Pradel G - Search Results

1

Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors.

Ettari R, Nizi E, Di Francesco ME, Dude MA, Pradel G, Vicík R, Schirmeister T, Micale N, Grasso S, Zappalà M. Ettari R, et al. Among authors: pradel g. J Med Chem. 2008 Feb 28;51(4):988-96. doi: 10.1021/jm701141u. Epub 2008 Jan 31. J Med Chem. 2008. PMID: 18232656

2

Synthesis and biological evaluation of papain-family cathepsin L-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antiprotozoal agents.

Ettari R, Pinto A, Tamborini L, Angelo IC, Grasso S, Zappalà M, Capodicasa N, Yzeiraj L, Gruber E, Aminake MN, Pradel G, Schirmeister T, De Micheli C, Conti P. Ettari R, et al. Among authors: pradel g. ChemMedChem. 2014 Aug;9(8):1817-25. doi: 10.1002/cmdc.201402079. Epub 2014 Jun 11. ChemMedChem. 2014. PMID: 24919925

3

Synthesis and evaluation of non-peptidic cysteine protease inhibitors of P. falciparum derived from etacrynic acid.

Dude MA, Kaeppler U, Herb M, Schiller M, Schulz F, Vedder B, Heppner S, Pradel G, Gut J, Rosenthal PJ, Schirmeister T, Leippe M, Gelhaus C. Dude MA, et al. Among authors: pradel g. Molecules. 2008 Dec 23;14(1):19-35. doi: 10.3390/molecules14010019. Molecules. 2008. PMID: 19104483 Free PMC article.

4

Bistacrine derivatives as new potent antimalarials.

Schmidt I, Pradel G, Sologub L, Golzmann A, Ngwa CJ, Kucharski A, Schirmeister T, Holzgrabe U. Schmidt I, et al. Among authors: pradel g. Bioorg Med Chem. 2016 Aug 15;24(16):3636-42. doi: 10.1016/j.bmc.2016.06.003. Epub 2016 Jun 4. Bioorg Med Chem. 2016. PMID: 27316542

5

Effect of protease inhibitors on exflagellation in Plasmodium falciparum.

Rupp I, Bosse R, Schirmeister T, Pradel G. Rupp I, et al. Among authors: pradel g. Mol Biochem Parasitol. 2008 Apr;158(2):208-12. doi: 10.1016/j.molbiopara.2007.12.009. Epub 2008 Jan 14. Mol Biochem Parasitol. 2008. PMID: 18243365

6

Sexual stage adhesion proteins form multi-protein complexes in the malaria parasite Plasmodium falciparum.

Simon N, Scholz SM, Moreira CK, Templeton TJ, Kuehn A, Dude MA, Pradel G. Simon N, et al. Among authors: pradel g. J Biol Chem. 2009 May 22;284(21):14537-46. doi: 10.1074/jbc.M808472200. Epub 2009 Mar 20. J Biol Chem. 2009. PMID: 19304662 Free PMC article.

7

PfCCp proteins of Plasmodium falciparum: gametocyte-specific expression and role in complement-mediated inhibition of exflagellation.

Scholz SM, Simon N, Lavazec C, Dude MA, Templeton TJ, Pradel G. Scholz SM, et al. Among authors: pradel g. Int J Parasitol. 2008 Mar;38(3-4):327-40. doi: 10.1016/j.ijpara.2007.08.009. Epub 2007 Sep 20. Int J Parasitol. 2008. PMID: 17950739

8

Inducible APOBEC3G-Vif double stable cell line as a high-throughput screening platform to identify antiviral compounds.

Nowotny B, Schneider T, Pradel G, Schirmeister T, Rethwilm A, Kirschner M. Nowotny B, et al. Among authors: pradel g. Antimicrob Agents Chemother. 2010 Jan;54(1):78-87. doi: 10.1128/AAC.00775-09. Epub 2009 Oct 19. Antimicrob Agents Chemother. 2010. PMID: 19841153 Free PMC article.

9

Synthesis and evaluation of hybrid drugs for a potential HIV/AIDS-malaria combination therapy.

Aminake MN, Mahajan A, Kumar V, Hans R, Wiesner L, Taylor D, de Kock C, Grobler A, Smith PJ, Kirschner M, Rethwilm A, Pradel G, Chibale K. Aminake MN, et al. Among authors: pradel g. Bioorg Med Chem. 2012 Sep 1;20(17):5277-89. doi: 10.1016/j.bmc.2012.06.038. Epub 2012 Jun 29. Bioorg Med Chem. 2012. PMID: 22858300

10

The bisnaphthalimides as new active lead compounds against Plasmodium falciparum.

Tischer M, Sologub L, Pradel G, Holzgrabe U. Tischer M, et al. Among authors: pradel g. Bioorg Med Chem. 2010 May 1;18(9):2998-3003. doi: 10.1016/j.bmc.2010.03.067. Epub 2010 Mar 29. Bioorg Med Chem. 2010. PMID: 20382538

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