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Page 1
Synthesis and cytotoxic activity of polyamine analogues of camptothecin.
Dallavalle S, Giannini G, Alloatti D, Casati A, Marastoni E, Musso L, Merlini L, Morini G, Penco S, Pisano C, Tinelli S, De Cesare M, Beretta GL, Zunino F. Dallavalle S, et al. Among authors: giannini g. J Med Chem. 2006 Aug 24;49(17):5177-86. doi: 10.1021/jm060285b. J Med Chem. 2006. PMID: 16913706
A novel atypical retinoid endowed with proapoptotic and antitumor activity.
Cincinelli R, Dallavalle S, Merlini L, Penco S, Pisano C, Carminati P, Giannini G, Vesci L, Gaetano C, Illy B, Zuco V, Supino R, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2003 Mar 13;46(6):909-12. doi: 10.1021/jm025593y. J Med Chem. 2003. PMID: 12620066
Synthesis and structure-activity relationships of a new series of retinoid-related biphenyl-4-ylacrylic acids endowed with antiproliferative and proapoptotic activity.
Cincinelli R, Dallavalle S, Nannei R, Carella S, De Zani D, Merlini L, Penco S, Garattini E, Giannini G, Pisano C, Vesci L, Carminati P, Zuco V, Zanchi C, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2005 Jul 28;48(15):4931-46. doi: 10.1021/jm049440h. J Med Chem. 2005. PMID: 16033272
Synthesis and biological activity of fluorinated combretastatin analogues.
Alloatti D, Giannini G, Cabri W, Lustrati I, Marzi M, Ciacci A, Gallo G, Tinti MO, Marcellini M, Riccioni T, Guglielmi MB, Carminati P, Pisano C. Alloatti D, et al. Among authors: giannini g. J Med Chem. 2008 May 8;51(9):2708-21. doi: 10.1021/jm701362m. Epub 2008 Apr 9. J Med Chem. 2008. PMID: 18396857
Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.
Taddei M, Ferrini S, Giannotti L, Corsi M, Manetti F, Giannini G, Vesci L, Milazzo FM, Alloatti D, Guglielmi MB, Castorina M, Cervoni ML, Barbarino M, Foderà R, Carollo V, Pisano C, Armaroli S, Cabri W. Taddei M, et al. Among authors: giannini g. J Med Chem. 2014 Mar 27;57(6):2258-74. doi: 10.1021/jm401536b. Epub 2014 Mar 17. J Med Chem. 2014. PMID: 24588105
Camptothecins in tumor homing via an RGD sequence mimetic.
Alloatti D, Giannini G, Vesci L, Castorina M, Pisano C, Badaloni E, Cabri W. Alloatti D, et al. Among authors: giannini g. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6509-12. doi: 10.1016/j.bmcl.2012.07.061. Epub 2012 Jul 26. Bioorg Med Chem Lett. 2012. PMID: 22959246
440 results