Grée R - Search Results

1

Preliminary Studies on the Activity of Mixed Polyphenol-Heterocyclic Systems Against B16-F10 Melanoma Cancer Cells.

Duy Vo D, Rouaud I, Le Devehat F, Gautier F, Barillé-Nion S, Juin P, Levoin N, Boustie J, Grée R. Duy Vo D, et al. Among authors: gree r. Med Chem. 2016;12(5):419-25. doi: 10.2174/1573406412666160129104603. Med Chem. 2016. PMID: 26825069

2

The small organic compound HA14-1 prevents Bcl-2 interaction with Bax to sensitize malignant glioma cells to induction of cell death.

Manero F, Gautier F, Gallenne T, Cauquil N, Grée D, Cartron PF, Geneste O, Grée R, Vallette FM, Juin P. Manero F, et al. Among authors: gree r, gree d. Cancer Res. 2006 Mar 1;66(5):2757-64. doi: 10.1158/0008-5472.CAN-05-2097. Cancer Res. 2006. PMID: 16510597

3

HA14-1, a small molecule inhibitor of Bcl-2, bypasses chemoresistance in leukaemia cells.

Oliver L, Mahé B, Gréé R, Vallette FM, Juin P. Oliver L, et al. Among authors: gree r. Leuk Res. 2007 Jun;31(6):859-63. doi: 10.1016/j.leukres.2006.11.010. Epub 2007 Jan 16. Leuk Res. 2007. PMID: 17224180

4

Mitochondrial targeting by use of lipid nanocapsules loaded with SV30, an analogue of the small-molecule Bcl-2 inhibitor HA14-1.

Weyland M, Manero F, Paillard A, Grée D, Viault G, Jarnet D, Menei P, Juin P, Chourpa I, Benoit JP, Grée R, Garcion E. Weyland M, et al. Among authors: gree r, gree d. J Control Release. 2011 Apr 10;151(1):74-82. doi: 10.1016/j.jconrel.2010.11.032. Epub 2010 Dec 5. J Control Release. 2011. PMID: 21138749 Free article.

5

Structure-activity relationship of selected polyphenol derivatives as inhibitors of Bax/Bcl-xL interaction.

Vo DD, Gautier F, Juin P, Grée R. Vo DD, et al. Among authors: gree r. Eur J Med Chem. 2012 May;51:286-93. doi: 10.1016/j.ejmech.2012.02.036. Epub 2012 Feb 25. Eur J Med Chem. 2012. PMID: 22425031

6

Hemisynthesis of selected embelin analogs and investigation of their proapoptotic activity against cancer cells.

Viault G, Babu KS, Gautier F, Barillé-Nion S, Juin P, Tasseau O, Grée R. Viault G, et al. Among authors: gree r. Med Chem. 2013 Dec;9(8):1028-34. doi: 10.2174/1573406411309080003. Med Chem. 2013. PMID: 23373598

7

Design, synthesis and biological evaluation of new inhibitors of Bax/Bcl-xL interaction in cancer cells.

Vo DD, Gautier F, Barillé-Nion S, Juin P, Levoin N, Grée R. Vo DD, et al. Among authors: gree r. Bioorg Med Chem Lett. 2014 Apr 1;24(7):1758-61. doi: 10.1016/j.bmcl.2014.02.035. Epub 2014 Feb 24. Bioorg Med Chem Lett. 2014. PMID: 24602902

8

A combination of in silico and SAR studies to identify binding hot spots of Bcl-xL inhibitors.

Levoin N, Vo DD, Gautier F, Barillé-Nion S, Juin P, Tasseau O, Grée R. Levoin N, et al. Among authors: gree r. Bioorg Med Chem. 2015 Apr 15;23(8):1747-57. doi: 10.1016/j.bmc.2015.02.060. Epub 2015 Mar 6. Bioorg Med Chem. 2015. PMID: 25797160 Free article.

9

Targeting PUMA/Bcl-xL interaction by new specific compounds to unleash apoptotic process in cancer cells.

Ramana Murthy AV, Narendar V, Kumar NS, Aparna P, Durga Bhavani AK, Gautier F, Barillé-Nion S, Juin P, Mosset P, Grée R, Levoin N. Ramana Murthy AV, et al. Among authors: gree r. Eur J Med Chem. 2019 Jan 15;162:334-347. doi: 10.1016/j.ejmech.2018.10.069. Epub 2018 Nov 2. Eur J Med Chem. 2019. PMID: 30453244

10

Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase.

Brahmaiah D, Kanaka Durga Bhavani A, Aparna P, Sampath Kumar N, Solhi H, Le Guevel R, Baratte B, Ruchaud S, Bach S, Singh Jadav S, Raji Reddy C, Roisnel T, Mosset P, Levoin N, Grée R. Brahmaiah D, et al. Among authors: gree r. Bioorg Med Chem. 2021 Feb 1;31:115962. doi: 10.1016/j.bmc.2020.115962. Epub 2020 Dec 31. Bioorg Med Chem. 2021. PMID: 33422908

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