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Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2.
ACS Med Chem Lett. 2012 Oct 19;3(12):1091-6. doi: 10.1021/ml3003346. eCollection 2012 Dec 13.
ACS Med Chem Lett. 2012.
PMID: 24900432
Free PMC article.
Cell-Based Drug Discovery: Identification and Optimization of Small Molecules that Reduce c-MYC Protein Levels in Cells.
Medina JR, Tian X, Li WH, Suarez D, Mack JF, LaFrance L, Martyr C, Brackley J, Di Marco C, Rivero R, Heerding DA, McHugh C, Minthorn E, Bhaskar A, Rubin J, Butticello M, Carpenter C, Nartey EN, Berrodin TJ, Kallal LA, Mangatt B.
Medina JR, et al.
J Med Chem. 2021 Nov 11;64(21):16056-16087. doi: 10.1021/acs.jmedchem.1c01416. Epub 2021 Oct 20.
J Med Chem. 2021.
PMID: 34669409
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Substituted dipiperidine alcohols as potent CCR2 antagonists.
Xia M, Hou C, Demong D, Pollack S, Pan M, Brackley J, Singer M, Matheis M, Cavender D, Wachter M.
Xia M, et al.
Bioorg Med Chem Lett. 2008 Jun 15;18(12):3562-4. doi: 10.1016/j.bmcl.2008.05.010. Epub 2008 May 4.
Bioorg Med Chem Lett. 2008.
PMID: 18487045
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Synthesis, structure-activity relationship and in vivo antiinflammatory efficacy of substituted dipiperidines as CCR2 antagonists.
Xia M, Hou C, DeMong DE, Pollack SR, Pan M, Brackley JA, Jain N, Gerchak C, Singer M, Malaviya R, Matheis M, Olini G, Cavender D, Wachter M.
Xia M, et al. Among authors: brackley ja.
J Med Chem. 2007 Nov 15;50(23):5561-3. doi: 10.1021/jm070902b. Epub 2007 Oct 11.
J Med Chem. 2007.
PMID: 17929797
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Synthesis and biological evaluation of phenyl piperidine derivatives as CCR2 antagonists.
Xia M, Hou C, Pollack S, Brackley J, DeMong D, Pan M, Singer M, Matheis M, Olini G, Cavender D, Wachter M.
Xia M, et al.
Bioorg Med Chem Lett. 2007 Nov 1;17(21):5964-8. doi: 10.1016/j.bmcl.2007.07.065. Epub 2007 Aug 21.
Bioorg Med Chem Lett. 2007.
PMID: 17869105
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