Scozzafava A - Search Results

1

Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide.

Di Fiore A, Monti SM, Hilvo M, Parkkila S, Romano V, Scaloni A, Pedone C, Scozzafava A, Supuran CT, De Simone G. Di Fiore A, et al. Among authors: scozzafava a. Proteins. 2009 Jan;74(1):164-75. doi: 10.1002/prot.22144. Proteins. 2009. PMID: 18618712

2

Carbonic anhydrase activators: human isozyme II is strongly activated by oligopeptides incorporating the carboxyterminal sequence of the bicarbonate anion exchanger AE1.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem Lett. 2002 Apr 22;12(8):1177-80. doi: 10.1016/s0960-894x(02)00121-x. Bioorg Med Chem Lett. 2002. PMID: 11934582

3

Carbonic anhydrase inhibitors.

Supuran CT, Scozzafava A, Casini A. Supuran CT, et al. Among authors: scozzafava a. Med Res Rev. 2003 Mar;23(2):146-89. doi: 10.1002/med.10025. Med Res Rev. 2003. PMID: 12500287 Review.

4

Hydroxyurea is a carbonic anhydrase inhibitor.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem. 2003 May 15;11(10):2241-6. doi: 10.1016/s0968-0896(03)00112-3. Bioorg Med Chem. 2003. PMID: 12713833

5

Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions.

Innocenti A, Lehtonen JM, Parkkila S, Scozzafava A, Supuran CT. Innocenti A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2004 Nov 1;14(21):5435-9. doi: 10.1016/j.bmcl.2004.07.086. Bioorg Med Chem Lett. 2004. PMID: 15454240

6

Benzolamide is not a membrane-impermeant carbonic anhydrase inhibitor.

Supuran CT, Scozzafava A. Supuran CT, et al. Among authors: scozzafava a. J Enzyme Inhib Med Chem. 2004 Jun;19(3):269-73. doi: 10.1080/14756360410001689559. J Enzyme Inhib Med Chem. 2004. PMID: 15499999 Free article.

7

Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.

Di Fiore A, De Simone G, Menchise V, Pedone C, Casini A, Scozzafava A, Supuran CT. Di Fiore A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2005 Apr 1;15(7):1937-42. doi: 10.1016/j.bmcl.2005.01.086. Bioorg Med Chem Lett. 2005. PMID: 15780637

8

Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.

De Simone G, Di Fiore A, Menchise V, Pedone C, Antel J, Casini A, Scozzafava A, Wurl M, Supuran CT. De Simone G, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2005 May 2;15(9):2315-20. doi: 10.1016/j.bmcl.2005.03.032. Bioorg Med Chem Lett. 2005. PMID: 15837316

9

Carbonic anhydrase inhibitors: stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II.

Menchise V, De Simone G, Alterio V, Di Fiore A, Pedone C, Scozzafava A, Supuran CT. Menchise V, et al. Among authors: scozzafava a. J Med Chem. 2005 Sep 8;48(18):5721-7. doi: 10.1021/jm050333c. J Med Chem. 2005. PMID: 16134940

10

Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II "selective" inhibitor celecoxib.

Di Fiore A, Pedone C, D'Ambrosio K, Scozzafava A, De Simone G, Supuran CT. Di Fiore A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2006 Jan 15;16(2):437-42. doi: 10.1016/j.bmcl.2005.09.040. Epub 2005 Nov 14. Bioorg Med Chem Lett. 2006. PMID: 16290146

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