Matesanz R - Search Results

1

Zampanolide, a potent new microtubule-stabilizing agent, covalently reacts with the taxane luminal site in tubulin α,β-heterodimers and microtubules.

Field JJ, Pera B, Calvo E, Canales A, Zurwerra D, Trigili C, Rodríguez-Salarichs J, Matesanz R, Kanakkanthara A, Wakefield SJ, Singh AJ, Jiménez-Barbero J, Northcote P, Miller JH, López JA, Hamel E, Barasoain I, Altmann KH, Díaz JF. Field JJ, et al. Among authors: matesanz r. Chem Biol. 2012 Jun 22;19(6):686-98. doi: 10.1016/j.chembiol.2012.05.008. Chem Biol. 2012. PMID: 22726683 Free PMC article.

2

Cyclostreptin binds covalently to microtubule pores and lumenal taxoid binding sites.

Buey RM, Calvo E, Barasoain I, Pineda O, Edler MC, Matesanz R, Cerezo G, Vanderwal CD, Day BW, Sorensen EJ, López JA, Andreu JM, Hamel E, Díaz JF. Buey RM, et al. Among authors: matesanz r. Nat Chem Biol. 2007 Feb;3(2):117-25. doi: 10.1038/nchembio853. Epub 2007 Jan 7. Nat Chem Biol. 2007. PMID: 17206139 Free article.

3

Overcoming tumor drug resistance with high-affinity taxanes: a SAR study of C2-modified 7-acyl-10-deacetyl cephalomannines.

Yang CG, Barasoain I, Li X, Matesanz R, Liu R, Sharom FJ, Yin DL, Díaz JF, Fang WS. Yang CG, et al. Among authors: matesanz r. ChemMedChem. 2007 May;2(5):691-701. doi: 10.1002/cmdc.200700002. ChemMedChem. 2007. PMID: 17385753

4

Synthesis, biological evaluations, and tubulin binding poses of C-2alpha sulfur linked taxol analogues.

Wang L, Alcaraz AA, Matesanz R, Yang CG, Barasoain I, Díaz JF, Li YZ, Snyder JP, Fang WS. Wang L, et al. Among authors: matesanz r. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3191-4. doi: 10.1016/j.bmcl.2007.03.026. Epub 2007 Mar 14. Bioorg Med Chem Lett. 2007. PMID: 17395465

5

Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studies.

La Regina G, Edler MC, Brancale A, Kandil S, Coluccia A, Piscitelli F, Hamel E, De Martino G, Matesanz R, Díaz JF, Scovassi AI, Prosperi E, Lavecchia A, Novellino E, Artico M, Silvestri R. La Regina G, et al. Among authors: matesanz r. J Med Chem. 2007 Jun 14;50(12):2865-74. doi: 10.1021/jm061479u. Epub 2007 May 12. J Med Chem. 2007. PMID: 17497841

6

The total synthesis and biological properties of the cytotoxic macrolide FD-891 and its non-natural (Z)-C12 isomer.

García-Fortanet J, Murga J, Carda M, Marco JA, Matesanz R, Díaz JF, Barasoain I. García-Fortanet J, et al. Among authors: matesanz r. Chemistry. 2007;13(18):5060-74. doi: 10.1002/chem.200700342. Chemistry. 2007. PMID: 17516610

7

The bound conformation of microtubule-stabilizing agents: NMR insights into the bioactive 3D structure of discodermolide and dictyostatin.

Canales A, Matesanz R, Gardner NM, Andreu JM, Paterson I, Díaz JF, Jiménez-Barbero J. Canales A, et al. Among authors: matesanz r. Chemistry. 2008;14(25):7557-69. doi: 10.1002/chem.200800039. Chemistry. 2008. PMID: 18449868

8

Optimization of taxane binding to microtubules: binding affinity dissection and incremental construction of a high-affinity analog of paclitaxel.

Matesanz R, Barasoain I, Yang CG, Wang L, Li X, de Inés C, Coderch C, Gago F, Barbero JJ, Andreu JM, Fang WS, Díaz JF. Matesanz R, et al. Chem Biol. 2008 Jun;15(6):573-85. doi: 10.1016/j.chembiol.2008.05.008. Chem Biol. 2008. PMID: 18559268

9

Synthesis and biological activities of high affinity taxane-based fluorescent probes.

Li X, Barasoain I, Matesanz R, Díaz JF, Fang WS. Li X, et al. Among authors: matesanz r. Bioorg Med Chem Lett. 2009 Feb 1;19(3):751-4. doi: 10.1016/j.bmcl.2008.12.018. Epub 2008 Dec 10. Bioorg Med Chem Lett. 2009. PMID: 19128972

10

Epothilone analogues with benzimidazole and quinoline side chains: chemical synthesis, antiproliferative activity, and interactions with tubulin.

Dietrich SA, Lindauer R, Stierlin C, Gertsch J, Matesanz R, Notararigo S, Díaz JF, Altmann KH. Dietrich SA, et al. Among authors: matesanz r. Chemistry. 2009 Oct 5;15(39):10144-57. doi: 10.1002/chem.200901376. Chemistry. 2009. PMID: 19697384

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