Evans KA - Search Results

1

3-Urea-1-(phenylmethyl)-pyridones as novel, potent, and selective EP3 receptor antagonists.

Li YH, Tseng PS, Evans KA, Jaworski JP, Morrow DM, Fries HE, Wu CW, Edwards RM, Jin J. Li YH, et al. Among authors: evans ka. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6744-7. doi: 10.1016/j.bmcl.2010.08.137. Bioorg Med Chem Lett. 2010. PMID: 20926294

2

Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists.

Jin J, Morales-Ramos A, Eidam P, Mecom J, Li Y, Brooks C, Hilfiker M, Zhang D, Wang N, Shi D, Tseng PS, Wheless K, Budzik B, Evans K, Jaworski JP, Jugus J, Leon L, Wu C, Pullen M, Karamshi B, Rao P, Ward E, Laping N, Evans C, Leach C, Holt D, Su X, Morrow D, Fries H, Thorneloe K, Edwards R. Jin J, et al. ACS Med Chem Lett. 2010 May 14;1(7):316-20. doi: 10.1021/ml100077x. eCollection 2010 Oct 14. ACS Med Chem Lett. 2010. PMID: 24900213 Free PMC article.

3

Synthesis and structure-activity relationships of a series of 3-aryl-4-isoxazolecarboxamides as a new class of TGR5 agonists.

Budzik BW, Evans KA, Wisnoski DD, Jin J, Rivero RA, Szewczyk GR, Jayawickreme C, Moncol DL, Yu H. Budzik BW, et al. Among authors: evans ka. Bioorg Med Chem Lett. 2010 Feb 15;20(4):1363-7. doi: 10.1016/j.bmcl.2010.01.003. Epub 2010 Jan 7. Bioorg Med Chem Lett. 2010. PMID: 20097073

4

Synthesis and structure-activity relationships of 3-phenyl-2-propenamides as inhibitors of glycogen phosphorylase a.

Li YH, Coppo FT, Evans KA, Graybill TL, Patel M, Gale J, Li H, Tavares F, Thomson SA. Li YH, et al. Among authors: evans ka. Bioorg Med Chem Lett. 2006 Nov 15;16(22):5892-6. doi: 10.1016/j.bmcl.2006.08.055. Epub 2006 Aug 30. Bioorg Med Chem Lett. 2006. PMID: 16942879

5

Amino acid anthranilamide derivatives as a new class of glycogen phosphorylase inhibitors.

Evans KA, Li YH, Coppo FT, Graybill TL, Cichy-Knight M, Patel M, Gale J, Li H, Thrall SH, Tew D, Tavares F, Thomson SA, Weiel JE, Boucheron JA, Clancy DC, Epperly AH, Golden PL. Evans KA, et al. Bioorg Med Chem Lett. 2008 Jul 15;18(14):4068-71. doi: 10.1016/j.bmcl.2008.05.102. Epub 2008 Jun 12. Bioorg Med Chem Lett. 2008. PMID: 18554908

6

Phenoxyacetic acids as PPARδ partial agonists: synthesis, optimization, and in vivo efficacy.

Evans KA, Shearer BG, Wisnoski DD, Shi D, Sparks SM, Sternbach DD, Winegar DA, Billin AN, Britt C, Way JM, Epperly AH, Leesnitzer LM, Merrihew RV, Xu RX, Lambert MH, Jin J. Evans KA, et al. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2345-50. doi: 10.1016/j.bmcl.2011.02.077. Epub 2011 Mar 15. Bioorg Med Chem Lett. 2011. PMID: 21414782

7

Discovery of 3-aryl-4-isoxazolecarboxamides as TGR5 receptor agonists.

Evans KA, Budzik BW, Ross SA, Wisnoski DD, Jin J, Rivero RA, Vimal M, Szewczyk GR, Jayawickreme C, Moncol DL, Rimele TJ, Armour SL, Weaver SP, Griffin RJ, Tadepalli SM, Jeune MR, Shearer TW, Chen ZB, Chen L, Anderson DL, Becherer JD, De Los Frailes M, Colilla FJ. Evans KA, et al. J Med Chem. 2009 Dec 24;52(24):7962-5. doi: 10.1021/jm901434t. J Med Chem. 2009. PMID: 19902954

8

An efficient, asymmetric solid-phase synthesis of benzothiadiazine-substituted tetramic acids: potent inhibitors of the hepatitis C virus RNA-dependent RNA polymerase.

Evans KA, Chai D, Graybill TL, Burton G, Sarisky RT, Lin-Goerke J, Johnston VK, Rivero RA. Evans KA, et al. Bioorg Med Chem Lett. 2006 Apr 15;16(8):2205-8. doi: 10.1016/j.bmcl.2006.01.034. Epub 2006 Feb 7. Bioorg Med Chem Lett. 2006. PMID: 16455253

9

A highly efficient, asymmetric synthesis of benzothiadiazine-substituted tetramic acids: potent inhibitors of hepatitis C virus RNA-dependent RNA polymerase.

Fitch DM, Evans KA, Chai D, Duffy KJ. Fitch DM, et al. Among authors: evans ka. Org Lett. 2005 Nov 24;7(24):5521-4. doi: 10.1021/ol052371w. Org Lett. 2005. PMID: 16288546

10

Novel synthesis of 5-amino-3-bromo-1-(tert-butyl)-1H-pyrazole-4-carbonitrile: a versatile intermediate for the preparation of 5-amino-3-aryl-1-(tert-butyl)-1H-pyrazole-4-carboxamides.

Bobko MA, Kaura AC, Evans KA, Su DS. Bobko MA, et al. Among authors: evans ka. Org Lett. 2012 Aug 3;14(15):3906-8. doi: 10.1021/ol301655f. Epub 2012 Jul 18. Org Lett. 2012. PMID: 22809236

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