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Page 1
2,4-Diaminopyrimidine MK2 inhibitors. Part II: Structure-based inhibitor optimization.
Harris CM, Ericsson AM, Argiriadi MA, Barberis C, Borhani DW, Burchat A, Calderwood DJ, Cunha GA, Dixon RW, Frank KE, Johnson EF, Kamens J, Kwak S, Li B, Mullen KD, Perron DC, Wang L, Wishart N, Wu X, Zhang X, Zmetra TR, Talanian RV. Harris CM, et al. Among authors: burchat a. Bioorg Med Chem Lett. 2010 Jan 1;20(1):334-7. doi: 10.1016/j.bmcl.2009.10.103. Epub 2009 Oct 29. Bioorg Med Chem Lett. 2010. PMID: 19926477
Discovery of thienopyridines as Src-family selective Lck inhibitors.
Abbott L, Betschmann P, Burchat A, Calderwood DJ, Davis H, Hrnciar P, Hirst GC, Li B, Morytko M, Mullen K, Yang B. Abbott L, et al. Among authors: burchat a. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1167-71. doi: 10.1016/j.bmcl.2006.12.035. Epub 2006 Dec 15. Bioorg Med Chem Lett. 2007. PMID: 17234410
Enabling structure-based drug design of Tyk2 through co-crystallization with a stabilizing aminoindazole inhibitor.
Argiriadi MA, Goedken ER, Banach D, Borhani DW, Burchat A, Dixon RW, Marcotte D, Overmeyer G, Pivorunas V, Sadhukhan R, Sousa S, Moore NS, Tomlinson M, Voss J, Wang L, Wishart N, Woller K, Talanian RV. Argiriadi MA, et al. Among authors: burchat a. BMC Struct Biol. 2012 Sep 20;12:22. doi: 10.1186/1472-6807-12-22. BMC Struct Biol. 2012. PMID: 22995073 Free PMC article.
Thienopyrrole acetic acids as antagonists of the CRTH2 receptor.
Bonafoux D, Abibi A, Bettencourt B, Burchat A, Ericsson A, Harris CM, Kebede T, Morytko M, McPherson M, Wallace G, Wu X. Bonafoux D, et al. Among authors: burchat a. Bioorg Med Chem Lett. 2011 Mar 15;21(6):1861-4. doi: 10.1016/j.bmcl.2011.01.008. Epub 2011 Jan 14. Bioorg Med Chem Lett. 2011. PMID: 21316222
HTRF-based assay for microsomal prostaglandin E2 synthase-1 activity.
Goedken ER, Gagnon AI, Overmeyer GT, Liu J, Petrillo RA, Burchat AF, Tomlinson MJ. Goedken ER, et al. Among authors: burchat af. J Biomol Screen. 2008 Aug;13(7):619-25. doi: 10.1177/1087057108321145. Epub 2008 Jul 14. J Biomol Screen. 2008. PMID: 18626113