Raub TJ - Search Results

1

QSAR Model of Unbound Brain-to-Plasma Partition Coefficient, K_p,uu,brain: Incorporating P-glycoprotein Efflux as a Variable.

Dolgikh E, Watson IA, Desai PV, Sawada GA, Morton S, Jones TM, Raub TJ. Dolgikh E, et al. Among authors: raub tj. J Chem Inf Model. 2016 Nov 28;56(11):2225-2233. doi: 10.1021/acs.jcim.6b00229. Epub 2016 Oct 13. J Chem Inf Model. 2016. PMID: 27684523

2

Integration of in silico and in vitro tools for scaffold optimization during drug discovery: predicting P-glycoprotein efflux.

Desai PV, Sawada GA, Watson IA, Raub TJ. Desai PV, et al. Among authors: raub tj. Mol Pharm. 2013 Apr 1;10(4):1249-61. doi: 10.1021/mp300555n. Epub 2013 Mar 1. Mol Pharm. 2013. PMID: 23363443

3

How hydrogen bonds impact P-glycoprotein transport and permeability.

Desai PV, Raub TJ, Blanco MJ. Desai PV, et al. Among authors: raub tj. Bioorg Med Chem Lett. 2012 Nov 1;22(21):6540-8. doi: 10.1016/j.bmcl.2012.08.059. Epub 2012 Aug 23. Bioorg Med Chem Lett. 2012. PMID: 23006604 Free article. Review.

4

Chalcogenopyrylium dyes as inhibitors/modulators of P-glycoprotein in multidrug-resistant cells.

Sawada GA, Raub TJ, William Higgins J, Brennan NK, Moore TM, Tombline G, Detty MR. Sawada GA, et al. Among authors: raub tj. Bioorg Med Chem. 2008 Nov 15;16(22):9745-56. doi: 10.1016/j.bmc.2008.09.065. Epub 2008 Sep 30. Bioorg Med Chem. 2008. PMID: 18849167

5

Breast cancer resistance protein interacts with various compounds in vitro, but plays a minor role in substrate efflux at the blood-brain barrier.

Zhao R, Raub TJ, Sawada GA, Kasper SC, Bacon JA, Bridges AS, Pollack GM. Zhao R, et al. Among authors: raub tj. Drug Metab Dispos. 2009 Jun;37(6):1251-8. doi: 10.1124/dmd.108.025064. Epub 2009 Mar 9. Drug Metab Dispos. 2009. PMID: 19273529 Free PMC article.

6

Brain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma Xenograft.

Raub TJ, Wishart GN, Kulanthaivel P, Staton BA, Ajamie RT, Sawada GA, Gelbert LM, Shannon HE, Sanchez-Martinez C, De Dios A. Raub TJ, et al. Drug Metab Dispos. 2015 Sep;43(9):1360-71. doi: 10.1124/dmd.114.062745. Epub 2015 Jul 6. Drug Metab Dispos. 2015. PMID: 26149830

7

Efficiency gains in tracer identification for nuclear imaging: can in vivo LC-MS/MS evaluation of small molecules screen for successful PET tracers?

Joshi EM, Need A, Schaus J, Chen Z, Benesh D, Mitch C, Morton S, Raub TJ, Phebus L, Barth V. Joshi EM, et al. Among authors: raub tj. ACS Chem Neurosci. 2014 Dec 17;5(12):1154-63. doi: 10.1021/cn500073j. Epub 2014 Oct 13. ACS Chem Neurosci. 2014. PMID: 25247893 Review.

8

In Silico and in Vitro Assessment of OATP1B1 Inhibition in Drug Discovery.

Danielson ML, Sawada GA, Raub TJ, Desai PV. Danielson ML, et al. Among authors: raub tj. Mol Pharm. 2018 Aug 6;15(8):3060-3068. doi: 10.1021/acs.molpharmaceut.8b00168. Epub 2018 Jul 5. Mol Pharm. 2018. PMID: 29927611

9

How well do lipophilicity parameters, MEEKC microemulsion capacity factor, and plasma protein binding predict CNS tissue binding?

Zamek-Gliszczynski MJ, Sprague KE, Espada A, Raub TJ, Morton SM, Manro JR, Molina-Martin M. Zamek-Gliszczynski MJ, et al. Among authors: raub tj. J Pharm Sci. 2012 May;101(5):1932-40. doi: 10.1002/jps.23081. Epub 2012 Feb 17. J Pharm Sci. 2012. PMID: 22344827

10

Expression of a widely distributed, novel sulfated membrane glycoprotein by bovine endothelia and certain transporting epithelia.

Raub TJ, Sawada GA, Kuentzel SL. Raub TJ, et al. J Histochem Cytochem. 1994 Sep;42(9):1237-50. doi: 10.1177/42.9.8064131. J Histochem Cytochem. 1994. PMID: 8064131

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