Kelder J - Search Results

1

A signaling-selective, nanomolar potent allosteric low molecular weight agonist for the human luteinizing hormone receptor.

van Koppen CJ, Zaman GJ, Timmers CM, Kelder J, Mosselman S, van de Lagemaat R, Smit MJ, Hanssen RG. van Koppen CJ, et al. Among authors: kelder j. Naunyn Schmiedebergs Arch Pharmacol. 2008 Nov;378(5):503-14. doi: 10.1007/s00210-008-0318-3. Epub 2008 Jun 13. Naunyn Schmiedebergs Arch Pharmacol. 2008. PMID: 18551279

2

Induction of ovulation by a potent, orally active, low molecular weight agonist (Org 43553) of the luteinizing hormone receptor.

van de Lagemaat R, Timmers CM, Kelder J, van Koppen C, Mosselman S, Hanssen RG. van de Lagemaat R, et al. Among authors: kelder j. Hum Reprod. 2009 Mar;24(3):640-8. doi: 10.1093/humrep/den412. Epub 2008 Dec 16. Hum Reprod. 2009. PMID: 19088107

3

Unique overlap in the prerequisites for thrombin inhibition and oral bioavailability resulting in potent oral antithrombotics.

Adang AE, de Man AP, Vogel GM, Grootenhuis PD, Smit MJ, Peters CA, Visser A, Rewinkel JB, van Dinther T, Lucas H, Kelder J, van Aelst S, Meuleman DG, van Boeckel CA. Adang AE, et al. Among authors: kelder j. J Med Chem. 2002 Sep 26;45(20):4419-32. doi: 10.1021/jm011110z. J Med Chem. 2002. PMID: 12238922

4

A comparison of the physicochemical and biological properties of mirtazapine and mianserin.

Kelder J, Funke C, De Boer T, Delbressine L, Leysen D, Nickolson V. Kelder J, et al. J Pharm Pharmacol. 1997 Apr;49(4):403-11. doi: 10.1111/j.2042-7158.1997.tb06814.x. J Pharm Pharmacol. 1997. PMID: 9232538

5

Comparison between steroid binding to membrane progesterone receptor alpha (mPRalpha) and to nuclear progesterone receptor: correlation with physicochemical properties assessed by comparative molecular field analysis and identification of mPRalpha-specific agonists.

Kelder J, Azevedo R, Pang Y, de Vlieg J, Dong J, Thomas P. Kelder J, et al. Steroids. 2010 Apr;75(4-5):314-22. doi: 10.1016/j.steroids.2010.01.010. Epub 2010 Jan 22. Steroids. 2010. PMID: 20096719 Free PMC article.

6

Polar molecular surface as a dominating determinant for oral absorption and brain penetration of drugs.

Kelder J, Grootenhuis PD, Bayada DM, Delbressine LP, Ploemen JP. Kelder J, et al. Pharm Res. 1999 Oct;16(10):1514-9. doi: 10.1023/a:1015040217741. Pharm Res. 1999. PMID: 10554091

7

Relation between the molecular electrostatic potential and activity of some FF-MAS related sterol compounds.

Boer DR, Kooijman H, van der Louw J, Groen M, Kelder J, Kroon J. Boer DR, et al. Among authors: kelder j. Bioorg Med Chem. 2001 Oct;9(10):2653-9. doi: 10.1016/s0968-0896(01)00189-4. Bioorg Med Chem. 2001. PMID: 11557353

8

Physicochemical properties and transport of steroids across Caco-2 cells.

Faassen F, Kelder J, Lenders J, Onderwater R, Vromans H. Faassen F, et al. Among authors: kelder j. Pharm Res. 2003 Feb;20(2):177-86. doi: 10.1023/a:1022210801734. Pharm Res. 2003. PMID: 12636155

9

Molecular modeling, mutational analysis and steroid specificity of the ligand binding pocket of mPRα (PAQR7): Shared ligand binding with AdipoR1 and its structural basis.

Kelder J, Pang Y, Dong J, Schaftenaar G, Thomas P. Kelder J, et al. J Steroid Biochem Mol Biol. 2022 May;219:106082. doi: 10.1016/j.jsbmb.2022.106082. Epub 2022 Feb 18. J Steroid Biochem Mol Biol. 2022. PMID: 35189329 Free article.

10

Steroid and G protein binding characteristics of the seatrout and human progestin membrane receptor alpha subtypes and their evolutionary origins.

Thomas P, Pang Y, Dong J, Groenen P, Kelder J, de Vlieg J, Zhu Y, Tubbs C. Thomas P, et al. Among authors: kelder j. Endocrinology. 2007 Feb;148(2):705-18. doi: 10.1210/en.2006-0974. Epub 2006 Nov 2. Endocrinology. 2007. PMID: 17082257

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