Coumar MS - Search Results

1

Homology modeling of DFG-in FMS-like tyrosine kinase 3 (FLT3) and structure-based virtual screening for inhibitor identification.

Ke YY, Singh VK, Coumar MS, Hsu YC, Wang WC, Song JS, Chen CH, Lin WH, Wu SH, Hsu JT, Shih C, Hsieh HP. Ke YY, et al. Among authors: coumar ms. Sci Rep. 2015 Jun 29;5:11702. doi: 10.1038/srep11702. Sci Rep. 2015. PMID: 26118648 Free PMC article.

2

2-[3-[2-[(2S)-2-Cyano-1-pyrrolidinyl]-2-oxoethylamino]-3-methyl-1-oxobutyl]- 1,2,3,4-tetrahydroisoquinoline: a potent, selective, and orally bioavailable dipeptide-derived inhibitor of dipeptidyl peptidase IV.

Tsu H, Chen X, Chen CT, Lee SJ, Chang CN, Kao KH, Coumar MS, Yeh YT, Chien CH, Wang HS, Lin KT, Chang YY, Wu SH, Chen YS, Lu IL, Wu SY, Tsai TY, Chen WC, Hsieh HP, Chao YS, Jiaang WT. Tsu H, et al. Among authors: coumar ms. J Med Chem. 2006 Jan 12;49(1):373-80. doi: 10.1021/jm0507781. J Med Chem. 2006. PMID: 16392822

3

Substituted pyrrolidine-2,4-dicarboxylic acid amides as potent dipeptidyl peptidase IV inhibitors.

Tsai TY, Coumar MS, Hsu T, Hsieh HP, Chien CH, Chen CT, Chang CN, Lo YK, Wu SH, Huang CY, Huang YW, Wang MH, Wu HY, Lee HJ, Chen X, Chao YS, Jiaang WT. Tsai TY, et al. Among authors: coumar ms. Bioorg Med Chem Lett. 2006 Jun 15;16(12):3268-72. doi: 10.1016/j.bmcl.2006.03.037. Epub 2006 Apr 11. Bioorg Med Chem Lett. 2006. PMID: 16581245

4

3-[2-((2S)-2-cyano-pyrrolidin-1-yl)-2-oxo-ethylamino]-3-methyl-butyramide analogues as selective DPP-IV inhibitors for the treatment of type-II diabetes.

Coumar MS, Chang CN, Chen CT, Chen X, Chien CH, Tsai TY, Cheng JH, Wu HY, Han CH, Wu SH, Huang YW, Hsu T, Hsu LJ, Chao YS, Hsieh HP, Jiaang WT. Coumar MS, et al. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1274-9. doi: 10.1016/j.bmcl.2006.12.019. Epub 2006 Dec 12. Bioorg Med Chem Lett. 2007. PMID: 17194587

5

Aurora kinase A inhibitors: identification, SAR exploration and molecular modeling of 6,7-dihydro-4H-pyrazolo-[1,5-a]pyrrolo[3,4-d]pyrimidine-5,8-dione scaffold.

Coumar MS, Wu JS, Leou JS, Tan UK, Chang CY, Chang TY, Lin WH, Hsu JT, Chao YS, Wu SY, Hsieh HP. Coumar MS, et al. Bioorg Med Chem Lett. 2008 Mar 1;18(5):1623-7. doi: 10.1016/j.bmcl.2008.01.068. Epub 2008 Jan 19. Bioorg Med Chem Lett. 2008. PMID: 18243698

6

Synthesis and structure-activity relationships of 2-amino-1-aroylnaphthalene and 2-hydroxy-1-aroylnaphthalenes as potent antitubulin agents.

Reddy GR, Kuo CC, Tan UK, Coumar MS, Chang CY, Chiang YK, Lai MJ, Yeh JY, Wu SY, Chang JY, Liou JP, Hsieh HP. Reddy GR, et al. Among authors: coumar ms. J Med Chem. 2008 Dec 25;51(24):8163-7. doi: 10.1021/jm8008635. J Med Chem. 2008. PMID: 19053773

7

Structure-based drug design of novel Aurora kinase A inhibitors: structural basis for potency and specificity.

Coumar MS, Leou JS, Shukla P, Wu JS, Dixit AK, Lin WH, Chang CY, Lien TW, Tan UK, Chen CH, Hsu JT, Chao YS, Wu SY, Hsieh HP. Coumar MS, et al. J Med Chem. 2009 Feb 26;52(4):1050-62. doi: 10.1021/jm801270e. J Med Chem. 2009. PMID: 19140666

8

Design and structural analysis of novel pharmacophores for potent and selective peroxisome proliferator-activated receptor gamma agonists.

Lin CH, Peng YH, Coumar MS, Chittimalla SK, Liao CC, Lyn PC, Huang CC, Lien TW, Lin WH, Hsu JT, Cheng JH, Chen X, Wu JS, Chao YS, Lee HJ, Juo CG, Wu SY, Hsieh HP. Lin CH, et al. Among authors: coumar ms. J Med Chem. 2009 Apr 23;52(8):2618-22. doi: 10.1021/jm801594x. J Med Chem. 2009. PMID: 19301897

9

Aurora kinase inhibitors in preclinical and clinical testing.

Cheung CH, Coumar MS, Hsieh HP, Chang JY. Cheung CH, et al. Among authors: coumar ms. Expert Opin Investig Drugs. 2009 Apr;18(4):379-98. doi: 10.1517/13543780902806392. Expert Opin Investig Drugs. 2009. PMID: 19335272 Review.

10

Advances in Aurora kinase inhibitor patents.

Coumar MS, Cheung CH, Chang JY, Hsieh HP. Coumar MS, et al. Expert Opin Ther Pat. 2009 Mar;19(3):321-56. doi: 10.1517/13543770802646949. Expert Opin Ther Pat. 2009. PMID: 19441907 Review.

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