Rokosz LL - Search Results

1

Synthesis and structure-activity relationships of new disubstituted phenyl-containing 3,4-diamino-3-cyclobutene-1,2-diones as CXCR2 receptor antagonists.

Lai G, Merritt JR, He Z, Feng D, Chao J, Czarniecki MF, Rokosz LL, Stauffer TM, Rindgen D, Taveras AG. Lai G, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2008 Mar 15;18(6):1864-8. doi: 10.1016/j.bmcl.2008.02.010. Epub 2008 Feb 10. Bioorg Med Chem Lett. 2008. PMID: 18304809

2

Discovery and SAR of 4-amino-2-biarylbutylurea MCH 1 receptor antagonists through solid-phase parallel synthesis.

Guo T, Hunter RC, Gu H, Rokosz LL, Stauffer TM, Hobbs DW. Guo T, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3691-5. doi: 10.1016/j.bmcl.2005.05.039. Bioorg Med Chem Lett. 2005. PMID: 15953726

3

Discovery and SAR of biaryl piperidine MCH1 receptor antagonists through solid-phase encoded combinatorial synthesis.

Guo T, Shao Y, Qian G, Rokosz LL, Stauffer TM, Hunter RC, Babu SD, Gu H, Hobbs DW. Guo T, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3696-700. doi: 10.1016/j.bmcl.2005.05.085. Bioorg Med Chem Lett. 2005. PMID: 15978811

4

Surfing the piperazine core of tricyclic farnesyltransferase inhibitors.

Rokosz LL, Huang CY, Reader JC, Stauffer TM, Chelsky D, Sigal NH, Ganguly AK, Baldwin JJ. Rokosz LL, et al. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5537-43. doi: 10.1016/j.bmcl.2005.08.074. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16202593

5

Synthesis and structure-activity relationships of 3,4-diaminocyclobut-3-ene-1,2-dione CXCR2 antagonists.

Merritt JR, Rokosz LL, Nelson KH Jr, Kaiser B, Wang W, Stauffer TM, Ozgur LE, Schilling A, Li G, Baldwin JJ, Taveras AG, Dwyer MP, Chao J. Merritt JR, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2006 Aug 1;16(15):4107-10. doi: 10.1016/j.bmcl.2006.04.082. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16697193

6

Discovery of 2-hydroxy-N,N-dimethyl-3-{2-[[(R)-1-(5- methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobut-1-enylamino}benzamide (SCH 527123): a potent, orally bioavailable CXCR2/CXCR1 receptor antagonist.

Dwyer MP, Yu Y, Chao J, Aki C, Chao J, Biju P, Girijavallabhan V, Rindgen D, Bond R, Mayer-Ezel R, Jakway J, Hipkin RW, Fossetta J, Gonsiorek W, Bian H, Fan X, Terminelli C, Fine J, Lundell D, Merritt JR, Rokosz LL, Kaiser B, Li G, Wang W, Stauffer T, Ozgur L, Baldwin J, Taveras AG. Dwyer MP, et al. Among authors: rokosz ll. J Med Chem. 2006 Dec 28;49(26):7603-6. doi: 10.1021/jm0609622. J Med Chem. 2006. PMID: 17181143

7

Discovery and preliminary evaluation of 5-(4-phenylbenzyl)oxazole-4-carboxamides as prostacyclin receptor antagonists.

Brescia MR, Rokosz LL, Cole AG, Stauffer TM, Lehrach JM, Auld DS, Henderson I, Webb ML. Brescia MR, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1211-5. doi: 10.1016/j.bmcl.2006.12.025. Epub 2006 Dec 12. Bioorg Med Chem Lett. 2007. PMID: 17239589

8

Design, synthesis, and evaluation of tetrahydroquinoline and pyrrolidine sulfonamide carbamates as gamma-secretase inhibitors.

Guo T, Gu H, Hobbs DW, Rokosz LL, Stauffer TM, Jacob B, Clader JW. Guo T, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3010-3. doi: 10.1016/j.bmcl.2007.03.055. Epub 2007 Mar 23. Bioorg Med Chem Lett. 2007. PMID: 17418571

9

Synthesis of 2-amino-5-benzoyl-4-(2-furyl)thiazoles as adenosine A(2A) receptor antagonists.

Cole AG, Stauffer TM, Rokosz LL, Metzger A, Dillard LW, Zeng W, Henderson I. Cole AG, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2009 Jan 15;19(2):378-81. doi: 10.1016/j.bmcl.2008.11.066. Epub 2008 Nov 24. Bioorg Med Chem Lett. 2009. PMID: 19059776

10

Synthesis and SAR studies of trisubstituted purinones as potent and selective adenosine A2A receptor antagonists.

Shao Y, Cole AG, Brescia MR, Qin LY, Duo J, Stauffer TM, Rokosz LL, McGuinness BF, Henderson I. Shao Y, et al. Among authors: rokosz ll. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1399-402. doi: 10.1016/j.bmcl.2009.01.042. Epub 2009 Jan 19. Bioorg Med Chem Lett. 2009. PMID: 19181527

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

23 results

Search Page

Filters