Jacobson KA - Search Results

1

Molecular recognition in the P2Y(14) receptor: Probing the structurally permissive terminal sugar moiety of uridine-5'-diphosphoglucose.

Ko H, Das A, Carter RL, Fricks IP, Zhou Y, Ivanov AA, Melman A, Joshi BV, Kovác P, Hajduch J, Kirk KL, Harden TK, Jacobson KA. Ko H, et al. Among authors: jacobson ka. Bioorg Med Chem. 2009 Jul 15;17(14):5298-311. doi: 10.1016/j.bmc.2009.05.024. Epub 2009 May 15. Bioorg Med Chem. 2009. PMID: 19502066 Free PMC article.

2

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

3

Adenosine A1 and A2 receptors: structure--function relationships.

van Galen PJ, Stiles GL, Michaels G, Jacobson KA. van Galen PJ, et al. Among authors: jacobson ka. Med Res Rev. 1992 Sep;12(5):423-71. doi: 10.1002/med.2610120502. Med Res Rev. 1992. PMID: 1513184 Free PMC article. Review. No abstract available.

4

In vivo imaging of insulin receptors in monkeys using 18F-labeled insulin and positron emission tomography.

Eastman RC, Carson RE, Jacobson KA, Shai Y, Channing MA, Dunn BB, Bacher JD, Baas E, Jones E, Kirk KL, et al. Eastman RC, et al. Among authors: jacobson ka. Diabetes. 1992 Jul;41(7):855-60. doi: 10.2337/diab.41.7.855. Diabetes. 1992. PMID: 1612200 Free PMC article.

5

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.

Jacobson KA, van Galen PJ, Williams M. Jacobson KA, et al. J Med Chem. 1992 Feb 7;35(3):407-22. doi: 10.1021/jm00081a001. J Med Chem. 1992. PMID: 1738138 Free PMC article. Review. No abstract available.

6

Muscarinic receptor binding and activation of second messengers by substituted N-methyl-N-[4-(1-azacycloalkyl)-2-butynyl]acetamides.

Bradbury BJ, Baumgold J, Paek R, Kammula U, Zimmet J, Jacobson KA. Bradbury BJ, et al. Among authors: jacobson ka. J Med Chem. 1991 Mar;34(3):1073-9. doi: 10.1021/jm00107a029. J Med Chem. 1991. PMID: 1848294

7

Functionalized congener approach to muscarinic antagonists: analogues of pirenzepine.

Karton Y, Bradbury BJ, Baumgold J, Paek R, Jacobson KA. Karton Y, et al. Among authors: jacobson ka. J Med Chem. 1991 Jul;34(7):2133-45. doi: 10.1021/jm00111a032. J Med Chem. 1991. PMID: 2066986 Free PMC article.

8

Functionalized congener approach for the design of novel muscarinic agents. Synthesis and pharmacological evaluation of N-methyl-N-[4-(1-pyrrolidinyl)-2-butynyl] amides.

Bradbury BJ, Baumgold J, Jacobson KA. Bradbury BJ, et al. Among authors: jacobson ka. J Med Chem. 1990 Feb;33(2):741-8. doi: 10.1021/jm00164a044. J Med Chem. 1990. PMID: 2153827

9

Evidence that a novel 8-phenyl-substituted xanthine derivative is a cardioselective adenosine receptor antagonist in vivo.

Fredholm BB, Jacobson KA, Jonzon B, Kirk KL, Li YO, Daly JW. Fredholm BB, et al. Among authors: jacobson ka. J Cardiovasc Pharmacol. 1987 Apr;9(4):396-400. doi: 10.1097/00005344-198704000-00003. J Cardiovasc Pharmacol. 1987. PMID: 2438501 Free PMC article.

10

Binary drugs: conjugates of purines and a peptide that bind to both adenosine and substance P receptors.

Jacobson KA, Lipkowski AW, Moody TW, Padgett W, Pijl E, Kirk KL, Daly JW. Jacobson KA, et al. J Med Chem. 1987 Aug;30(8):1529-32. doi: 10.1021/jm00391a046. J Med Chem. 1987. PMID: 2441057 Free PMC article.

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