Bräuner-Osborne H - Search Results

1

Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold.

Johansson H, Boesgaard MW, Nørskov-Lauritsen L, Larsen I, Kuhne S, Gloriam DE, Bräuner-Osborne H, Sejer Pedersen D. Johansson H, et al. J Med Chem. 2015 Nov 25;58(22):8938-51. doi: 10.1021/acs.jmedchem.5b01254. Epub 2015 Nov 16. J Med Chem. 2015. PMID: 26516782

2

Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors.

Bräuner-Osborne H, Ebert B, Brann MR, Falch E, Krogsgaard-Larsen P. Bräuner-Osborne H, et al. J Med Chem. 1995 Jun 9;38(12):2188-95. doi: 10.1021/jm00012a019. J Med Chem. 1995. PMID: 7783150

3

A new highly selective metabotropic excitatory amino acid agonist: 2-amino-4-(3-hydroxy-5-methylisoxazol-4-yl)butyric acid.

Bräuner-Osborne H, Sløk FA, Skjaerbaek N, Ebert B, Sekiyama N, Nakanishi S, Krogsgaard-Larsen P. Bräuner-Osborne H, et al. J Med Chem. 1996 Aug 2;39(16):3188-94. doi: 10.1021/jm9602569. J Med Chem. 1996. PMID: 8759641

4

(S)-homo-AMPA, a specific agonist at the mGlu6 subtype of metabotropic glutamic acid receptors.

Ahmadian H, Nielsen B, Bräuner-Osborne H, Johansen TN, Stensbøl TB, Sløk FA, Sekiyama N, Nakanishi S, Krogsgaard-Larsen P, Madsen U. Ahmadian H, et al. J Med Chem. 1997 Oct 24;40(22):3700-5. doi: 10.1021/jm9703597. J Med Chem. 1997. PMID: 9357538

5

Synthesis and pharmacology of N-alkylated derivatives of the excitotoxin ibotenic acid.

Madsen U, Dumpis MA, Bräuner-Osborne H, Piotrovsky LB. Madsen U, et al. Bioorg Med Chem Lett. 1998 Jun 16;8(12):1563-8. doi: 10.1016/s0960-894x(98)00264-9. Bioorg Med Chem Lett. 1998. PMID: 9873391

6

Synthesis and muscarinic receptor pharmacology of a series of 4,5,6,7-tetrahydroisothiazolo[4,5-c]pyridine bioisosteres of arecoline.

Pedersen H, Bräuner-Osborne H, Ball RG, Frydenvang K, Meier E, Bøgesø KP, Krogsgaard-Larsen P. Pedersen H, et al. Bioorg Med Chem. 1999 May;7(5):795-809. doi: 10.1016/s0968-0896(99)00033-4. Bioorg Med Chem. 1999. PMID: 10400332

7

Ionotropic excitatory amino acid receptor ligands. Synthesis and pharmacology of a new amino acid AMPA antagonist.

Madsen U, Sløk FA, Stensbøl TB, Bräuner-Osborne H, Lützhøft HH, Poulsen MV, Eriksen L, Krogsgaard-Larsen P. Madsen U, et al. Eur J Med Chem. 2000 Jan;35(1):69-76. doi: 10.1016/s0223-5234(00)00104-5. Eur J Med Chem. 2000. PMID: 10733604

8

Ligands for glutamate receptors: design and therapeutic prospects.

Bräuner-Osborne H, Egebjerg J, Nielsen EO, Madsen U, Krogsgaard-Larsen P. Bräuner-Osborne H, et al. J Med Chem. 2000 Jul 13;43(14):2609-45. doi: 10.1021/jm000007r. J Med Chem. 2000. PMID: 10893301 Review. No abstract available.

9

Construction of a high affinity zinc binding site in the metabotropic glutamate receptor mGluR1: noncompetitive antagonism originating from the amino-terminal domain of a family C G-protein-coupled receptor.

Jensen AA, Sheppard PO, Jensen LB, O'Hara PJ, Bräuner-Osborne H. Jensen AA, et al. J Biol Chem. 2001 Mar 30;276(13):10110-8. doi: 10.1074/jbc.M007220200. Epub 2000 Dec 22. J Biol Chem. 2001. PMID: 11133983 Free article.

10

Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors.

Madsen U, Bräuner-Osborne H, Frydenvang K, Hvene L, Johansen TN, Nielsen B, Sánchez C, Stensbøl TB, Bischoff F, Krogsgaard-Larsen P. Madsen U, et al. J Med Chem. 2001 Mar 29;44(7):1051-9. doi: 10.1021/jm000441t. J Med Chem. 2001. PMID: 11297452

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

224 results

Search Page

Filters