Svensson R - Search Results

1

Preclinical characterization of acyl sulfonimidamides: potential carboxylic acid bioisosteres with tunable properties.

Borhade SR, Svensson R, Brandt P, Artursson P, Arvidsson PI, Sandström A. Borhade SR, et al. Among authors: svensson r. ChemMedChem. 2015 Mar;10(3):455-60. doi: 10.1002/cmdc.201402497. Epub 2015 Jan 28. ChemMedChem. 2015. PMID: 25630705

2

Optimizing solubility and permeability of a biopharmaceutics classification system (BCS) class 4 antibiotic drug using lipophilic fragments disturbing the crystal lattice.

Tehler U, Fagerberg JH, Svensson R, Larhed M, Artursson P, Bergström CA. Tehler U, et al. Among authors: svensson r. J Med Chem. 2013 Mar 28;56(6):2690-4. doi: 10.1021/jm301721e. Epub 2013 Mar 19. J Med Chem. 2013. PMID: 23432334 Free article.

3

Achiral pyrazinone-based inhibitors of the hepatitis C virus NS3 protease and drug-resistant variants with elongated substituents directed toward the S2 pocket.

Gising J, Belfrage AK, Alogheli H, Ehrenberg A, Åkerblom E, Svensson R, Artursson P, Karlén A, Danielson UH, Larhed M, Sandström A. Gising J, et al. Among authors: svensson r. J Med Chem. 2014 Mar 13;57(5):1790-801. doi: 10.1021/jm301887f. Epub 2013 Apr 2. J Med Chem. 2014. PMID: 23517538

4

Constrained H-Phe-Phe-NH2 analogues with high affinity to the substance P 1-7 binding site and with improved metabolic stability and cell permeability.

Fransson R, Sköld C, Kratz JM, Svensson R, Artursson P, Nyberg F, Hallberg M, Sandström A. Fransson R, et al. Among authors: svensson r. J Med Chem. 2013 Jun 27;56(12):4953-65. doi: 10.1021/jm400209h. Epub 2013 Jun 17. J Med Chem. 2013. PMID: 23735006 Free article.

5

Novel Peptidomimetic Hepatitis C Virus NS3/4A Protease Inhibitors Spanning the P2-P1' Region.

Lampa AK, Bergman SM, Gustafsson SS, Alogheli H, Akerblom EB, Lindeberg GG, Svensson RM, Artursson P, Danielson UH, Karlén A, Sandström A. Lampa AK, et al. ACS Med Chem Lett. 2013 Aug 2;5(3):249-54. doi: 10.1021/ml400217r. eCollection 2014 Mar 13. ACS Med Chem Lett. 2013. PMID: 24900813 Free PMC article.

6

Vinylated linear P2 pyrimidinyloxyphenylglycine based inhibitors of the HCV NS3/4A protease and corresponding macrocycles.

Lampa A, Alogheli H, Ehrenberg AE, Åkerblom E, Svensson R, Artursson P, Danielson UH, Karlén A, Sandström A. Lampa A, et al. Among authors: svensson r. Bioorg Med Chem. 2014 Dec 1;22(23):6595-6615. doi: 10.1016/j.bmc.2014.10.010. Bioorg Med Chem. 2014. PMID: 25456385

7

Exploration and pharmacokinetic profiling of phenylalanine based carbamates as novel substance p 1-7 analogues.

Fransson R, Nordvall G, Bylund J, Carlsson-Jonsson A, Kratz JM, Svensson R, Artursson P, Hallberg M, Sandström A. Fransson R, et al. Among authors: svensson r. ACS Med Chem Lett. 2014 Oct 29;5(12):1272-7. doi: 10.1021/ml5002954. eCollection 2014 Dec 11. ACS Med Chem Lett. 2014. PMID: 25516784 Free PMC article.

8

Importance of N- and C-terminal residues of substance P 1-7 for alleviating allodynia in mice after peripheral administration.

Skogh A, Lesniak A, Gaugaz FZ, Svensson R, Lindeberg G, Fransson R, Nyberg F, Hallberg M, Sandström A. Skogh A, et al. Among authors: svensson r. Eur J Pharm Sci. 2017 Aug 30;106:345-351. doi: 10.1016/j.ejps.2017.06.004. Epub 2017 Jun 3. Eur J Pharm Sci. 2017. PMID: 28587787

9

Anti-Rift Valley fever virus activity in vitro, pre-clinical pharmacokinetics and oral bioavailability of benzavir-2, a broad-acting antiviral compound.

Islam MK, Strand M, Saleeb M, Svensson R, Baranczewski P, Artursson P, Wadell G, Ahlm C, Elofsson M, Evander M. Islam MK, et al. Among authors: svensson r. Sci Rep. 2018 Jan 31;8(1):1925. doi: 10.1038/s41598-018-20362-9. Sci Rep. 2018. PMID: 29386590 Free PMC article.

10

In vitro and in silico strategies to identify OATP1B1 inhibitors and predict clinical drug-drug interactions.

Karlgren M, Ahlin G, Bergström CA, Svensson R, Palm J, Artursson P. Karlgren M, et al. Among authors: svensson r. Pharm Res. 2012 Feb;29(2):411-26. doi: 10.1007/s11095-011-0564-9. Epub 2011 Aug 23. Pharm Res. 2012. PMID: 21861202 Free PMC article.

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