Cheung AW - Search Results

1

7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors.

Cheung AW, Banner B, Bose J, Kim K, Li S, Marcopulos N, Orzechowski L, Sergi JA, Thakkar KC, Wang BB, Yun W, Zwingelstein C, Berthel S, Olivier AR. Cheung AW, et al. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7518-22. doi: 10.1016/j.bmcl.2012.10.035. Epub 2012 Oct 16. Bioorg Med Chem Lett. 2012. PMID: 23122867

2

Discovery of benzothiazole-based adenosine A2B receptor antagonists with improved A2A selectivity.

Firooznia F, Cheung AW, Brinkman J, Grimsby J, Gubler ML, Hamid R, Marcopulos N, Ramsey G, Tan J, Wen Y, Sarabu R. Firooznia F, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2011 Apr 1;21(7):1933-6. doi: 10.1016/j.bmcl.2011.02.053. Epub 2011 Feb 17. Bioorg Med Chem Lett. 2011. PMID: 21388809

3

4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: drug-like and non-xanthine based A2B adenosine receptor antagonists.

Cheung AW, Brinkman J, Firooznia F, Flohr A, Grimsby J, Gubler ML, Guertin K, Hamid R, Marcopulos N, Norcross RD, Qi L, Ramsey G, Tan J, Wen Y, Sarabu R. Cheung AW, et al. Bioorg Med Chem Lett. 2010 Jul 15;20(14):4140-6. doi: 10.1016/j.bmcl.2010.05.056. Epub 2010 May 20. Bioorg Med Chem Lett. 2010. PMID: 20541935

4

Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the potential treatment of obesity and diabetes.

Qian Y, Wertheimer SJ, Ahmad M, Cheung AW, Firooznia F, Hamilton MM, Hayden S, Li S, Marcopulos N, McDermott L, Tan J, Yun W, Guo L, Pamidimukkala A, Chen Y, Huang KS, Ramsey GB, Whittard T, Conde-Knape K, Taub R, Rondinone CM, Tilley J, Bolin D. Qian Y, et al. Among authors: cheung aw. J Med Chem. 2011 Apr 14;54(7):2433-46. doi: 10.1021/jm101580m. Epub 2011 Mar 17. J Med Chem. 2011. PMID: 21413799

5

A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptides.

Sun H, Greeley DN, Chu XJ, Cheung A, Danho W, Swistok J, Wang Y, Zhao C, Chen L, Fry DC. Sun H, et al. Bioorg Med Chem. 2004 May 15;12(10):2671-7. doi: 10.1016/j.bmc.2004.03.017. Bioorg Med Chem. 2004. PMID: 15110848

6

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: histidine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Jan 6;13(1):133-7. doi: 10.1016/s0960-894x(02)00830-2. Bioorg Med Chem Lett. 2003. PMID: 12467633

7

Preparation of human Melanocortin-4 receptor agonist libraries: linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2.

Cheung AW, Qi L, Gore V, Chu XJ, Bartkovitz D, Kurylko G, Swistok J, Danho W, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5504-8. doi: 10.1016/j.bmcl.2005.08.083. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16203134

8

Structure-activity relationship of cyclic peptide penta-c[Asp-His(6)-DPhe(7)-Arg(8)-Trp(9)-Lys]-NH(2) at the human melanocortin-1 and -4 receptors: His(6) substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Apr 7;13(7):1307-11. doi: 10.1016/s0960-894x(03)00114-8. Bioorg Med Chem Lett. 2003. PMID: 12657270

9

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: arginine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Franco L, Yagaloff K, Chen L. Cheung AW, et al. Bioorg Med Chem Lett. 2002 Sep 2;12(17):2407-10. doi: 10.1016/s0960-894x(02)00459-6. Bioorg Med Chem Lett. 2002. PMID: 12161144

10

Structure-activity relationship of linear peptide Bu-His6-DPhe7-Arg8-Trp9-Gly10-NH2 at the human melanocortin-1 and -4 receptors: DPhe7 and Trp9 substitution.

Danho W, Swistok J, Cheung AW, Kurylko G, Franco L, Chu XJ, Chen L, Yagaloff K. Danho W, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2003 Feb 24;13(4):649-52. doi: 10.1016/s0960-894x(02)01052-1. Bioorg Med Chem Lett. 2003. PMID: 12639550

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