Medda F - Search Results

1

Facile and rapid route for the synthesis of novel conformationally constrained norstatine analogs via PADAM-cyclization methodology.

Shaw AY, Medda F, Hulme C. Shaw AY, et al. Among authors: medda f. Tetrahedron Lett. 2012 Mar 14;53(11):1313-1315. doi: 10.1016/j.tetlet.2011.12.073. Tetrahedron Lett. 2012. PMID: 22368307 Free PMC article.

2

Exploiting the Divalent Nature of Isonitriles: a novel Pictet-Spengler Amidination process.

Medda F, Hulme C. Medda F, et al. Tetrahedron Lett. 2014 May 1;55(22):3328-3331. doi: 10.1016/j.tetlet.2014.04.043. Tetrahedron Lett. 2014. PMID: 24954960 Free PMC article.

3

Synthesis and biological activity of 2-aminothiazoles as novel inhibitors of PGE2 production in cells.

Smith B, Chang HH, Medda F, Gokhale V, Dietrich J, Davis A, Meuillet EJ, Hulme C. Smith B, et al. Among authors: medda f. Bioorg Med Chem Lett. 2012 May 15;22(10):3567-70. doi: 10.1016/j.bmcl.2012.03.013. Epub 2012 Mar 28. Bioorg Med Chem Lett. 2012. PMID: 22516282 Free PMC article.

4

Synthesis and biological activity of aminophthalazines and aminopyridazines as novel inhibitors of PGE2 production in cells.

Medda F, Sells E, Chang HH, Dietrich J, Chappeta S, Smith B, Gokhale V, Meuillet EJ, Hulme C. Medda F, et al. Bioorg Med Chem Lett. 2013 Jan 15;23(2):528-31. doi: 10.1016/j.bmcl.2012.11.030. Epub 2012 Nov 21. Bioorg Med Chem Lett. 2013. PMID: 23237838 Free PMC article.

5

Recent advances in the design, synthesis, and biological evaluation of selective DYRK1A inhibitors: a new avenue for a disease modifying treatment of Alzheimer's?

Smith B, Medda F, Gokhale V, Dunckley T, Hulme C. Smith B, et al. Among authors: medda f. ACS Chem Neurosci. 2012 Nov 21;3(11):857-72. doi: 10.1021/cn300094k. Epub 2012 Aug 28. ACS Chem Neurosci. 2012. PMID: 23173067 Free PMC article. Review.

6

3-(4-Bromo-phen-yl)-1-butyl-5-[1-(2-chloro-6-methyl-phen-yl)-1H-tetra-zol-5-yl]imidazolidine-2,4-dione.

Hall GB, Medda F, Roberts SA, Hulme C. Hall GB, et al. Among authors: medda f. Acta Crystallogr Sect E Struct Rep Online. 2013 Jun 15;69(Pt 7):o1102-3. doi: 10.1107/S1600536813016000. eCollection 2013. Acta Crystallogr Sect E Struct Rep Online. 2013. PMID: 24046663 Free PMC article.

7

Synthesis of diverse nitrogen-enriched heterocyclic scaffolds using a suite of tunable one-pot multicomponent reactions.

Martinez-Ariza G, Ayaz M, Medda F, Hulme C. Martinez-Ariza G, et al. Among authors: medda f. J Org Chem. 2014 Jun 6;79(11):5153-62. doi: 10.1021/jo500723d. Epub 2014 May 19. J Org Chem. 2014. PMID: 24788091 Free PMC article.

8

Novel cambinol analogs as sirtuin inhibitors: synthesis, biological evaluation, and rationalization of activity.

Medda F, Russell RJ, Higgins M, McCarthy AR, Campbell J, Slawin AM, Lane DP, Lain S, Westwood NJ. Medda F, et al. J Med Chem. 2009 May 14;52(9):2673-82. doi: 10.1021/jm8014298. J Med Chem. 2009. PMID: 19419202 Free PMC article.

9

DYRK1A inhibition as potential treatment for Alzheimer's disease.

Stotani S, Giordanetto F, Medda F. Stotani S, et al. Among authors: medda f. Future Med Chem. 2016 Apr;8(6):681-96. doi: 10.4155/fmc-2016-0013. Epub 2016 Apr 13. Future Med Chem. 2016. PMID: 27073990 Review.

10

Inhibitors to Overcome Secondary Mutations in the Stem Cell Factor Receptor KIT.

Kaitsiotou H, Keul M, Hardick J, Mühlenberg T, Ketzer J, Ehrt C, Krüll J, Medda F, Koch O, Giordanetto F, Bauer S, Rauh D. Kaitsiotou H, et al. Among authors: medda f. J Med Chem. 2017 Nov 9;60(21):8801-8815. doi: 10.1021/acs.jmedchem.7b00841. Epub 2017 Oct 24. J Med Chem. 2017. PMID: 28991465

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