Busca P - Search Results

1

Molecular modeling study of the induced-fit effect on kinase inhibition: the case of fibroblast growth factor receptor 3 (FGFR3).

Li Y, Delamar M, Busca P, Prestat G, Le Corre L, Legeai-Mallet L, Hu R, Zhang R, Barbault F. Li Y, et al. Among authors: busca p. J Comput Aided Mol Des. 2015 Jul;29(7):619-41. doi: 10.1007/s10822-015-9841-8. Epub 2015 Mar 26. J Comput Aided Mol Des. 2015. PMID: 25808135

2

A novel tyrosine kinase inhibitor restores chondrocyte differentiation and promotes bone growth in a gain-of-function Fgfr3 mouse model.

Jonquoy A, Mugniery E, Benoist-Lasselin C, Kaci N, Le Corre L, Barbault F, Girard AL, Le Merrer Y, Busca P, Schibler L, Munnich A, Legeai-Mallet L. Jonquoy A, et al. Among authors: busca p. Hum Mol Genet. 2012 Feb 15;21(4):841-51. doi: 10.1093/hmg/ddr514. Epub 2011 Nov 9. Hum Mol Genet. 2012. PMID: 22072392

3

Synthesis and biological evaluation of a triazole-based library of pyrido[2,3-d]pyrimidines as FGFR3 tyrosine kinase inhibitors.

Le Corre L, Girard AL, Aubertin J, Radvanyi F, Benoist-Lasselin C, Jonquoy A, Mugniery E, Legeai-Mallet L, Busca P, Le Merrer Y. Le Corre L, et al. Among authors: busca p. Org Biomol Chem. 2010 May 7;8(9):2164-73. doi: 10.1039/b923882d. Epub 2010 Mar 11. Org Biomol Chem. 2010. PMID: 20401393

4

Synthesis of purin-2-yl and purin-6-yl-aminoglucitols as C-nucleosidic ATP mimics and biological evaluation as FGFR3 inhibitors.

Tak-Tak L, Barbault F, Maurel F, Busca P, Le Merrer Y. Tak-Tak L, et al. Among authors: busca p. Eur J Med Chem. 2011 Apr;46(4):1254-62. doi: 10.1016/j.ejmech.2011.01.048. Epub 2011 Feb 3. Eur J Med Chem. 2011. PMID: 21334122

5

Tyrosine kinase inhibitor NVP-BGJ398 functionally improves FGFR3-related dwarfism in mouse model.

Komla-Ebri D, Dambroise E, Kramer I, Benoist-Lasselin C, Kaci N, Le Gall C, Martin L, Busca P, Barbault F, Graus-Porta D, Munnich A, Kneissel M, Di Rocco F, Biosse-Duplan M, Legeai-Mallet L. Komla-Ebri D, et al. Among authors: busca p. J Clin Invest. 2016 May 2;126(5):1871-84. doi: 10.1172/JCI83926. Epub 2016 Apr 11. J Clin Invest. 2016. PMID: 27064282 Free PMC article.

6

Reductive Cleavage of Aromatic and Heteroaromatic Ester Functions via Copper-Catalyzed Proto-Decarbomethoxylation.

Fichez J, Prestat G, Busca P. Fichez J, et al. Among authors: busca p. Org Lett. 2018 May 4;20(9):2724-2727. doi: 10.1021/acs.orglett.8b00930. Epub 2018 Apr 25. Org Lett. 2018. PMID: 29693397

7

Microwave-assisted preparation of 4-amino-3-cyano-5-methoxycarbonyl-N-arylpyrazoles as building blocks for the diversity-oriented synthesis of pyrazole-based polycyclic scaffolds.

Le Corre L, Tak-Tak L, Guillard A, Prestat G, Gravier-Pelletier C, Busca P. Le Corre L, et al. Among authors: busca p. Org Biomol Chem. 2015 Jan 14;13(2):409-23. doi: 10.1039/c4ob01951b. Epub 2014 Nov 4. Org Biomol Chem. 2015. PMID: 25369050

8

Discovery, SAR study and ADME properties of methyl 4-amino-3-cyano-1-(2-benzyloxyphenyl)-1H-pyrazole-5-carboxylate as an HIV-1 replication inhibitor.

Fichez J, Soulie C, Le Corre L, Sayon S, Priet S, Alvarez K, Delelis O, Gizzi P, Prestat G, Gravier-Pelletier C, Marcelin AG, Calvez V, Busca P. Fichez J, et al. Among authors: busca p. RSC Med Chem. 2020 Apr 27;11(5):577-582. doi: 10.1039/d0md00025f. eCollection 2020 May 1. RSC Med Chem. 2020. PMID: 33479659 Free PMC article.

9

Destabilization of the human RED-SMU1 splicing complex as a basis for host-directed antiinfluenza strategy.

Ashraf U, Tengo L, Le Corre L, Fournier G, Busca P, McCarthy AA, Rameix-Welti MA, Gravier-Pelletier C, Ruigrok RWH, Jacob Y, Vidalain PO, Pietrancosta N, Crépin T, Naffakh N. Ashraf U, et al. Among authors: busca p. Proc Natl Acad Sci U S A. 2019 May 28;116(22):10968-10977. doi: 10.1073/pnas.1901214116. Epub 2019 May 10. Proc Natl Acad Sci U S A. 2019. PMID: 31076555 Free PMC article.

10

Synthesis and biological evaluation of chemical tools for the study of Dolichol Linked Oligosaccharide Diphosphatase (DLODP).

Bosco M, Massarweh A, Iatmanen-Harbi S, Bouhss A, Chantret I, Busca P, Moore SE, Gravier-Pelletier C. Bosco M, et al. Among authors: busca p. Eur J Med Chem. 2017 Jan 5;125:952-964. doi: 10.1016/j.ejmech.2016.10.013. Epub 2016 Oct 8. Eur J Med Chem. 2017. PMID: 27769035

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