Cherkasov A - Search Results

1

Discovery of 1H-indole-2-carboxamides as novel inhibitors of the androgen receptor binding function 3 (BF3).

Ban F, Leblanc E, Li H, Munuganti RS, Frewin K, Rennie PS, Cherkasov A. Ban F, et al. Among authors: cherkasov a. J Med Chem. 2014 Aug 14;57(15):6867-72. doi: 10.1021/jm500684r. Epub 2014 Jul 25. J Med Chem. 2014. PMID: 25025737

2

Successful in silico discovery of novel nonsteroidal ligands for human sex hormone binding globulin.

Cherkasov A, Shi Z, Fallahi M, Hammond GL. Cherkasov A, et al. J Med Chem. 2005 May 5;48(9):3203-13. doi: 10.1021/jm049087f. J Med Chem. 2005. PMID: 15857126

3

Progressive docking: a hybrid QSAR/docking approach for accelerating in silico high throughput screening.

Cherkasov A, Ban F, Li Y, Fallahi M, Hammond GL. Cherkasov A, et al. J Med Chem. 2006 Dec 14;49(25):7466-78. doi: 10.1021/jm060961+. J Med Chem. 2006. PMID: 17149875

4

Indel-based targeting of essential proteins in human pathogens that have close host orthologue(s): discovery of selective inhibitors for Leishmania donovani elongation factor-1alpha.

Nandan D, Lopez M, Ban F, Huang M, Li Y, Reiner NE, Cherkasov A. Nandan D, et al. Among authors: cherkasov a. Proteins. 2007 Apr 1;67(1):53-64. doi: 10.1002/prot.21278. Proteins. 2007. PMID: 17243179

5

An updated steroid benchmark set and its application in the discovery of novel nanomolar ligands of sex hormone-binding globulin.

Cherkasov A, Ban F, Santos-Filho O, Thorsteinson N, Fallahi M, Hammond GL. Cherkasov A, et al. J Med Chem. 2008 Apr 10;51(7):2047-56. doi: 10.1021/jm7011485. Epub 2008 Mar 11. J Med Chem. 2008. PMID: 18330978

6

In silico identification of anthropogenic chemicals as ligands of zebrafish sex hormone binding globulin.

Thorsteinson N, Ban F, Santos-Filho O, Tabaei SM, Miguel-Queralt S, Underhill C, Cherkasov A, Hammond GL. Thorsteinson N, et al. Among authors: cherkasov a. Toxicol Appl Pharmacol. 2009 Jan 1;234(1):47-57. doi: 10.1016/j.taap.2008.07.014. Epub 2008 Jul 25. Toxicol Appl Pharmacol. 2009. PMID: 18725242

7

Identification of novel antibacterial peptides by chemoinformatics and machine learning.

Fjell CD, Jenssen H, Hilpert K, Cheung WA, Panté N, Hancock RE, Cherkasov A. Fjell CD, et al. Among authors: cherkasov a. J Med Chem. 2009 Apr 9;52(7):2006-15. doi: 10.1021/jm8015365. J Med Chem. 2009. PMID: 19296598

8

Inhibitors of androgen receptor activation function-2 (AF2) site identified through virtual screening.

Axerio-Cilies P, Lack NA, Nayana MR, Chan KH, Yeung A, Leblanc E, Guns ES, Rennie PS, Cherkasov A. Axerio-Cilies P, et al. Among authors: cherkasov a. J Med Chem. 2011 Sep 22;54(18):6197-205. doi: 10.1021/jm200532b. Epub 2011 Aug 29. J Med Chem. 2011. PMID: 21846139

9

Targeting the binding function 3 (BF3) site of the human androgen receptor through virtual screening.

Lack NA, Axerio-Cilies P, Tavassoli P, Han FQ, Chan KH, Feau C, LeBlanc E, Guns ET, Guy RK, Rennie PS, Cherkasov A. Lack NA, et al. Among authors: cherkasov a. J Med Chem. 2011 Dec 22;54(24):8563-73. doi: 10.1021/jm201098n. Epub 2011 Nov 18. J Med Chem. 2011. PMID: 22047606 Free PMC article.

10

Optimization and structure-activity relationships of a series of potent inhibitors of methicillin-resistant Staphylococcus aureus (MRSA) pyruvate kinase as novel antimicrobial agents.

Kumar NS, Amandoron EA, Cherkasov A, Finlay BB, Gong H, Jackson L, Kaur S, Lian T, Moreau A, Labrière C, Reiner NE, See RH, Strynadka NC, Thorson L, Wong EW, Worrall L, Zoraghi R, Young RN. Kumar NS, et al. Among authors: cherkasov a. Bioorg Med Chem. 2012 Dec 15;20(24):7069-82. doi: 10.1016/j.bmc.2012.10.002. Epub 2012 Oct 17. Bioorg Med Chem. 2012. PMID: 23141418

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