Winum JY - Search Results

1

3-Halo-3-nitro-aza/thioflavanones: DNMT inhibitors with a two-site binding mode in the hDNMT3A catalytic pocket.

Serhouni A, Calzaferri F, Bessina Y, van der Lee A, Arimondo PB, Louet M, Winum JY, Lopez M. Serhouni A, et al. Among authors: winum jy. Bioorg Med Chem. 2024 Nov 28;118:117988. doi: 10.1016/j.bmc.2024.117988. Online ahead of print. Bioorg Med Chem. 2024. PMID: 39689413 Free article.

2

Novel anticancer drug discovery strategies targeting hypoxia-inducible factors.

Mustafa M, Rashed M, Winum JY. Mustafa M, et al. Among authors: winum jy. Expert Opin Drug Discov. 2025 Jan;20(1):103-121. doi: 10.1080/17460441.2024.2442739. Epub 2024 Dec 17. Expert Opin Drug Discov. 2025. PMID: 39670847 Review.

3

Exploring the binding mode of phenyl and vinyl boronic acids to human carbonic anhydrases.

Esposito D, Monti SM, Supuran CT, Winum JY, De Simone G, Alterio V. Esposito D, et al. Among authors: winum jy. Int J Biol Macromol. 2024 Dec;282(Pt 2):136873. doi: 10.1016/j.ijbiomac.2024.136873. Epub 2024 Oct 23. Int J Biol Macromol. 2024. PMID: 39454912 Free article.

4

Benzoxaborinine, New Chemotype for Carbonic Anhydrase Inhibition: Ex Novo Synthesis, Crystallography, In Silico Studies, and Anti-Melanoma Cell Line Activity.

Giovannuzzi S, Nikitjuka A, Angeli A, Smietana M, Massardi ML, Turati M, Ronca R, Bonardi A, Nocentini A, Ferraroni M, Supuran CT, Winum JY. Giovannuzzi S, et al. Among authors: winum jy. J Med Chem. 2024 Oct 24;67(20):18221-18234. doi: 10.1021/acs.jmedchem.4c01516. Epub 2024 Oct 8. J Med Chem. 2024. PMID: 39378331

5

Photodynamic therapy alone or in combination to counteract bacterial infections.

Clément S, Winum JY. Clément S, et al. Among authors: winum jy. Expert Opin Ther Pat. 2024 Jun;34(6):401-414. doi: 10.1080/13543776.2024.2327308. Epub 2024 Mar 11. Expert Opin Ther Pat. 2024. PMID: 38439633 Review.

6

Boron-containing carbonic anhydrases inhibitors.

Giovannuzzi S, Nikitjuka A, Pereira Resende BR, Smietana M, Nocentini A, Supuran CT, Winum JY. Giovannuzzi S, et al. Among authors: winum jy. Bioorg Chem. 2024 Feb;143:106976. doi: 10.1016/j.bioorg.2023.106976. Epub 2023 Nov 19. Bioorg Chem. 2024. PMID: 38000350 Review.

7

Are tumour-associated carbonic anhydrases genuine therapeutic targets for photodynamic therapy?

Merabti A, Richeter S, Supuran CT, Clement S, Winum JY. Merabti A, et al. Among authors: winum jy. Expert Opin Ther Targets. 2023 Jul-Dec;27(9):817-826. doi: 10.1080/14728222.2023.2255380. Epub 2023 Sep 13. Expert Opin Ther Targets. 2023. PMID: 37668158 Review.

8

6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography.

Nocentini A, Bonardi A, Bazzicalupi C, Alterio V, Esposito D, Monti SM, Smietana M, De Simone G, Supuran CT, Gratteri P, Winum JY. Nocentini A, et al. Among authors: winum jy. J Med Chem. 2023 Jun 22;66(12):8118-8129. doi: 10.1021/acs.jmedchem.3c00433. Epub 2023 Jun 7. J Med Chem. 2023. PMID: 37283561

9

The importance of sulfur-containing motifs in drug design and discovery.

Mustafa M, Winum JY. Mustafa M, et al. Among authors: winum jy. Expert Opin Drug Discov. 2022 May;17(5):501-512. doi: 10.1080/17460441.2022.2044783. Epub 2022 Feb 25. Expert Opin Drug Discov. 2022. PMID: 35193437

10

1,5-Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors.

Ismail C, Nocentini A, Supuran CT, Winum JY, Gharbi R. Ismail C, et al. Among authors: winum jy. Arch Pharm (Weinheim). 2022 Mar;355(3):e2100405. doi: 10.1002/ardp.202100405. Epub 2021 Dec 3. Arch Pharm (Weinheim). 2022. PMID: 34862650

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