Brancale A - Search Results

1

Synthesis and CYP24A1 inhibitory activity of (E)-2-(2-substituted benzylidene)- and 2-(2-substituted benzyl)-6-methoxy-tetralones.

Aboraia AS, Makowski B, Bahja A, Prosser D, Brancale A, Jones G, Simons C. Aboraia AS, et al. Among authors: brancale a. Eur J Med Chem. 2010 Oct;45(10):4427-34. doi: 10.1016/j.ejmech.2010.07.001. Epub 2010 Jul 8. Eur J Med Chem. 2010. PMID: 20655626

2

Potent and selective inhibition of varicella-zoster virus (VZV) by nucleoside analogues with an unusual bicyclic base.

McGuigan C, Yarnold CJ, Jones G, Velázquez S, Barucki H, Brancale A, Andrei G, Snoeck R, De Clercq E, Balzarini J. McGuigan C, et al. Among authors: brancale a. J Med Chem. 1999 Nov 4;42(22):4479-84. doi: 10.1021/jm990346o. J Med Chem. 1999. PMID: 10579812

3

Furano pyrimidines as novel potent and selective anti-VZV agents.

McGuigan C, Brancale A, Barucki H, Srinivasan S, Jones G, Pathirana R, Carangio A, Blewett S, Luoni G, Bidet O, Jukes A, Jarvis C, Andrei G, Snoeck R, De Clercq E, Balzarini J. McGuigan C, et al. Among authors: brancale a. Antivir Chem Chemother. 2001 Mar;12(2):77-89. doi: 10.1177/095632020101200201. Antivir Chem Chemother. 2001. PMID: 11527045 Free article. Review.

4

Novel bicyclic furanopyrimidines with dual anti-VZV and -HCMV activity.

McGuigan C, Brancale A, Andrei G, Snoeck R, De Clercq E, Balzarini J. McGuigan C, et al. Among authors: brancale a. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4511-3. doi: 10.1016/j.bmcl.2003.08.028. Bioorg Med Chem Lett. 2003. PMID: 14643358

5

Novel tetralone-derived retinoic acid metabolism blocking agents: synthesis and in vitro evaluation with liver microsomal and MCF-7 CYP26A1 cell assays.

Yee SW, Jarno L, Gomaa MS, Elford C, Ooi LL, Coogan MP, McClelland R, Nicholson RI, Evans BA, Brancale A, Simons C. Yee SW, et al. Among authors: brancale a. J Med Chem. 2005 Nov 17;48(23):7123-31. doi: 10.1021/jm0501681. J Med Chem. 2005. PMID: 16279770

6

Novel potential anticancer naphthyl phosphoramidates of BVdU: separation of diastereoisomers and assignment of the absolute configuration of the phosphorus center.

Congiatu C, Brancale A, Mason MD, Jiang WG, McGuigan C. Congiatu C, et al. Among authors: brancale a. J Med Chem. 2006 Jan 26;49(2):452-5. doi: 10.1021/jm0509896. J Med Chem. 2006. PMID: 16420029

7

Homology model of human retinoic acid metabolising enzyme cytochrome P450 26A1 (CYP26A1): active site architecture and ligand binding.

Gomaa MS, Yee SW, Milbourne CE, Barbera MC, Simons C, Brancale A. Gomaa MS, et al. Among authors: brancale a. J Enzyme Inhib Med Chem. 2006 Aug;21(4):361-9. doi: 10.1080/14756360600742014. J Enzyme Inhib Med Chem. 2006. PMID: 17059167 Free article.

8

Homology model of 1alpha,25-dihydroxyvitamin D3 24-hydroxylase cytochrome P450 24A1 (CYP24A1): active site architecture and ligand binding.

Gomaa MS, Simons C, Brancale A. Gomaa MS, et al. Among authors: brancale a. J Steroid Biochem Mol Biol. 2007 Apr;104(1-2):53-60. doi: 10.1016/j.jsbmb.2006.09.041. Epub 2007 Jan 19. J Steroid Biochem Mol Biol. 2007. PMID: 17240137

9

Design and synthesis of substituted imidazole and triazole N-phenylbenzo[d]oxazolamine inhibitors of retinoic acid metabolizing enzyme CYP26.

Pautus S, Aboraia AS, Bassett CE, Brancale A, Coogan MP, Simons C. Pautus S, et al. Among authors: brancale a. J Enzyme Inhib Med Chem. 2009 Apr;24(2):487-98. doi: 10.1080/14756360802218334. J Enzyme Inhib Med Chem. 2009. PMID: 18608743 Free article.

10

Novel azolyl-(phenylmethyl)]aryl/heteroarylamines: potent CYP26 inhibitors and enhancers of all-trans retinoic acid activity in neuroblastoma cells.

Gomaa MS, Armstrong JL, Bobillon B, Veal GJ, Brancale A, Redfern CP, Simons C. Gomaa MS, et al. Among authors: brancale a. Bioorg Med Chem. 2008 Sep 1;16(17):8301-13. doi: 10.1016/j.bmc.2007.06.048. Epub 2007 Jun 29. Bioorg Med Chem. 2008. PMID: 18722776

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