Grazioso G - Search Results

1

Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors.

Pinto A, Conti P, Grazioso G, Tamborini L, Madsen U, Nielsen B, De Micheli C. Pinto A, et al. Among authors: grazioso g. Eur J Med Chem. 2011 Feb;46(2):787-93. doi: 10.1016/j.ejmech.2010.12.020. Epub 2010 Dec 23. Eur J Med Chem. 2011. PMID: 21220180

2

Design, synthesis, and pharmacological characterization of novel, potent NMDA receptor antagonists.

Conti P, De Amici M, Grazioso G, Roda G, Barberis Negra FF, Nielsen B, Stensbøl TB, Madsen U, Bräuner-Osborne H, Frydenvang K, De Sarro G, Toma L, De Micheli C. Conti P, et al. Among authors: grazioso g. J Med Chem. 2004 Dec 30;47(27):6740-8. doi: 10.1021/jm049409f. J Med Chem. 2004. PMID: 15615523

3

Development of a three-dimensional model for the N-methyl-D-aspartate NR2A subunit.

Grazioso G, Moretti L, Scapozza L, De Amici M, De Micheli C. Grazioso G, et al. J Med Chem. 2005 Aug 25;48(17):5489-94. doi: 10.1021/jm050174x. J Med Chem. 2005. PMID: 16107147

4

Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids.

Conti P, De Amici M, Grazioso G, Roda G, Pinto A, Hansen KB, Nielsen B, Madsen U, Bräuner-Osborne H, Egebjerg J, Vestri V, Pellegrini-Giampietro DE, Sibille P, Acher FC, De Micheli C. Conti P, et al. Among authors: grazioso g. J Med Chem. 2005 Oct 6;48(20):6315-25. doi: 10.1021/jm0504499. J Med Chem. 2005. PMID: 16190758

5

Synthesis, chiral resolution, and enantiopharmacology of a potent 2,3-benzodiazepine derivative as noncompetitive AMPA receptor antagonist.

Zappalà M, Postorino G, Micale N, Caccamese S, Parrinello N, Grazioso G, Roda G, Menniti FS, De Sarro G, Grasso S. Zappalà M, et al. Among authors: grazioso g. J Med Chem. 2006 Jan 26;49(2):575-81. doi: 10.1021/jm050552y. J Med Chem. 2006. PMID: 16420043

6

Synthesis of novel N1-substituted bicyclic pyrazole amino acids and evaluation of their interaction with glutamate receptors.

Conti P, Grazioso G, di Ventimiglia SJ, Pinto A, Roda G, Madsen U, Bräuner-Osborne H, Nielsen B, Costagli C, Galli A. Conti P, et al. Among authors: grazioso g. Chem Biodivers. 2005 Jun;2(6):748-57. doi: 10.1002/cbdv.200590052. Chem Biodivers. 2005. PMID: 17192018

7

Synthesis of conformationally constrained glutamic acid homologues and investigation of their pharmacological profiles.

Conti P, Pinto A, Tamborini L, Grazioso G, De Sarro G, Bräuner-Osborne H, Szabo G, Gábor Hársing L, De Micheli C. Conti P, et al. Among authors: grazioso g. ChemMedChem. 2007 Nov;2(11):1639-47. doi: 10.1002/cmdc.200700118. ChemMedChem. 2007. PMID: 17849399

8

Alpha7 nicotinic acetylcholine receptor agonists: prediction of their binding affinity through a molecular mechanics Poisson-Boltzmann surface area approach.

Grazioso G, Cavalli A, De Amici M, Recanatini M, De Micheli C. Grazioso G, et al. J Comput Chem. 2008 Nov 30;29(15):2593-602. doi: 10.1002/jcc.21019. J Comput Chem. 2008. PMID: 18478580

9

New analogues of epiboxidine incorporating the 4,5-dihydroisoxazole nucleus: synthesis, binding affinity at neuronal nicotinic acetylcholine receptors, and molecular modeling investigations.

Dallanoce C, Magrone P, Bazza P, Grazioso G, Rizzi L, Riganti L, Gotti C, Clementi F, Frydenvang K, De Amici M. Dallanoce C, et al. Among authors: grazioso g. Chem Biodivers. 2009 Feb;6(2):244-59. doi: 10.1002/cbdv.200800077. Chem Biodivers. 2009. PMID: 19235154

10

Insights into docking and scoring neuronal alpha4beta2 nicotinic receptor agonists using molecular dynamics simulations and QM/MM calculations.

Sgrignani J, Bonaccini C, Grazioso G, Chioccioli M, Cavalli A, Gratteri P. Sgrignani J, et al. Among authors: grazioso g. J Comput Chem. 2009 Nov 30;30(15):2443-54. doi: 10.1002/jcc.21251. J Comput Chem. 2009. PMID: 19360794

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