Thomas BF - Search Results

1

Diarylureas as allosteric modulators of the cannabinoid CB1 receptor: structure-activity relationship studies on 1-(4-chlorophenyl)-3-{3-[6-(pyrrolidin-1-yl)pyridin-2-yl]phenyl}urea (PSNCBAM-1).

German N, Decker AM, Gilmour BP, Gay EA, Wiley JL, Thomas BF, Zhang Y. German N, et al. Among authors: thomas bf. J Med Chem. 2014 Sep 25;57(18):7758-69. doi: 10.1021/jm501042u. Epub 2014 Sep 4. J Med Chem. 2014. PMID: 25162172 Free PMC article.

2

Synthesis and biological evaluation of bivalent ligands for the cannabinoid 1 receptor.

Zhang Y, Gilliam A, Maitra R, Damaj MI, Tajuba JM, Seltzman HH, Thomas BF. Zhang Y, et al. Among authors: thomas bf. J Med Chem. 2010 Oct 14;53(19):7048-60. doi: 10.1021/jm1006676. J Med Chem. 2010. PMID: 20845959 Free PMC article.

3

Diaryl urea analogues of SB-334867 as orexin-1 receptor antagonists.

Perrey DA, Gilmour BP, Runyon SP, Thomas BF, Zhang Y. Perrey DA, et al. Among authors: thomas bf. Bioorg Med Chem Lett. 2011 May 15;21(10):2980-5. doi: 10.1016/j.bmcl.2011.03.048. Epub 2011 Mar 21. Bioorg Med Chem Lett. 2011. PMID: 21478014 Free PMC article.

4

Substituted tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

Perrey DA, German NA, Gilmour BP, Li JX, Harris DL, Thomas BF, Zhang Y. Perrey DA, et al. Among authors: thomas bf. J Med Chem. 2013 Sep 12;56(17):6901-16. doi: 10.1021/jm400720h. Epub 2013 Aug 26. J Med Chem. 2013. PMID: 23941044 Free PMC article.

5

Truncated Orexin Peptides: Structure-Activity Relationship Studies.

German NA, Decker AM, Gilmour BP, Thomas BF, Zhang Y. German NA, et al. Among authors: thomas bf. ACS Med Chem Lett. 2013 Dec 12;4(12):1224-1227. doi: 10.1021/ml400333a. ACS Med Chem Lett. 2013. PMID: 24707347 Free PMC article.

6

Toward the Development of Bivalent Ligand Probes of Cannabinoid CB1 and Orexin OX1 Receptor Heterodimers.

Perrey DA, Gilmour BP, Thomas BF, Zhang Y. Perrey DA, et al. Among authors: thomas bf. ACS Med Chem Lett. 2014 Mar 25;5(6):634-8. doi: 10.1021/ml4004759. eCollection 2014 Jun 12. ACS Med Chem Lett. 2014. PMID: 24944734 Free PMC article.

7

Effect of 1-substitution on tetrahydroisoquinolines as selective antagonists for the orexin-1 receptor.

Perrey DA, German NA, Decker AM, Thorn D, Li JX, Gilmour BP, Thomas BF, Harris DL, Runyon SP, Zhang Y. Perrey DA, et al. Among authors: thomas bf. ACS Chem Neurosci. 2015 Apr 15;6(4):599-614. doi: 10.1021/cn500330v. Epub 2015 Feb 12. ACS Chem Neurosci. 2015. PMID: 25643283 Free PMC article.

8

Structure-activity relationships of substituted 1H-indole-2-carboxamides as CB1 receptor allosteric modulators.

Nguyen T, German N, Decker AM, Li JX, Wiley JL, Thomas BF, Kenakin TP, Zhang Y. Nguyen T, et al. Among authors: thomas bf. Bioorg Med Chem. 2015 May 1;23(9):2195-2203. doi: 10.1016/j.bmc.2015.02.058. Epub 2015 Mar 7. Bioorg Med Chem. 2015. PMID: 25797163 Free PMC article.

9

The importance of the 6- and 7-positions of tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

Perrey DA, Decker AM, Li JX, Gilmour BP, Thomas BF, Harris DL, Runyon SP, Zhang Y. Perrey DA, et al. Among authors: thomas bf. Bioorg Med Chem. 2015 Sep 1;23(17):5709-24. doi: 10.1016/j.bmc.2015.07.013. Epub 2015 Jul 16. Bioorg Med Chem. 2015. PMID: 26216017 Free PMC article.

10

Allosteric Modulation: An Alternate Approach Targeting the Cannabinoid CB1 Receptor.

Nguyen T, Li JX, Thomas BF, Wiley JL, Kenakin TP, Zhang Y. Nguyen T, et al. Among authors: thomas bf. Med Res Rev. 2017 May;37(3):441-474. doi: 10.1002/med.21418. Epub 2016 Nov 23. Med Res Rev. 2017. PMID: 27879006 Free PMC article. Review.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

129 results

Search Page

Filters