Hanessian S - Search Results

1

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

Auzzas L, Larsson A, Matera R, Baraldi A, Deschênes-Simard B, Giannini G, Cabri W, Battistuzzi G, Gallo G, Ciacci A, Vesci L, Pisano C, Hanessian S. Auzzas L, et al. Among authors: hanessian s. J Med Chem. 2010 Dec 9;53(23):8387-99. doi: 10.1021/jm101092u. Epub 2010 Nov 12. J Med Chem. 2010. PMID: 21073160

2

Probing the importance of spacial and conformational domains in captopril analogs for angiotensin converting enzyme activity.

Hanessian S, Reinhold U, Saulnier M, Claridge S. Hanessian S, et al. Bioorg Med Chem Lett. 1998 Aug 18;8(16):2123-8. doi: 10.1016/s0960-894x(98)00377-1. Bioorg Med Chem Lett. 1998. PMID: 9873498

3

Exploration of beta-turn scaffolding motifs as components of sialyl Le(X) mimetics and their relevance to P-selectin.

Hanessian S, Huynh HK, Reddy GV, McNaughton-Smith G, Ernst B, Kolb HC, Magnani J, Sweeley C. Hanessian S, et al. Bioorg Med Chem Lett. 1998 Oct 6;8(19):2803-8. doi: 10.1016/s0960-894x(98)00500-9. Bioorg Med Chem Lett. 1998. PMID: 9873626

4

Asymmetric synthesis of L-azetidine-2-carboxylic acid and 3-substituted congeners--conformationally constrained analogs of phenylalanine, naphthylalanine, and leucine.

Hanessian S, Bernstein N, Yang RY, Maguire R. Hanessian S, et al. Bioorg Med Chem Lett. 1999 May 17;9(10):1437-42. doi: 10.1016/s0960-894x(99)00218-8. Bioorg Med Chem Lett. 1999. PMID: 10360752

5

Picking the S1, S1' and S2' pockets of matrix metalloproteinases. A niche for potent acyclic sulfonamide inhibitors.

Hanessian S, Bouzbouz S, Boudon A, Tucker GC, Peyroulan D. Hanessian S, et al. Bioorg Med Chem Lett. 1999 Jun 21;9(12):1691-6. doi: 10.1016/s0960-894x(99)00259-0. Bioorg Med Chem Lett. 1999. PMID: 10397503

6

Synthesis of a phostone glycomimetic of the endothelin converting enzyme inhibitor phosphoramidon.

Hanessian S, Rogel O. Hanessian S, et al. Bioorg Med Chem Lett. 1999 Aug 16;9(16):2441-6. doi: 10.1016/s0960-894x(99)00401-1. Bioorg Med Chem Lett. 1999. PMID: 10476884

7

Exploring the chiral space within the active site of alpha-thrombin with a constrained mimic of D-Phe-Pro-Arg--design, synthesis, inhibitory activity, and X-ray structure of an enzyme-inhibitor complex.

Hanessian S, Balaux E, Musil D, Olsson LL, Nilsson I. Hanessian S, et al. Bioorg Med Chem Lett. 2000 Feb 7;10(3):243-7. doi: 10.1016/s0960-894x(99)00669-1. Bioorg Med Chem Lett. 2000. PMID: 10698445

8

Design and synthesis of mimics of S-adenosyl-L-homocysteine as potential inhibitors of erythromycin methyltransferases.

Hanessian S, Sgarbi PW. Hanessian S, et al. Bioorg Med Chem Lett. 2000 Mar 6;10(5):433-7. doi: 10.1016/s0960-894x(00)00021-4. Bioorg Med Chem Lett. 2000. PMID: 10743942

9

Design and synthesis of functionalized glycomers as non-peptidic ligands for SH2 binding and as inhibitors of A-431 human epidermoid and HT-29 colon carcinoma cell lines.

Hanessian S, Saavedra OM, Xie F, Amboldi N, Battistini C. Hanessian S, et al. Bioorg Med Chem Lett. 2000 Mar 6;10(5):439-42. doi: 10.1016/s0960-894x(00)00022-6. Bioorg Med Chem Lett. 2000. PMID: 10743943

10

N-Aryl sulfonyl homocysteine hydroxamate inhibitors of matrix metalloproteinases: further probing of the S(1), S(1)', and S(2)' pockets.

Hanessian S, Moitessier N, Gauchet C, Viau M. Hanessian S, et al. J Med Chem. 2001 Sep 13;44(19):3066-73. doi: 10.1021/jm010097f. J Med Chem. 2001. PMID: 11543675

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