Di Santo R - Search Results

1

In vitro screening of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives as antiprotozoal agents and docking studies on Trypanosoma cruzi CYP51.

De Vita D, Moraca F, Zamperini C, Pandolfi F, Di Santo R, Matheeussen A, Maes L, Tortorella S, Scipione L. De Vita D, et al. Among authors: di santo r. Eur J Med Chem. 2016 May 4;113:28-33. doi: 10.1016/j.ejmech.2016.02.028. Epub 2016 Feb 15. Eur J Med Chem. 2016. PMID: 26922226

2

Antifungal agents. 9. 3-Aryl-4-[alpha-(1H-imidazol-1-yl)arylmethyl]pyrroles: a new class of potent anti-Candida agents.

Artico M, Di Santo R, Costi R, Massa S, Retico A, Artico M, Apuzzo G, Simonetti G, Strippoli V. Artico M, et al. Among authors: di santo r. J Med Chem. 1995 Oct 13;38(21):4223-33. doi: 10.1021/jm00021a011. J Med Chem. 1995. PMID: 7473549

3

Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling.

Artico M, Di Santo R, Costi R, Novellino E, Greco G, Massa S, Tramontano E, Marongiu ME, De Montis A, La Colla P. Artico M, et al. Among authors: di santo r. J Med Chem. 1998 Oct 8;41(21):3948-60. doi: 10.1021/jm9707232. J Med Chem. 1998. PMID: 9767632

4

Antifungal agents. 10. New derivatives of 1-[(aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-candida activity, and quantitative structure-analysis relationship studies.

Tafi A, Costi R, Botta M, Di Santo R, Corelli F, Massa S, Ciacci A, Manetti F, Artico M. Tafi A, et al. Among authors: di santo r. J Med Chem. 2002 Jun 20;45(13):2720-32. doi: 10.1021/jm011087h. J Med Chem. 2002. PMID: 12061875

5

Design, synthesis, and biological activities of pyrrolylethanoneamine derivatives, a novel class of monoamine oxidases inhibitors.

Di Santo R, Costi R, Roux A, Artico M, Befani O, Meninno T, Agostinelli E, Palmegiani P, Turini P, Cirilli R, Ferretti R, Gallinella B, La Torre F. Di Santo R, et al. J Med Chem. 2005 Jun 30;48(13):4220-3. doi: 10.1021/jm050172c. J Med Chem. 2005. PMID: 15974574

6

Antifungal agents. 11. N-substituted derivatives of 1-[(aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: synthesis, anti-Candida activity, and QSAR studies.

Di Santo R, Tafi A, Costi R, Botta M, Artico M, Corelli F, Forte M, Caporuscio F, Angiolella L, Palamara AT. Di Santo R, et al. J Med Chem. 2005 Aug 11;48(16):5140-53. doi: 10.1021/jm048997u. J Med Chem. 2005. PMID: 16078834

7

Simple but highly effective three-dimensional chemical-feature-based pharmacophore model for diketo acid derivatives as hepatitis C virus RNA-dependent RNA polymerase inhibitors.

Di Santo R, Fermeglia M, Ferrone M, Paneni MS, Costi R, Artico M, Roux A, Gabriele M, Tardif KD, Siddiqui A, Pricl S. Di Santo R, et al. J Med Chem. 2005 Oct 6;48(20):6304-14. doi: 10.1021/jm0504454. J Med Chem. 2005. PMID: 16190757 Free article.

8

Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action.

Di Santo R, Costi R, Roux A, Artico M, Lavecchia A, Marinelli L, Novellino E, Palmisano L, Andreotti M, Amici R, Galluzzo CM, Nencioni L, Palamara AT, Pommier Y, Marchand C. Di Santo R, et al. J Med Chem. 2006 Mar 23;49(6):1939-45. doi: 10.1021/jm0511583. J Med Chem. 2006. PMID: 16539381 Free PMC article.

9

Arylthiopyrrole (AThP) derivatives as non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis, structure-activity relationships, and docking studies (part 1).

Di Santo R, Costi R, Artico M, Miele G, Lavecchia A, Novellino E, Bergamini A, Cancio R, Maga G. Di Santo R, et al. ChemMedChem. 2006 Dec;1(12):1367-78. doi: 10.1002/cmdc.200600119. ChemMedChem. 2006. PMID: 17089433

10

Cinnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase.

Costi R, Di Santo R, Artico M, Miele G, Valentini P, Novellino E, Cereseto A. Costi R, et al. Among authors: di santo r. J Med Chem. 2007 Apr 19;50(8):1973-7. doi: 10.1021/jm060943s. Epub 2007 Mar 10. J Med Chem. 2007. PMID: 17348637

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