Aso K - Search Results

1

Melanin-concentrating hormone receptor 1 antagonists: synthesis, structure-activity relationship, docking studies, and biological evaluation of 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives.

Kasai S, Kamaura M, Kamata M, Aso K, Ogino H, Nakano Y, Watanabe K, Kaisho T, Tawada M, Nagisa Y, Takekawa S, Kato K, Suzuki N, Ishihara Y. Kasai S, et al. Among authors: aso k. Bioorg Med Chem. 2011 Nov 1;19(21):6261-73. doi: 10.1016/j.bmc.2011.09.007. Epub 2011 Sep 10. Bioorg Med Chem. 2011. PMID: 21975069

2

Discovery, synthesis and biological evaluation of isoquinolones as novel and highly selective JNK inhibitors (1).

Asano Y, Kitamura S, Ohra T, Aso K, Igata H, Tamura T, Kawamoto T, Tanaka T, Sogabe S, Matsumoto S, Yamaguchi M, Kimura H, Itoh F. Asano Y, et al. Among authors: aso k. Bioorg Med Chem. 2008 Apr 15;16(8):4715-32. doi: 10.1016/j.bmc.2008.02.027. Epub 2008 Feb 13. Bioorg Med Chem. 2008. PMID: 18313304

3

Discovery of pyrrolo[2,3-d]pyrimidin-4-ones as corticotropin-releasing factor 1 receptor antagonists with a carbonyl-based hydrogen bonding acceptor.

Aso K, Kobayashi K, Mochizuki M, Kanzaki N, Sako Y, Yano T. Aso K, et al. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2365-71. doi: 10.1016/j.bmcl.2011.02.086. Epub 2011 Feb 26. Bioorg Med Chem Lett. 2011. PMID: 21414781

4

Structure-Based Design and Synthesis of 3-Amino-1,5-dihydro-4H-pyrazolopyridin-4-one Derivatives as Tyrosine Kinase 2 Inhibitors.

Yogo T, Nagamiya H, Seto M, Sasaki S, Shih-Chung H, Ohba Y, Tokunaga N, Lee GN, Rhim CY, Yoon CH, Cho SY, Skene R, Yamamoto S, Satou Y, Kuno M, Miyazaki T, Nakagawa H, Okabe A, Marui S, Aso K, Yoshida M. Yogo T, et al. Among authors: aso k. J Med Chem. 2016 Jan 28;59(2):733-49. doi: 10.1021/acs.jmedchem.5b01857. Epub 2016 Jan 8. J Med Chem. 2016. PMID: 26701356

5

Design and Synthesis of Benzimidazoles As Novel Corticotropin-Releasing Factor 1 Receptor Antagonists.

Mochizuki M, Kori M, Kobayashi K, Yano T, Sako Y, Tanaka M, Kanzaki N, Gyorkos AC, Corrette CP, Cho SY, Pratt SA, Aso K. Mochizuki M, et al. Among authors: aso k. J Med Chem. 2016 Mar 24;59(6):2551-66. doi: 10.1021/acs.jmedchem.5b01715. Epub 2016 Mar 7. J Med Chem. 2016. PMID: 26901666

6

Discovery of a 7-arylaminobenzimidazole series as novel CRF1 receptor antagonists.

Mochizuki M, Kori M, Kono M, Yano T, Sako Y, Tanaka M, Kanzaki N, Gyorkos AC, Corrette CP, Aso K. Mochizuki M, et al. Among authors: aso k. Bioorg Med Chem. 2016 Oct 1;24(19):4675-4691. doi: 10.1016/j.bmc.2016.08.005. Epub 2016 Aug 4. Bioorg Med Chem. 2016. PMID: 27567079

7

Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF₁ receptor antagonist.

Mochizuki M, Kojima T, Kobayashi K, Kotani E, Ishichi Y, Kanzaki N, Nakagawa H, Okuda T, Kosugi Y, Yano T, Sako Y, Tanaka M, Aso K. Mochizuki M, et al. Among authors: aso k. Bioorg Med Chem. 2017 Mar 1;25(5):1556-1570. doi: 10.1016/j.bmc.2016.11.011. Epub 2016 Nov 8. Bioorg Med Chem. 2017. PMID: 28174066

8

Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists.

Tokumaru K, Ito Y, Nomura I, Nakahata T, Shimizu Y, Kurimoto E, Aoyama K, Aso K. Tokumaru K, et al. Among authors: aso k. Bioorg Med Chem. 2017 Jun 15;25(12):3098-3115. doi: 10.1016/j.bmc.2017.03.064. Epub 2017 Apr 1. Bioorg Med Chem. 2017. PMID: 28433511

9

Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists.

Kojima T, Mochizuki M, Takai T, Hoashi Y, Morimoto S, Seto M, Nakamura M, Kobayashi K, Sako Y, Tanaka M, Kanzaki N, Kosugi Y, Yano T, Aso K. Kojima T, et al. Among authors: aso k. Bioorg Med Chem. 2018 May 15;26(9):2229-2250. doi: 10.1016/j.bmc.2018.01.020. Epub 2018 Feb 8. Bioorg Med Chem. 2018. PMID: 29459145

10

Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists.

Nakahata T, Tokumaru K, Ito Y, Ishii N, Setoh M, Shimizu Y, Harasawa T, Aoyama K, Hamada T, Kori M, Aso K. Nakahata T, et al. Among authors: aso k. Bioorg Med Chem. 2018 May 1;26(8):1598-1608. doi: 10.1016/j.bmc.2018.02.005. Epub 2018 Feb 10. Bioorg Med Chem. 2018. PMID: 29478803

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

484 results

Search Page

Filters