Brickmann K - Search Results

1

5-alkyl-1,3-oxazole derivatives of 6-amino-nicotinic acids as alkyl ester bioisosteres are antagonists of the P2Y12 receptor.

Bach P, Boström J, Brickmann K, Burgess LE, Clarke D, Groneberg RD, Harvey DM, Laird ER, O'Sullivan M, Zetterberg F. Bach P, et al. Among authors: brickmann k. Future Med Chem. 2013 Nov;5(17):2037-56. doi: 10.4155/fmc.13.171. Future Med Chem. 2013. PMID: 24215345

2

Synthesis, structure-property relationships and pharmacokinetic evaluation of ethyl 6-aminonicotinate sulfonylureas as antagonists of the P2Y₁₂ receptor.

Bach P, Boström J, Brickmann K, van Giezen JJ, Groneberg RD, Harvey DM, O'Sullivan M, Zetterberg F. Bach P, et al. Among authors: brickmann k. Eur J Med Chem. 2013 Jul;65:360-75. doi: 10.1016/j.ejmech.2013.04.007. Epub 2013 May 15. Eur J Med Chem. 2013. PMID: 23747805

3

A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y12 receptor.

Bach P, Boström J, Brickmann K, van Giezen JJ, Hovland R, Petersson AU, Ray A, Zetterberg F. Bach P, et al. Among authors: brickmann k. Bioorg Med Chem Lett. 2011 May 15;21(10):2877-81. doi: 10.1016/j.bmcl.2011.03.088. Epub 2011 Mar 30. Bioorg Med Chem Lett. 2011. PMID: 21507636

4

Design of small molecule inhibitors of acetyl-CoA carboxylase 1 and 2 showing reduction of hepatic malonyl-CoA levels in vivo in obese Zucker rats.

Bengtsson C, Blaho S, Saitton DB, Brickmann K, Broddefalk J, Davidsson O, Drmota T, Folmer R, Hallberg K, Hallén S, Hovland R, Isin E, Johannesson P, Kull B, Larsson LO, Löfgren L, Nilsson KE, Noeske T, Oakes N, Plowright AT, Schnecke V, Ståhlberg P, Sörme P, Wan H, Wellner E, Oster L. Bengtsson C, et al. Among authors: brickmann k. Bioorg Med Chem. 2011 May 15;19(10):3039-53. doi: 10.1016/j.bmc.2011.04.014. Epub 2011 Apr 13. Bioorg Med Chem. 2011. PMID: 21515056

5

Conformations and receptor activity of desmopressin analogues, which contain gamma-turn mimetics or a psi[CH(2)O] isostere.

Hedenström M, Yuan Z, Brickmann K, Carlsson J, Ekholm K, Johansson B, Kreutz E, Nilsson A, Sethson I, Kihlberg J. Hedenström M, et al. Among authors: brickmann k. J Med Chem. 2002 Jun 6;45(12):2501-11. doi: 10.1021/jm011073b. J Med Chem. 2002. PMID: 12036358

6

Synthesis and pharmacological evaluation of an analogue of the peptide hormone oxytocin that contains a mimetic of an inverse gamma-turn.

Yuan Z, Blomberg D, Sethson I, Brickmann K, Ekholm K, Johansson B, Nilsson A, Kihlberg J. Yuan Z, et al. Among authors: brickmann k. J Med Chem. 2002 Jun 6;45(12):2512-9. doi: 10.1021/jm0110744. J Med Chem. 2002. PMID: 12036359

7

Synthesis and conformational studies of a beta-turn mimetic incorporated in Leu-enkephalin.

Blomberg D, Hedenström M, Kreye P, Sethson I, Brickmann K, Kihlberg J. Blomberg D, et al. Among authors: brickmann k. J Org Chem. 2004 May 14;69(10):3500-8. doi: 10.1021/jo0356863. J Org Chem. 2004. PMID: 15132562

8

Design, synthesis and biological evaluation of thrombin inhibitors based on a pyridine scaffold.

Blomberg D, Fex T, Xue Y, Brickmann K, Kihlberg J. Blomberg D, et al. Among authors: brickmann k. Org Biomol Chem. 2007 Aug 21;5(16):2599-605. doi: 10.1039/b705344d. Org Biomol Chem. 2007. PMID: 18019535

9

Synthesis and biological evaluation of leucine enkephalin turn mimetics.

Blomberg D, Kreye P, Fowler C, Brickmann K, Kihlberg J. Blomberg D, et al. Among authors: brickmann k. Org Biomol Chem. 2006 Feb 7;4(3):416-23. doi: 10.1039/b515618a. Epub 2006 Jan 9. Org Biomol Chem. 2006. PMID: 16446799

10

The Value of Median Nerve Sonography as a Predictor for Short- and Long-Term Clinical Outcomes in Patients with Carpal Tunnel Syndrome: A Prospective Long-Term Follow-Up Study.

Marschall A, Ficjian A, Stradner MH, Husic R, Zauner D, Seel W, Simmet NE, Klammer A, Heizer P, Brickmann K, Gretler J, Fürst-Moazedi FC, Thonhofer R, Hermann J, Graninger WB, Quasthoff S, Dejaco C. Marschall A, et al. Among authors: brickmann k. PLoS One. 2016 Sep 23;11(9):e0162288. doi: 10.1371/journal.pone.0162288. eCollection 2016. PLoS One. 2016. PMID: 27662617 Free PMC article.

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