Rosenthal PJ - Search Results

1

New cis-configured aziridine-2-carboxylates as aspartic acid protease inhibitors.

Büchold C, Hemberger Y, Heindl C, Welker A, Degel B, Pfeuffer T, Staib P, Schneider S, Rosenthal PJ, Gut J, Morschhäuser J, Bringmann G, Schirmeister T. Büchold C, et al. Among authors: rosenthal pj. ChemMedChem. 2011 Jan 3;6(1):141-52. doi: 10.1002/cmdc.201000370. ChemMedChem. 2011. PMID: 21082722

2

Screening of protease inhibitors as antiplasmodial agents. Part I: Aziridines and epoxides.

Schulz F, Gelhaus C, Degel B, Vicik R, Heppner S, Breuning A, Leippe M, Gut J, Rosenthal PJ, Schirmeister T. Schulz F, et al. Among authors: rosenthal pj. ChemMedChem. 2007 Aug;2(8):1214-24. doi: 10.1002/cmdc.200700070. ChemMedChem. 2007. PMID: 17562535

3

On-bead screening of a combinatorial fumaric acid derived peptide library yields antiplasmodial cysteine protease inhibitors with unusual peptide sequences.

Machon U, Büchold C, Stempka M, Schirmeister T, Gelhaus C, Leippe M, Gut J, Rosenthal PJ, Kisker C, Leyh M, Schmuck C. Machon U, et al. Among authors: rosenthal pj. J Med Chem. 2009 Sep 24;52(18):5662-72. doi: 10.1021/jm900629w. J Med Chem. 2009. PMID: 19715342

4

Michael acceptor based antiplasmodial and antitrypanosomal cysteine protease inhibitors with unusual amino acids.

Breuning A, Degel B, Schulz F, Büchold C, Stempka M, Machon U, Heppner S, Gelhaus C, Leippe M, Leyh M, Kisker C, Rath J, Stich A, Gut J, Rosenthal PJ, Schmuck C, Schirmeister T. Breuning A, et al. Among authors: rosenthal pj. J Med Chem. 2010 Mar 11;53(5):1951-63. doi: 10.1021/jm900946n. J Med Chem. 2010. PMID: 20131843

5

Synthesis and evaluation of non-peptidic cysteine protease inhibitors of P. falciparum derived from etacrynic acid.

Dude MA, Kaeppler U, Herb M, Schiller M, Schulz F, Vedder B, Heppner S, Pradel G, Gut J, Rosenthal PJ, Schirmeister T, Leippe M, Gelhaus C. Dude MA, et al. Among authors: rosenthal pj. Molecules. 2008 Dec 23;14(1):19-35. doi: 10.3390/molecules14010019. Molecules. 2008. PMID: 19104483 Free PMC article.

6

Development of antitrypanosomal and antiplasmodial nonpeptidic cysteine protease inhibitors based on N-protected-guanidino-furan and -pyrrole building blocks.

Langolf S, Machon U, Ehlers M, Sicking W, Schirmeister T, Büchhold C, Gelhaus C, Rosenthal PJ, Schmuck C. Langolf S, et al. Among authors: rosenthal pj. ChemMedChem. 2011 Sep 5;6(9):1581-6. doi: 10.1002/cmdc.201100189. Epub 2011 Jun 15. ChemMedChem. 2011. PMID: 21678556 No abstract available.

7

An endoperoxide-based hybrid approach to deliver falcipain inhibitors inside malaria parasites.

Oliveira R, Newton AS, Guedes RC, Miranda D, Amewu RK, Srivastava A, Gut J, Rosenthal PJ, O'Neill PM, Ward SA, Lopes F, Moreira R. Oliveira R, et al. Among authors: rosenthal pj. ChemMedChem. 2013 Sep;8(9):1528-36. doi: 10.1002/cmdc.201300202. Epub 2013 Jul 12. ChemMedChem. 2013. PMID: 23853126

8

Drug delivery to the malaria parasite using an arterolane-like scaffold.

Fontaine SD, Spangler B, Gut J, Lauterwasser EM, Rosenthal PJ, Renslo AR. Fontaine SD, et al. Among authors: rosenthal pj. ChemMedChem. 2015 Jan;10(1):47-51. doi: 10.1002/cmdc.201402362. Epub 2014 Oct 14. ChemMedChem. 2015. PMID: 25314098 Free PMC article.

9

Enantiopure Indolizinoindolones with in vitro Activity against Blood- and Liver-Stage Malaria Parasites.

Pereira NA, Monteiro Â, Machado M, Gut J, Molins E, Perry MJ, Dourado J, Moreira R, Rosenthal PJ, Prudêncio M, Santos MM. Pereira NA, et al. Among authors: rosenthal pj. ChemMedChem. 2015 Dec;10(12):2080-9. doi: 10.1002/cmdc.201500429. Epub 2015 Nov 3. ChemMedChem. 2015. PMID: 26525306

10

Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites.

Carrasco MP, Machado M, Gonçalves L, Sharma M, Gut J, Lukens AK, Wirth DF, André V, Duarte MT, Guedes RC, Dos Santos DJ, Rosenthal PJ, Mazitschek R, Prudêncio M, Moreira R. Carrasco MP, et al. Among authors: rosenthal pj. ChemMedChem. 2016 Oct 6;11(19):2194-2204. doi: 10.1002/cmdc.201600327. Epub 2016 Aug 19. ChemMedChem. 2016. PMID: 27538856

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