Girard GR - Search Results

1

Development of potent and selective small-molecule human Urotensin-II antagonists.

McAtee JJ, Dodson JW, Dowdell SE, Girard GR, Goodman KB, Hilfiker MA, Sehon CA, Sha D, Wang GZ, Wang N, Viet AQ, Zhang D, Aiyar NV, Behm DJ, Carballo LH, Evans CA, Fries HE, Nagilla R, Roethke TJ, Xu X, Yuan CC, Douglas SA, Neeb MJ. McAtee JJ, et al. Among authors: girard gr. Bioorg Med Chem Lett. 2008 Jun 15;18(12):3500-3. doi: 10.1016/j.bmcl.2008.05.027. Epub 2008 May 10. Bioorg Med Chem Lett. 2008. PMID: 18502123

2

Potent and selective small-molecule human urotensin-II antagonists with improved pharmacokinetic profiles.

McAtee JJ, Dodson JW, Dowdell SE, Erhard K, Girard GR, Goodman KB, Hilfiker MA, Jin J, Sehon CA, Sha D, Shi D, Wang F, Wang GZ, Wang N, Wang Y, Viet AQ, Yuan CC, Zhang D, Aiyar NV, Behm DJ, Carballo LH, Evans CA, Fries HE, Nagilla R, Roethke TJ, Xu X, Douglas SA, Neeb MJ. McAtee JJ, et al. Among authors: girard gr. Bioorg Med Chem Lett. 2008 Jul 1;18(13):3716-9. doi: 10.1016/j.bmcl.2008.05.058. Epub 2008 May 20. Bioorg Med Chem Lett. 2008. PMID: 18524591

3

Potent nonpeptide angiotensin II receptor antagonists. 2. 1-(Carboxybenzyl)imidazole-5-acrylic acids.

Keenan RM, Weinstock J, Finkelstein JA, Franz RG, Gaitanopoulos DE, Girard GR, Hill DT, Morgan TM, Samanen JM, Peishoff CE, et al. Keenan RM, et al. Among authors: girard gr. J Med Chem. 1993 Jun 25;36(13):1880-92. doi: 10.1021/jm00065a011. J Med Chem. 1993. PMID: 8515425

4

Imidazole-5-acrylic acids: potent nonpeptide angiotensin II receptor antagonists designed using a novel peptide pharmacophore model.

Keenan RM, Weinstock J, Finkelstein JA, Franz RG, Gaitanopoulos DE, Girard GR, Hill DT, Morgan TM, Samanen JM, Hempel J, et al. Keenan RM, et al. Among authors: girard gr. J Med Chem. 1992 Oct 16;35(21):3858-72. doi: 10.1021/jm00099a013. J Med Chem. 1992. PMID: 1433195

5

1-(carboxybenzyl)imidazole-5-acrylic acids: potent and selective angiotensin II receptor antagonists.

Weinstock J, Keenan RM, Samanen J, Hempel J, Finkelstein JA, Franz RG, Gaitanopoulos DE, Girard GR, Gleason JG, Hill DT, et al. Weinstock J, et al. Among authors: girard gr. J Med Chem. 1991 Apr;34(4):1514-7. doi: 10.1021/jm00108a043. J Med Chem. 1991. PMID: 2016730 No abstract available.

6

Tetrahydrothiadiazoloisoquinolines: synthesis and inhibition of phenylethanolamine-N-methyltransferase.

Girard GR, Bondinell WE, Hillegass LM, Holden KG, Pendleton RG, Uzinskas I. Girard GR, et al. J Med Chem. 1989 Jul;32(7):1566-71. doi: 10.1021/jm00127a027. J Med Chem. 1989. PMID: 2738892

7

Cytotoxicity and antitumor activity of some tetrahedral bis(diphosphino)gold(I) chelates.

Berners-Price SJ, Girard GR, Hill DT, Sutton BM, Jarrett PS, Faucette LF, Johnson RK, Mirabelli CK, Sadler PJ. Berners-Price SJ, et al. Among authors: girard gr. J Med Chem. 1990 May;33(5):1386-92. doi: 10.1021/jm00167a017. J Med Chem. 1990. PMID: 2329559

8

Orally active and potent inhibitors of gamma-aminobutyric acid uptake.

Ali FE, Bondinell WE, Dandridge PA, Frazee JS, Garvey E, Girard GR, Kaiser C, Ku TW, Lafferty JJ, Moonsammy GI, et al. Ali FE, et al. Among authors: girard gr. J Med Chem. 1985 May;28(5):653-60. doi: 10.1021/jm50001a020. J Med Chem. 1985. PMID: 2985785

9

Antitumor activity of bis(diphenylphosphino)alkanes, their gold(I) coordination complexes, and related compounds.

Mirabelli CK, Hill DT, Faucette LF, McCabe FL, Girard GR, Bryan DB, Sutton BM, Bartus JO, Crooke ST, Johnson RK. Mirabelli CK, et al. Among authors: girard gr. J Med Chem. 1987 Dec;30(12):2181-90. doi: 10.1021/jm00395a004. J Med Chem. 1987. PMID: 3681888

10

Inhibitors of phenylethanolamine N-methyltransferase and epinephrine biosynthesis. 1. Chloro-substituted 1,2,3,4-tetrahydroisoquinolines.

Bondinell WE, Chapin FW, Girard GR, Kaiser C, Krog AJ, Pavloff AM, Schwartz MS, Silvestri JS, Vaidya PD, Lam BL, Wellman GR, Pendleton RG. Bondinell WE, et al. Among authors: girard gr. J Med Chem. 1980 May;23(5):506-11. doi: 10.1021/jm00179a007. J Med Chem. 1980. PMID: 7381849

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