Bradbury BJ - Search Results

1

Muscarinic receptor binding and activation of second messengers by substituted N-methyl-N-[4-(1-azacycloalkyl)-2-butynyl]acetamides.

Bradbury BJ, Baumgold J, Paek R, Kammula U, Zimmet J, Jacobson KA. Bradbury BJ, et al. J Med Chem. 1991 Mar;34(3):1073-9. doi: 10.1021/jm00107a029. J Med Chem. 1991. PMID: 1848294

2

Functionalized congener approach to muscarinic antagonists: analogues of pirenzepine.

Karton Y, Bradbury BJ, Baumgold J, Paek R, Jacobson KA. Karton Y, et al. Among authors: bradbury bj. J Med Chem. 1991 Jul;34(7):2133-45. doi: 10.1021/jm00111a032. J Med Chem. 1991. PMID: 2066986 Free PMC article.

3

Functionalized congener approach for the design of novel muscarinic agents. Synthesis and pharmacological evaluation of N-methyl-N-[4-(1-pyrrolidinyl)-2-butynyl] amides.

Bradbury BJ, Baumgold J, Jacobson KA. Bradbury BJ, et al. J Med Chem. 1990 Feb;33(2):741-8. doi: 10.1021/jm00164a044. J Med Chem. 1990. PMID: 2153827

4

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. Among authors: bradbury bj. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

5

Synthesis and complement inhibitory activity of B/C/D-ring analogues of the fungal metabolite 6,7-diformyl-3',4',4a',5',6',7',8',8a'-octahydro-4,6',7'-trihydroxy- 2',5',5',8a'-tetramethylspiro[1'(2'H)-naphthalene-2(3H)-benzofuran].

Bradbury BJ, Bartyzel P, Kaufman TS, Nieto MJ, Sindelar RD, Scesney SM, Gaumond BR, Marsh HC Jr. Bradbury BJ, et al. J Med Chem. 2003 Jun 19;46(13):2697-705. doi: 10.1021/jm0204284. J Med Chem. 2003. PMID: 12801233

6

Exploration of the activity of 7-pyrrolidino-8-methoxyisothiazoloquinolones against methicillin-resistant Staphylococcus aureus (MRSA).

Kim HY, Wiles JA, Wang Q, Pais GC, Lucien E, Hashimoto A, Nelson DM, Thanassi JA, Podos SD, Deshpande M, Pucci MJ, Bradbury BJ. Kim HY, et al. Among authors: bradbury bj. J Med Chem. 2011 May 12;54(9):3268-82. doi: 10.1021/jm101604v. Epub 2011 Apr 15. J Med Chem. 2011. PMID: 21425851

7

Isothiazoloquinolones with enhanced antistaphylococcal activities against multidrug-resistant strains: effects of structural modifications at the 6-, 7-, and 8-positions.

Wang Q, Lucien E, Hashimoto A, Pais GC, Nelson DM, Song Y, Thanassi JA, Marlor CW, Thoma CL, Cheng J, Podos SD, Ou Y, Deshpande M, Pucci MJ, Buechter DD, Bradbury BJ, Wiles JA. Wang Q, et al. Among authors: bradbury bj. J Med Chem. 2007 Jan 25;50(2):199-210. doi: 10.1021/jm060844e. J Med Chem. 2007. PMID: 17228862

8

Biological evaluation of isothiazoloquinolones containing aromatic heterocycles at the 7-position: In vitro activity of a series of potent antibacterial agents that are effective against methicillin-resistant Staphylococcus aureus.

Wiles JA, Song Y, Wang Q, Lucien E, Hashimoto A, Cheng J, Marlor CW, Ou Y, Podos SD, Thanassi JA, Thoma CL, Deshpande M, Pucci MJ, Bradbury BJ. Wiles JA, et al. Among authors: bradbury bj. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1277-81. doi: 10.1016/j.bmcl.2005.11.064. Epub 2005 Dec 7. Bioorg Med Chem Lett. 2006. PMID: 16337789

9

Mammalian metabolism of phencyclidine.

Baker JK, Wohlford JG, Bradbury BJ, Wirth PW. Baker JK, et al. Among authors: bradbury bj. J Med Chem. 1981 Jun;24(6):666-9. doi: 10.1021/jm00138a004. J Med Chem. 1981. PMID: 7252975 No abstract available.

10

Selenophene-containing inhibitors of type IIA bacterial topoisomerases.

Wiles JA, Phadke AS, Bradbury BJ, Pucci MJ, Thanassi JA, Deshpande M. Wiles JA, et al. Among authors: bradbury bj. J Med Chem. 2011 May 12;54(9):3418-25. doi: 10.1021/jm2002124. Epub 2011 Apr 13. J Med Chem. 2011. PMID: 21443219

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