Slusarczyk M - Search Results

1

Anti-flavivirus Activity of Different Tritylated Pyrimidine and Purine Nucleoside Analogues.

McGuigan C, Serpi M, Slusarczyk M, Ferrari V, Pertusati F, Meneghesso S, Derudas M, Farleigh L, Zanetta P, Bugert J. McGuigan C, et al. Among authors: slusarczyk m. ChemistryOpen. 2016 Jan 21;5(3):227-35. doi: 10.1002/open.201500216. eCollection 2016 Jun. ChemistryOpen. 2016. PMID: 27551659 Free PMC article.

2

Synthetic Approaches for the Preparation of Phosphoramidate Prodrugs of 2'-Deoxypseudoisocytidine.

Serpi M, De Biasi R, Pertusati F, Slusarczyk M, McGuigan C. Serpi M, et al. Among authors: slusarczyk m. ChemistryOpen. 2017 May 5;6(3):424-436. doi: 10.1002/open.201700019. eCollection 2017 Jun. ChemistryOpen. 2017. PMID: 28638776 Free PMC article.

3

Symmetrical Diamidates as a Class of Phosphate Prodrugs to Deliver the 5'-Monophosphate Forms of Anticancer Nucleoside Analogues.

Slusarczyk M, Ferrari V, Serpi M, Gönczy B, Balzarini J, McGuigan C. Slusarczyk M, et al. ChemMedChem. 2018 Nov 6;13(21):2305-2316. doi: 10.1002/cmdc.201800504. ChemMedChem. 2018. PMID: 30199147

4

Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides.

McGuigan C, Bourdin C, Derudas M, Hamon N, Hinsinger K, Kandil S, Madela K, Meneghesso S, Pertusati F, Serpi M, Slusarczyk M, Chamberlain S, Kolykhalov A, Vernachio J, Vanpouille C, Introini A, Margolis L, Balzarini J. McGuigan C, et al. Among authors: slusarczyk m. Eur J Med Chem. 2013;70:326-40. doi: 10.1016/j.ejmech.2013.09.047. Epub 2013 Oct 9. Eur J Med Chem. 2013. PMID: 24177359 Free PMC article.

5

Synthesis and biological evaluation of phosphoramidate prodrugs of two analogues of 2-deoxy-d-ribose-1-phosphate directed to the discovery of two carbasugars as new potential anti-HIV leads.

Hamon N, Slusarczyk M, Serpi M, Balzarini J, McGuigan C. Hamon N, et al. Among authors: slusarczyk m. Bioorg Med Chem. 2015 Feb 15;23(4):829-38. doi: 10.1016/j.bmc.2014.12.039. Epub 2014 Dec 25. Bioorg Med Chem. 2015. PMID: 25616343 Free PMC article.

6

Synthesis and biological evaluation of 6-substituted-5-fluorouridine ProTides.

Slusarczyk M, Ferla S, Brancale A, McGuigan C. Slusarczyk M, et al. Bioorg Med Chem. 2018 Feb 1;26(3):551-565. doi: 10.1016/j.bmc.2017.11.037. Epub 2017 Dec 2. Bioorg Med Chem. 2018. PMID: 29277307 Free article.

7

Phosphoramidates and phosphonamidates (ProTides) with antiviral activity.

Slusarczyk M, Serpi M, Pertusati F. Slusarczyk M, et al. Antivir Chem Chemother. 2018 Jan-Dec;26:2040206618775243. doi: 10.1177/2040206618775243. Antivir Chem Chemother. 2018. PMID: 29792071 Free PMC article. Review.

8

Synthesis of phosphoramidate prodrugs: ProTide approach.

Serpi M, Madela K, Pertusati F, Slusarczyk M. Serpi M, et al. Among authors: slusarczyk m. Curr Protoc Nucleic Acid Chem. 2013 Jun;Chapter 15:15.5.1-15.5.15. doi: 10.1002/0471142700.nc1505s53. Curr Protoc Nucleic Acid Chem. 2013. PMID: 23775807

9

Phosphoramidate ProTides of the anticancer agent FUDR successfully deliver the preformed bioactive monophosphate in cells and confer advantage over the parent nucleoside.

McGuigan C, Murziani P, Slusarczyk M, Gonczy B, Vande Voorde J, Liekens S, Balzarini J. McGuigan C, et al. Among authors: slusarczyk m. J Med Chem. 2011 Oct 27;54(20):7247-58. doi: 10.1021/jm200815w. Epub 2011 Sep 27. J Med Chem. 2011. PMID: 21892829

10

Single Diastereomers of the Clinical Anticancer ProTide Agents NUC-1031 and NUC-3373 Preferentially Target Cancer Stem Cells In Vitro.

Slusarczyk M, Serpi M, Ghazaly E, Kariuki BM, McGuigan C, Pepper C. Slusarczyk M, et al. J Med Chem. 2021 Jun 24;64(12):8179-8193. doi: 10.1021/acs.jmedchem.0c02194. Epub 2021 Jun 4. J Med Chem. 2021. PMID: 34085825

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