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Discovery and structure-activity relationships of new steroidal compounds bearing a carboxy-terminal side chain as androgen receptor pure antagonists.
Tachibana K, Imaoka I, Yoshino H, Kato N, Nakamura M, Ohta M, Kawata H, Taniguchi K, Ishikura N, Nagamuta M, Onuma E, Sato H. Tachibana K, et al. Among authors: kawata h. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5573-6. doi: 10.1016/j.bmcl.2007.07.090. Epub 2007 Aug 22. Bioorg Med Chem Lett. 2007. PMID: 17804229
Discovery of an orally-active nonsteroidal androgen receptor pure antagonist and the structure-activity relationships of its derivatives.
Tachibana K, Imaoka I, Shiraishi T, Yoshino H, Nakamura M, Ohta M, Kawata H, Taniguchi K, Ishikura N, Tsunenari T, Saito H, Nagamuta M, Nakagawa T, Takanashi K, Onuma E, Sato H. Tachibana K, et al. Among authors: kawata h. Chem Pharm Bull (Tokyo). 2008 Nov;56(11):1555-61. doi: 10.1248/cpb.56.1555. Chem Pharm Bull (Tokyo). 2008. PMID: 18981605 Free article.
Design and synthesis of an androgen receptor pure antagonist (CH5137291) for the treatment of castration-resistant prostate cancer.
Yoshino H, Sato H, Shiraishi T, Tachibana K, Emura T, Honma A, Ishikura N, Tsunenari T, Watanabe M, Nishimoto A, Nakamura R, Nakagawa T, Ohta M, Takata N, Furumoto K, Kimura K, Kawata H. Yoshino H, et al. Among authors: kawata h. Bioorg Med Chem. 2010 Dec 1;18(23):8150-7. doi: 10.1016/j.bmc.2010.10.023. Epub 2010 Oct 15. Bioorg Med Chem. 2010. PMID: 21050768
CH5137291, an androgen receptor nuclear translocation-inhibiting compound, inhibits the growth of castration-resistant prostate cancer cells.
Ishikura N, Kawata H, Nishimoto A, Nakamura R, Tsunenari T, Watanabe M, Tachibana K, Shiraishi T, Yoshino H, Honma A, Emura T, Ohta M, Nakagawa T, Houjo T, Corey E, Vessella RL, Aoki Y, Sato H. Ishikura N, et al. Among authors: kawata h. Int J Oncol. 2015 Apr;46(4):1560-72. doi: 10.3892/ijo.2015.2860. Epub 2015 Jan 30. Int J Oncol. 2015. PMID: 25634071
A novel nonsecosteroidal VDR agonist (CH5036249) exhibits efficacy in a spontaneous benign prostatic hyperplasia beagle model.
Taniguchi K, Katagiri K, Kashiwagi H, Harada S, Sugimoto Y, Shimizu Y, Arakawa H, Ito T, Yamazaki M, Watanabe T, Kato A, Hoshino E, Takahashi T, Esaki T, Suzuki M, Takeda S, Ichikawa F, Harada A, Sekiguchi N, Ishigai M, Kawata H, Yoneya T, Onuma E, Sudoh M, Aoki Y. Taniguchi K, et al. Among authors: kawata h. J Steroid Biochem Mol Biol. 2010 Jul;121(1-2):204-7. doi: 10.1016/j.jsbmb.2010.03.043. Epub 2010 Mar 18. J Steroid Biochem Mol Biol. 2010. PMID: 20304062
407 results