Opletalova V - Search Results

1

7-MEOTA-donepezil like compounds as cholinesterase inhibitors: Synthesis, pharmacological evaluation, molecular modeling and QSAR studies.

Korabecny J, Dolezal R, Cabelova P, Horova A, Hruba E, Ricny J, Sedlacek L, Nepovimova E, Spilovska K, Andrs M, Musilek K, Opletalova V, Sepsova V, Ripova D, Kuca K. Korabecny J, et al. Among authors: opletalova v. Eur J Med Chem. 2014 Jul 23;82:426-38. doi: 10.1016/j.ejmech.2014.05.066. Epub 2014 May 27. Eur J Med Chem. 2014. PMID: 24929293

2

Novel series of bispyridinium compounds bearing a (Z)-but-2-ene linker--synthesis and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase.

Musilek K, Holas O, Kuca K, Jun D, Dohnal V, Opletalova V, Dolezal M. Musilek K, et al. Among authors: opletalova v. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3172-6. doi: 10.1016/j.bmcl.2007.03.025. Epub 2007 Mar 13. Bioorg Med Chem Lett. 2007. PMID: 17383875

3

Monoquaternary pyridinium salts with modified side chain-synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase.

Musilek K, Kucera J, Jun D, Dohnal V, Opletalova V, Kuca K. Musilek K, et al. Among authors: opletalova v. Bioorg Med Chem. 2008 Sep 1;16(17):8218-23. doi: 10.1016/j.bmc.2008.07.036. Epub 2008 Jul 20. Bioorg Med Chem. 2008. PMID: 18676153

4

Synthesis and in vitro evaluation of N-alkyl-7-methoxytacrine hydrochlorides as potential cholinesterase inhibitors in Alzheimer disease.

Korabecny J, Musilek K, Holas O, Binder J, Zemek F, Marek J, Pohanka M, Opletalova V, Dohnal V, Kuca K. Korabecny J, et al. Among authors: opletalova v. Bioorg Med Chem Lett. 2010 Oct 15;20(20):6093-5. doi: 10.1016/j.bmcl.2010.08.044. Epub 2010 Aug 16. Bioorg Med Chem Lett. 2010. PMID: 20817518

5

Synthesis and in vitro evaluation of N-(Bromobut-3-en-2-yl)-7-methoxy-1,2,3,4-tetrahydroacridin-9-amine as a cholinesterase inhibitor with regard to Alzheimer's disease treatment.

Korabecny J, Musilek K, Holas O, Nepovimova E, Jun D, Zemek F, Opletalova V, Patocka J, Dohnal V, Nachon F, Hroudova J, Fisar Z, Kuca K. Korabecny J, et al. Among authors: opletalova v. Molecules. 2010 Dec 2;15(12):8804-12. doi: 10.3390/molecules15128804. Molecules. 2010. PMID: 21127466 Free PMC article.

6

Preparation, in vitro screening and molecular modelling of symmetrical 4-tert-butylpyridinium cholinesterase inhibitors--analogues of SAD-128.

Musilek K, Roder J, Komloova M, Holas O, Hrabinova M, Pohanka M, Dohnal V, Opletalova V, Kuca K, Jung YS. Musilek K, et al. Among authors: opletalova v. Bioorg Med Chem Lett. 2011 Jan 1;21(1):150-4. doi: 10.1016/j.bmcl.2010.11.051. Epub 2010 Nov 16. Bioorg Med Chem Lett. 2011. PMID: 21144749

7

Synthesis and in vitro evaluation of 7-methoxy-N-(pent-4-enyl)-1,2,3,4-tetrahydroacridin-9-amine-new tacrine derivate with cholinergic properties.

Korabecny J, Musilek K, Zemek F, Horova A, Holas O, Nepovimova E, Opletalova V, Hroudova J, Fisar Z, Jung YS, Kuca K. Korabecny J, et al. Among authors: opletalova v. Bioorg Med Chem Lett. 2011 Nov 1;21(21):6563-6. doi: 10.1016/j.bmcl.2011.08.042. Epub 2011 Aug 22. Bioorg Med Chem Lett. 2011. PMID: 21920739

8

Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase.

Musilek K, Holas O, Jun D, Dohnal V, Gunn-Moore F, Opletalova V, Dolezal M, Kuca K. Musilek K, et al. Among authors: opletalova v. Bioorg Med Chem. 2007 Nov 1;15(21):6733-41. doi: 10.1016/j.bmc.2007.08.002. Epub 2007 Aug 10. Bioorg Med Chem. 2007. PMID: 17764957

9

Synthesis of monooxime-monocarbamoyl bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against tabun- and paraoxon-inhibited acetylcholinesterase.

Musilek K, Holas O, Kuca K, Jun D, Dohnal V, Opletalova V, Dolezal M. Musilek K, et al. Among authors: opletalova v. J Enzyme Inhib Med Chem. 2008 Feb;23(1):70-6. doi: 10.1080/14756360701383981. J Enzyme Inhib Med Chem. 2008. PMID: 18341256 Free article.

10

Monooxime-monocarbamoyl Bispyridinium Xylene-Linked Reactivators of Acetylcholinesterase-Synthesis, In vitro and Toxicity Evaluation, and Docking Studies.

Musilek K, Holas O, Misik J, Pohanka M, Novotny L, Dohnal V, Opletalova V, Kuca K. Musilek K, et al. Among authors: opletalova v. ChemMedChem. 2010 Feb 1;5(2):247-54. doi: 10.1002/cmdc.200900455. ChemMedChem. 2010. PMID: 20058292

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