi E, Di Francesco ME, Micale N, Grasso S, Zappalà M, Vicík R, Schirmeister T. Ettari R, et al. Among authors: grasso s. ChemMedChem. 2008 Jul;3(7):1030-3. doi: 10.1002/cmdc.200800050. ChemMedChem. 2008. PMID: 18428116 No abstract available.

7

Novel peptidomimetics containing a vinyl ester moiety as highly potent and selective falcipain-2 inhibitors.

Ettari R, Micale N, Schirmeister T, Gelhaus C, Leippe M, Nizi E, Di Francesco ME, Grasso S, Zappalà M. Ettari R, et al. Among authors: grasso s. J Med Chem. 2009 Apr 9;52(7):2157-60. doi: 10.1021/jm900047j. J Med Chem. 2009. PMID: 19296600

8

Falcipain-2 inhibitors.

Ettari R, Bova F, Zappalà M, Grasso S, Micale N. Ettari R, et al. Among authors: grasso s. Med Res Rev. 2010 Jan;30(1):136-67. doi: 10.1002/med.20163. Med Res Rev. 2010. PMID: 19526594 Review.

9

Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors.

Micale N, Ettari R, Schirmeister T, Evers A, Gelhaus C, Leippe M, Zappalà M, Grasso S. Micale N, et al. Among authors: grasso s. Bioorg Med Chem. 2009 Sep 15;17(18):6505-11. doi: 10.1016/j.bmc.2009.08.013. Epub 2009 Aug 12. Bioorg Med Chem. 2009. PMID: 19709887

10

Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain.

Ettari R, Zappalà M, Micale N, Schirmeister T, Gelhaus C, Leippe M, Evers A, Grasso S. Ettari R, et al. Among authors: grasso s. Eur J Med Chem. 2010 Jul;45(7):3228-33. doi: 10.1016/j.ejmech.2010.04.003. Epub 2010 Apr 14. Eur J Med Chem. 2010. PMID: 20434817

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