Ghelardini C - Search Results

1

Synthesis, in vivo evaluation, and molecular modeling studies of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide derivatives. Identification of a bifunctional hydrogen bond area related to the inverse agonism.

Guerrini G, Ciciani G, Cambi G, Bruni F, Selleri S, Guarino C, Melani F, Montali M, Martini C, Ghelardini C, Norcini M, Costanzo A. Guerrini G, et al. Among authors: ghelardini c. J Med Chem. 2009 Aug 13;52(15):4668-82. doi: 10.1021/jm801599a. J Med Chem. 2009. PMID: 19591485

2

Presynaptic cholinergic modulators as potent cognition enhancers and analgesic drugs. 1. Tropic and 2-phenylpropionic acid esters.

Gualtieri F, Conti G, Dei S, Giovannoni MP, Nannucci F, Romanelli MN, Scapecchi S, Teodori E, Fanfani L, Ghelardini C, et al. Gualtieri F, et al. Among authors: ghelardini c. J Med Chem. 1994 May 27;37(11):1704-11. doi: 10.1021/jm00037a022. J Med Chem. 1994. PMID: 8201605

3

Mono- and disubstituted-3,8-diazabicyclo[3.2.1]octane derivatives as analgesics structurally related to epibatidine: synthesis, activity, and modeling.

Barlocco D, Cignarella G, Tondi D, Vianello P, Villa S, Bartolini A, Ghelardini C, Galeotti N, Anderson DJ, Kuntzweiler TA, Colombo D, Toma L. Barlocco D, et al. Among authors: ghelardini c. J Med Chem. 1998 Feb 26;41(5):674-81. doi: 10.1021/jm970427p. J Med Chem. 1998. PMID: 9513595

4

Hybridized and isosteric analogues of N1-acetyl-N4-dimethyl-piperazinium iodide (ADMP) and N1-phenyl-N4-dimethyl-piperazinium iodide (DMPP) with central nicotinic action.

Manetti D, Bartolini A, Borea PA, Bellucci C, Dei S, Ghelardini C, Gualtieri F, Romanelli MN, Scapecchi S, Teodori E, Varani K. Manetti D, et al. Among authors: ghelardini c. Bioorg Med Chem. 1999 Mar;7(3):457-65. doi: 10.1016/s0968-0896(98)00259-4. Bioorg Med Chem. 1999. PMID: 10220032

5

Design, synthesis, and preliminary pharmacological evaluation of 1, 4-diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic agents.

Manetti D, Ghelardini C, Bartolini A, Bellucci C, Dei S, Galeotti N, Gualtieri F, Romanelli MN, Scapecchi S, Teodori E. Manetti D, et al. Among authors: ghelardini c. J Med Chem. 2000 May 18;43(10):1969-74. doi: 10.1021/jm991170t. J Med Chem. 2000. PMID: 10821709

6

Molecular simplification of 1,4-diazabicyclo[4.3.0]nonan-9-ones gives piperazine derivatives that maintain high nootropic activity.

Manetti D, Ghelardini C, Bartolini A, Dei S, Galeotti N, Gualtieri F, Romanelli MN, Teodori E. Manetti D, et al. Among authors: ghelardini c. J Med Chem. 2000 Nov 16;43(23):4499-507. doi: 10.1021/jm000972h. J Med Chem. 2000. PMID: 11087574

7

Structure-affinity relationships of a unique nicotinic ligand: N(1)-dimethyl-N(4)-phenylpiperazinium iodide (DMPP).

Romanelli MN, Manetti D, Scapecchi S, Borea PA, Dei S, Bartolini A, Ghelardini C, Gualtieri F, Guandalini L, Varani K. Romanelli MN, et al. Among authors: ghelardini c. J Med Chem. 2001 Nov 8;44(23):3946-55. doi: 10.1021/jm010901y. J Med Chem. 2001. PMID: 11689081

8

Novel potent 5-HT(3) receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities.

Cappelli A, Anzini M, Vomero S, Mennuni L, Makovec F, Doucet E, Hamon M, Menziani MC, De Benedetti PG, Giorgi G, Ghelardini C, Collina S. Cappelli A, et al. Among authors: ghelardini c. Bioorg Med Chem. 2002 Mar;10(3):779-801. doi: 10.1016/s0968-0896(01)00332-7. Bioorg Med Chem. 2002. PMID: 11814868

9

[(3-Chlorophenyl)piperazinylpropyl]pyridazinones and analogues as potent antinociceptive agents.

Giovannoni MP, Vergelli C, Ghelardini C, Galeotti N, Bartolini A, Dal Piaz V. Giovannoni MP, et al. Among authors: ghelardini c. J Med Chem. 2003 Mar 13;46(6):1055-9. doi: 10.1021/jm021057u. J Med Chem. 2003. PMID: 12620082

10

4-Aminopiperidine derivatives as a new class of potent cognition enhancing drugs.

Manetti D, Martini E, Ghelardini C, Dei S, Galeotti N, Guandalini L, Romanelli MN, Scapecchi S, Teodori E, Bartolini A, Gualtieri F. Manetti D, et al. Among authors: ghelardini c. Bioorg Med Chem Lett. 2003 Jul 21;13(14):2303-6. doi: 10.1016/s0960-894x(03)00437-2. Bioorg Med Chem Lett. 2003. PMID: 12824022

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