Tkachenko S - Search Results

1

Recombinant yeast screen for new inhibitors of human acetyl-CoA carboxylase 2 identifies potential drugs to treat obesity.

Marjanovic J, Chalupska D, Patenode C, Coster A, Arnold E, Ye A, Anesi G, Lu Y, Okun I, Tkachenko S, Haselkorn R, Gornicki P. Marjanovic J, et al. Among authors: tkachenko s. Proc Natl Acad Sci U S A. 2010 May 18;107(20):9093-8. doi: 10.1073/pnas.1003721107. Epub 2010 May 3. Proc Natl Acad Sci U S A. 2010. PMID: 20439761 Free PMC article.

2

1,3-Dioxo-4-methyl-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines as potent caspase-3 inhibitors.

Kravchenko DV, Kysil VV, Ilyn AP, Tkachenko SE, Maliarchouk S, Okun IM, Ivachtchenko AV. Kravchenko DV, et al. Among authors: tkachenko se. Bioorg Med Chem Lett. 2005 Apr 1;15(7):1841-5. doi: 10.1016/j.bmcl.2005.02.027. Bioorg Med Chem Lett. 2005. PMID: 15780618

3

Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. Synthesis and SAR of 2-substituted 4-methyl-8-(morpholine-4-sulfonyl)-pyrrolo[3,4-c]quinoline-1,3-diones.

Kravchenko DV, Kysil VM, Tkachenko SE, Maliarchouk S, Okun IM, Ivachtchenko AV. Kravchenko DV, et al. Among authors: tkachenko se. Eur J Med Chem. 2005 Dec;40(12):1377-83. doi: 10.1016/j.ejmech.2005.07.011. Epub 2005 Sep 15. Eur J Med Chem. 2005. PMID: 16169127

4

Synthesis and caspase-3 inhibitory activity of 8-sulfonyl-1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines.

Kravchenko DV, Kysil VM, Tkachenko SE, Maliarchouk S, Okun IM, Ivachtchenko AV. Kravchenko DV, et al. Among authors: tkachenko se. Farmaco. 2005 Oct;60(10):804-9. doi: 10.1016/j.farmac.2005.08.001. Epub 2005 Sep 21. Farmaco. 2005. PMID: 16182295

5

8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.

Ivachtchenko AV, Mitkin OD, Tkachenko SE, Okun IM, Kysil VM. Ivachtchenko AV, et al. Eur J Med Chem. 2010 Feb;45(2):782-9. doi: 10.1016/j.ejmech.2009.10.035. Epub 2009 Oct 31. Eur J Med Chem. 2010. PMID: 19939513

6

Synthesis and biological evaluation of novel gamma-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists.

Ivachtchenko AV, Frolov EB, Mitkin OD, Kysil VM, Khvat AV, Okun IM, Tkachenko SE. Ivachtchenko AV, et al. Bioorg Med Chem Lett. 2009 Jun 15;19(12):3183-7. doi: 10.1016/j.bmcl.2009.04.128. Epub 2009 May 3. Bioorg Med Chem Lett. 2009. PMID: 19443217

7

Synthesis and structure-activity relationship of 4-substituted 2-(2-acetyloxyethyl)-8-(morpholine-4-sulfonyl)pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors.

Kravchenko DV, Kuzovkova YA, Kysil VM, Tkachenko SE, Maliarchouk S, Okun IM, Balakin KV, Ivachtchenko AV. Kravchenko DV, et al. Among authors: tkachenko se. J Med Chem. 2005 Jun 2;48(11):3680-3. doi: 10.1021/jm048987t. J Med Chem. 2005. PMID: 15916416

8

Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists.

Ivachtchenko AV, Golovina ES, Kadieva MG, Kysil VM, Mitkin OD, Tkachenko SE, Okun I. Ivachtchenko AV, et al. Among authors: tkachenko se. Bioorg Med Chem. 2011 Feb 15;19(4):1482-91. doi: 10.1016/j.bmc.2010.12.055. Epub 2011 Jan 5. Bioorg Med Chem. 2011. PMID: 21277782

9

2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: new series of highly potent and specific serotonin 5-HT6 receptor antagonists.

Ivachtchenko AV, Golovina ES, Kadieva MG, Koryakova AG, Mitkin OD, Tkachenko SE, Kysil VM, Okun I. Ivachtchenko AV, et al. Among authors: tkachenko se. Eur J Med Chem. 2011 Apr;46(4):1189-97. doi: 10.1016/j.ejmech.2011.01.038. Epub 2011 Feb 1. Eur J Med Chem. 2011. PMID: 21333408

10

Synthesis and structure-activity relationship (SAR) of (5,7-disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as potent serotonin 5-HT(6) receptor (5-HT(6)R) antagonists.

Ivachtchenko AV, Golovina ES, Kadieva MG, Kysil VM, Mitkin OD, Tkachenko SE, Okun IM. Ivachtchenko AV, et al. Among authors: tkachenko se. J Med Chem. 2011 Dec 8;54(23):8161-73. doi: 10.1021/jm201079g. Epub 2011 Nov 10. J Med Chem. 2011. PMID: 22029285

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