Ellman JA - Search Results

1

Tetrafluorophenoxymethyl ketone cruzain inhibitors with improved pharmacokinetic properties as therapeutic leads for Chagas' disease.

Neitz RJ, Bryant C, Chen S, Gut J, Hugo Caselli E, Ponce S, Chowdhury S, Xu H, Arkin MR, Ellman JA, Renslo AR. Neitz RJ, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2015 Nov 1;25(21):4834-4837. doi: 10.1016/j.bmcl.2015.06.066. Epub 2015 Jun 23. Bioorg Med Chem Lett. 2015. PMID: 26144347 Free PMC article.

2

Expedient method for the solid-phase synthesis of aspartic acid protease inhibitors directed toward the generation of libraries.

Kick EK, Ellman JA. Kick EK, et al. Among authors: ellman ja. J Med Chem. 1995 Apr 28;38(9):1427-30. doi: 10.1021/jm00009a002. J Med Chem. 1995. PMID: 7739000 No abstract available.

3

Novel inhibitors of alpha 4 beta 1 integrin receptor interactions through library synthesis and screening.

Souers AJ, Virgilio AA, Schürer SS, Ellman JA, Kogan TP, West HE, Ankener W, Vanderslice P. Souers AJ, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 1998 Sep 8;8(17):2297-302. doi: 10.1016/s0960-894x(98)00416-8. Bioorg Med Chem Lett. 1998. PMID: 9873531

4

Potent, low-molecular-weight non-peptide inhibitors of malarial aspartyl protease plasmepsin II.

Haque TS, Skillman AG, Lee CE, Habashita H, Gluzman IY, Ewing TJ, Goldberg DE, Kuntz ID, Ellman JA. Haque TS, et al. Among authors: ellman ja. J Med Chem. 1999 Apr 22;42(8):1428-40. doi: 10.1021/jm980641t. J Med Chem. 1999. PMID: 10212129

5

Optimization of a somatostatin mimetic via constrained amino acid and backbone incorporation.

Souers AJ, Rosenquist A, Jarvie EM, Ladlow M, Feniuk W, Ellman JA. Souers AJ, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2000 Dec 18;10(24):2731-3. doi: 10.1016/s0960-894x(00)00552-7. Bioorg Med Chem Lett. 2000. PMID: 11133079

6

Identification of potent and selective mechanism-based inhibitors of the cysteine protease cruzain using solid-phase parallel synthesis.

Huang L, Lee A, Ellman JA. Huang L, et al. Among authors: ellman ja. J Med Chem. 2002 Jan 31;45(3):676-84. doi: 10.1021/jm010333m. J Med Chem. 2002. PMID: 11806719

7

Tyrosylprotein sulfotransferase inhibitors generated by combinatorial target-guided ligand assembly.

Kehoe JW, Maly DJ, Verdugo DE, Armstrong JI, Cook BN, Ouyang YB, Moore KL, Ellman JA, Bertozzi CR. Kehoe JW, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2002 Feb 11;12(3):329-32. doi: 10.1016/s0960-894x(01)00744-2. Bioorg Med Chem Lett. 2002. PMID: 11814789

8

Design and synthesis of novel inhibitors of gelatinase B.

Wang X, Choe Y, Craik CS, Ellman JA. Wang X, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2002 Aug 19;12(16):2201-4. doi: 10.1016/s0960-894x(02)00365-7. Bioorg Med Chem Lett. 2002. PMID: 12127537

9

General solid-phase method to prepare novel cyclic ketone inhibitors of the cysteine protease cruzain.

Huang L, Ellman JA. Huang L, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2993-6. doi: 10.1016/s0960-894x(02)00619-4. Bioorg Med Chem Lett. 2002. PMID: 12270191

10

Crystal structures of reversible ketone-Based inhibitors of the cysteine protease cruzain.

Huang L, Brinen LS, Ellman JA. Huang L, et al. Among authors: ellman ja. Bioorg Med Chem. 2003 Jan 2;11(1):21-9. doi: 10.1016/s0968-0896(02)00427-3. Bioorg Med Chem. 2003. PMID: 12467703

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