Jacobson KA - Search Results

1

Synthesis and evaluation of 1,2,4-triazolo[1,5-c]pyrimidine derivatives as A2A receptor-selective antagonists.

Shinkre BA, Kumar TS, Gao ZG, Deflorian F, Jacobson KA, Trenkle WC. Shinkre BA, et al. Among authors: jacobson ka. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5690-4. doi: 10.1016/j.bmcl.2010.08.021. Epub 2010 Aug 10. Bioorg Med Chem Lett. 2010. PMID: 20801028 Free PMC article.

2

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

3

Muscarinic receptor binding and activation of second messengers by substituted N-methyl-N-[4-(1-azacycloalkyl)-2-butynyl]acetamides.

Bradbury BJ, Baumgold J, Paek R, Kammula U, Zimmet J, Jacobson KA. Bradbury BJ, et al. Among authors: jacobson ka. J Med Chem. 1991 Mar;34(3):1073-9. doi: 10.1021/jm00107a029. J Med Chem. 1991. PMID: 1848294

4

Functionalized congener approach to muscarinic antagonists: analogues of pirenzepine.

Karton Y, Bradbury BJ, Baumgold J, Paek R, Jacobson KA. Karton Y, et al. Among authors: jacobson ka. J Med Chem. 1991 Jul;34(7):2133-45. doi: 10.1021/jm00111a032. J Med Chem. 1991. PMID: 2066986 Free PMC article.

5

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Jacobson KA, Barone S, Kammula U, Stiles GL. Jacobson KA, et al. J Med Chem. 1989 May;32(5):1043-51. doi: 10.1021/jm00125a019. J Med Chem. 1989. PMID: 2709373 Free PMC article.

6

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

7

Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors.

Siddiqi SM, Jacobson KA, Esker JL, Olah ME, Ji XD, Melman N, Tiwari KN, Secrist JA 3rd, Schneller SW, Cristalli G, et al. Siddiqi SM, et al. Among authors: jacobson ka. J Med Chem. 1995 Mar 31;38(7):1174-88. doi: 10.1021/jm00007a014. J Med Chem. 1995. PMID: 7707320 Free PMC article.

8

Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors.

Jacobson KA, Siddiqi SM, Olah ME, Ji XD, Melman N, Bellamkonda K, Meshulam Y, Stiles GL, Kim HO. Jacobson KA, et al. J Med Chem. 1995 May 12;38(10):1720-35. doi: 10.1021/jm00010a017. J Med Chem. 1995. PMID: 7752196 Free PMC article.

9

Structure-activity relationships of 1,3-dialkylxanthine derivatives at rat A3 adenosine receptors.

Kim HO, Ji XD, Melman N, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Sep 30;37(20):3373-82. doi: 10.1021/jm00046a022. J Med Chem. 1994. PMID: 7932565 Free PMC article.

10

2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors.

Kim HO, Ji XD, Siddiqi SM, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Oct 14;37(21):3614-21. doi: 10.1021/jm00047a018. J Med Chem. 1994. PMID: 7932588 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

852 results

Search Page

Filters