Runyon SP - Search Results

1

Effect of 1-substitution on tetrahydroisoquinolines as selective antagonists for the orexin-1 receptor.

Perrey DA, German NA, Decker AM, Thorn D, Li JX, Gilmour BP, Thomas BF, Harris DL, Runyon SP, Zhang Y. Perrey DA, et al. Among authors: runyon sp. ACS Chem Neurosci. 2015 Apr 15;6(4):599-614. doi: 10.1021/cn500330v. Epub 2015 Feb 12. ACS Chem Neurosci. 2015. PMID: 25643283 Free PMC article.

2

Identifying structural features on 1,1-diphenyl-hexahydro-oxazolo[3,4-a]pyrazin-3-ones critical for Neuropeptide S antagonist activity.

Zhang Y, Gilmour BP, Navarro HA, Runyon SP. Zhang Y, et al. Among authors: runyon sp. Bioorg Med Chem Lett. 2008 Jul 15;18(14):4064-7. doi: 10.1016/j.bmcl.2008.05.098. Epub 2008 Jun 12. Bioorg Med Chem Lett. 2008. PMID: 18555684 Free PMC article.

3

Diaryl urea analogues of SB-334867 as orexin-1 receptor antagonists.

Perrey DA, Gilmour BP, Runyon SP, Thomas BF, Zhang Y. Perrey DA, et al. Among authors: runyon sp. Bioorg Med Chem Lett. 2011 May 15;21(10):2980-5. doi: 10.1016/j.bmcl.2011.03.048. Epub 2011 Mar 21. Bioorg Med Chem Lett. 2011. PMID: 21478014 Free PMC article.

4

Antagonism of the neuropeptide S receptor with RTI-118 decreases cocaine self-administration and cocaine-seeking behavior in rats.

Schmoutz CD, Zhang Y, Runyon SP, Goeders NE. Schmoutz CD, et al. Among authors: runyon sp. Pharmacol Biochem Behav. 2012 Dec;103(2):332-7. doi: 10.1016/j.pbb.2012.09.003. Epub 2012 Sep 12. Pharmacol Biochem Behav. 2012. PMID: 22982682 Free PMC article.

5

Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: possible confounding effects on in vivo and in vitro studies.

McElhinny CJ Jr, Lewin AH, Mascarella SW, Runyon S, Brieaddy L, Carroll FI. McElhinny CJ Jr, et al. Bioorg Med Chem Lett. 2012 Nov 1;22(21):6661-4. doi: 10.1016/j.bmcl.2012.08.109. Epub 2012 Sep 7. Bioorg Med Chem Lett. 2012. PMID: 23031594

6

Discovery of N-{4-[(3-hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide analogues as selective kappa opioid receptor antagonists.

Kormos CM, Jin C, Cueva JP, Runyon SP, Thomas JB, Brieaddy LE, Mascarella SW, Navarro HA, Gilmour BP, Carroll FI. Kormos CM, et al. Among authors: runyon sp. J Med Chem. 2013 Jun 13;56(11):4551-67. doi: 10.1021/jm400275h. Epub 2013 May 16. J Med Chem. 2013. PMID: 23651437 Free PMC article.

7

Effect of the 3- and 4-methyl groups on the opioid receptor properties of N-substituted trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidines.

Kormos CM, Cueva JP, Gichinga MG, Runyon SP, Thomas JB, Brieaddy LE, Mascarella SW, Gilmour BP, Navarro HA, Carroll FI. Kormos CM, et al. Among authors: runyon sp. J Med Chem. 2014 Apr 10;57(7):3140-7. doi: 10.1021/jm500184j. Epub 2014 Mar 26. J Med Chem. 2014. PMID: 24635568 Free PMC article.

8

Identifying structural determinants of potency for analogs of apelin-13: integration of C-terminal truncation with structure-activity.

Zhang Y, Maitra R, Harris DL, Dhungana S, Snyder R, Runyon SP. Zhang Y, et al. Among authors: runyon sp. Bioorg Med Chem. 2014 Jun 1;22(11):2992-7. doi: 10.1016/j.bmc.2014.04.001. Epub 2014 Apr 13. Bioorg Med Chem. 2014. PMID: 24755525

9

Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound.

Thomas JB, Giddings AM, Wiethe RW, Olepu S, Warner KR, Sarret P, Gendron L, Longpre JM, Zhang Y, Runyon SP, Gilmour BP. Thomas JB, et al. Among authors: runyon sp. J Med Chem. 2014 Jun 26;57(12):5318-32. doi: 10.1021/jm5003843. Epub 2014 Jun 5. J Med Chem. 2014. PMID: 24856674 Free PMC article.

10

Identification of neuropeptide S antagonists: structure-activity relationship studies, X-ray crystallography, and in vivo evaluation.

Hassler C, Zhang Y, Gilmour B, Graf T, Fennell T, Snyder R, Deschamps JR, Reinscheid RK, Garau C, Runyon SP. Hassler C, et al. Among authors: runyon sp. ACS Chem Neurosci. 2014 Aug 20;5(8):731-44. doi: 10.1021/cn500113c. Epub 2014 Jul 11. ACS Chem Neurosci. 2014. PMID: 24964000 Free PMC article.

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