Tuccinardi T - Search Results

1

Discovery of N-hydroxyindole-based inhibitors of human lactate dehydrogenase isoform A (LDH-A) as starvation agents against cancer cells.

Granchi C, Roy S, Giacomelli C, Macchia M, Tuccinardi T, Martinelli A, Lanza M, Betti L, Giannaccini G, Lucacchini A, Funel N, León LG, Giovannetti E, Peters GJ, Palchaudhuri R, Calvaresi EC, Hergenrother PJ, Minutolo F. Granchi C, et al. Among authors: tuccinardi t. J Med Chem. 2011 Mar 24;54(6):1599-612. doi: 10.1021/jm101007q. Epub 2011 Feb 18. J Med Chem. 2011. PMID: 21332213

2

Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives.

Ferrarini PL, Betti L, Cavallini T, Giannaccini G, Lucacchini A, Manera C, Martinelli A, Ortore G, Saccomanni G, Tuccinardi T. Ferrarini PL, et al. Among authors: tuccinardi t. J Med Chem. 2004 Jun 3;47(12):3019-31. doi: 10.1021/jm030977p. J Med Chem. 2004. PMID: 15163184

3

A new development of matrix metalloproteinase inhibitors: twin hydroxamic acids as potent inhibitors of MMPs.

Rossello A, Nuti E, Catalani MP, Carelli P, Orlandini E, Rapposelli S, Tuccinardi T, Atkinson SJ, Murphy G, Balsamo A. Rossello A, et al. Among authors: tuccinardi t. Bioorg Med Chem Lett. 2005 May 2;15(9):2311-4. doi: 10.1016/j.bmcl.2005.03.002. Bioorg Med Chem Lett. 2005. PMID: 15837315

4

1,8-Naphthyridin-4-one derivatives as new ligands of A2A adenosine receptors.

Manera C, Betti L, Cavallini T, Giannaccini G, Martinelli A, Ortore G, Saccomanni G, Trincavelli L, Tuccinardi T, Ferrarini PL. Manera C, et al. Among authors: tuccinardi t. Bioorg Med Chem Lett. 2005 Oct 15;15(20):4604-10. doi: 10.1016/j.bmcl.2005.06.064. Bioorg Med Chem Lett. 2005. PMID: 16099648

5

Adenosine receptor modelling. A1/A2a selectivity.

Tuccinardi T, Ortore G, Manera C, Saccomanni G, Martinelli A. Tuccinardi T, et al. Eur J Med Chem. 2006 Mar;41(3):321-9. doi: 10.1016/j.ejmech.2005.09.011. Epub 2006 Jan 19. Eur J Med Chem. 2006. PMID: 16427161

6

Cannabinoid CB2/CB1 selectivity. Receptor modeling and automated docking analysis.

Tuccinardi T, Ferrarini PL, Manera C, Ortore G, Saccomanni G, Martinelli A. Tuccinardi T, et al. J Med Chem. 2006 Feb 9;49(3):984-94. doi: 10.1021/jm050875u. J Med Chem. 2006. PMID: 16451064

7

A theoretical study to investigate D2DAR/D4DAR selectivity: receptor modeling and molecular docking of dopaminergic ligands.

Ortore G, Tuccinardi T, Bertini S, Martinelli A. Ortore G, et al. Among authors: tuccinardi t. J Med Chem. 2006 Feb 23;49(4):1397-407. doi: 10.1021/jm051046b. J Med Chem. 2006. PMID: 16480275

8

Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides.

Tuccinardi T, Martinelli A, Nuti E, Carelli P, Balzano F, Uccello-Barretta G, Murphy G, Rossello A. Tuccinardi T, et al. Bioorg Med Chem. 2006 Jun 15;14(12):4260-76. doi: 10.1016/j.bmc.2006.01.056. Epub 2006 Feb 17. Bioorg Med Chem. 2006. PMID: 16483784

9

Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models.

Tafi A, Bernardini C, Botta M, Corelli F, Andreini M, Martinelli A, Ortore G, Baraldi PG, Fruttarolo F, Borea PA, Tuccinardi T. Tafi A, et al. Among authors: tuccinardi t. J Med Chem. 2006 Jul 13;49(14):4085-97. doi: 10.1021/jm051112+. J Med Chem. 2006. PMID: 16821770

10

Proposal of a new binding orientation for non-peptide AT1 antagonists: homology modeling, docking and three-dimensional quantitative structure-activity relationship analysis.

Tuccinardi T, Calderone V, Rapposelli S, Martinelli A. Tuccinardi T, et al. J Med Chem. 2006 Jul 13;49(14):4305-16. doi: 10.1021/jm060338p. J Med Chem. 2006. PMID: 16821790

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

223 results

Search Page

Filters