Deflorian F - Search Results

1

Structural basis of the selectivity of the beta(2)-adrenergic receptor for fluorinated catecholamines.

Pooput C, Rosemond E, Karpiak J, Deflorian F, Vilar S, Costanzi S, Wess J, Kirk KL. Pooput C, et al. Among authors: deflorian f. Bioorg Med Chem. 2009 Dec 1;17(23):7987-92. doi: 10.1016/j.bmc.2009.10.015. Epub 2009 Oct 13. Bioorg Med Chem. 2009. PMID: 19857969 Free PMC article.

2

Probing GPCR structure: adenosine and P2Y nucleotide receptors.

Jacobson KA, Costanzi S, Deflorian F. Jacobson KA, et al. Among authors: deflorian f. Methods Enzymol. 2013;520:199-217. doi: 10.1016/B978-0-12-391861-1.00009-5. Methods Enzymol. 2013. PMID: 23332701 Free PMC article.

3

Pharmacochemistry of the platelet purinergic receptors.

Jacobson KA, Deflorian F, Mishra S, Costanzi S. Jacobson KA, et al. Among authors: deflorian f. Purinergic Signal. 2011 Sep;7(3):305-24. doi: 10.1007/s11302-011-9216-0. Epub 2011 Feb 18. Purinergic Signal. 2011. PMID: 21484092 Free PMC article.

4

Understanding the structural and functional differences between mouse thyrotropin-releasing hormone receptors 1 and 2.

Deflorian F, Engel S, Colson AO, Raaka BM, Gershengorn MC, Costanzi S. Deflorian F, et al. Proteins. 2008 May 1;71(2):783-94. doi: 10.1002/prot.21763. Proteins. 2008. PMID: 17979196

5

Examining the chirality, conformation and selective kinase inhibition of 3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)piperidin-1-yl)-3-oxopropanenitrile (CP-690,550).

Jiang JK, Ghoreschi K, Deflorian F, Chen Z, Perreira M, Pesu M, Smith J, Nguyen DT, Liu EH, Leister W, Costanzi S, O'Shea JJ, Thomas CJ. Jiang JK, et al. Among authors: deflorian f. J Med Chem. 2008 Dec 25;51(24):8012-8. doi: 10.1021/jm801142b. J Med Chem. 2008. PMID: 19053756 Free PMC article.

6

Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening.

Tosh DK, Phan K, Gao ZG, Gakh AA, Xu F, Deflorian F, Abagyan R, Stevens RC, Jacobson KA, Katritch V. Tosh DK, et al. Among authors: deflorian f. J Med Chem. 2012 May 10;55(9):4297-308. doi: 10.1021/jm300095s. Epub 2012 Apr 30. J Med Chem. 2012. PMID: 22486652 Free PMC article.

7

Evaluation of molecular modeling of agonist binding in light of the crystallographic structure of an agonist-bound A₂A adenosine receptor.

Deflorian F, Kumar TS, Phan K, Gao ZG, Xu F, Wu H, Katritch V, Stevens RC, Jacobson KA. Deflorian F, et al. J Med Chem. 2012 Jan 12;55(1):538-52. doi: 10.1021/jm201461q. Epub 2011 Dec 12. J Med Chem. 2012. PMID: 22104008 Free PMC article.

8

Structure-guided design of A(3) adenosine receptor-selective nucleosides: combination of 2-arylethynyl and bicyclo[3.1.0]hexane substitutions.

Tosh DK, Deflorian F, Phan K, Gao ZG, Wan TC, Gizewski E, Auchampach JA, Jacobson KA. Tosh DK, et al. Among authors: deflorian f. J Med Chem. 2012 May 24;55(10):4847-60. doi: 10.1021/jm300396n. Epub 2012 May 16. J Med Chem. 2012. PMID: 22559880 Free PMC article.

9

Structural sweet spot for A1 adenosine receptor activation by truncated (N)-methanocarba nucleosides: receptor docking and potent anticonvulsant activity.

Tosh DK, Paoletta S, Deflorian F, Phan K, Moss SM, Gao ZG, Jiang X, Jacobson KA. Tosh DK, et al. Among authors: deflorian f. J Med Chem. 2012 Sep 27;55(18):8075-90. doi: 10.1021/jm300965a. Epub 2012 Sep 10. J Med Chem. 2012. PMID: 22921089 Free PMC article.

10

Molecular probes for the A2A adenosine receptor based on a pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine scaffold.

Kumar TS, Mishra S, Deflorian F, Yoo LS, Phan K, Kecskés M, Szabo A, Shinkre B, Gao ZG, Trenkle W, Jacobson KA. Kumar TS, et al. Among authors: deflorian f. Bioorg Med Chem Lett. 2011 May 1;21(9):2740-5. doi: 10.1016/j.bmcl.2010.11.082. Epub 2010 Nov 21. Bioorg Med Chem Lett. 2011. PMID: 21185184 Free PMC article.

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